CN1142929C - 制备2-烷基-3-氨基噻吩衍生物的方法以及3-氨基噻吩衍生物 - Google Patents

制备2-烷基-3-氨基噻吩衍生物的方法以及3-氨基噻吩衍生物 Download PDF

Info

Publication number
CN1142929C
CN1142929C CNB001040979A CN00104097A CN1142929C CN 1142929 C CN1142929 C CN 1142929C CN B001040979 A CNB001040979 A CN B001040979A CN 00104097 A CN00104097 A CN 00104097A CN 1142929 C CN1142929 C CN 1142929C
Authority
CN
China
Prior art keywords
group
methyl
hydrogen atom
formula
halogen atom
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
CNB001040979A
Other languages
English (en)
Chinese (zh)
Other versions
CN1267671A (zh
Inventor
ʤ��ԣ֮
胜田裕之
����һ
石井圣一
冨谷完治
小高建次
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Mitsui Chemicals Inc
Original Assignee
Mitsui Chemicals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mitsui Chemicals Inc filed Critical Mitsui Chemicals Inc
Publication of CN1267671A publication Critical patent/CN1267671A/zh
Application granted granted Critical
Publication of CN1142929C publication Critical patent/CN1142929C/zh
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14Radicals substituted by singly bound hetero atoms other than halogen
    • C07D333/20Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D333/40Thiophene-2-carboxylic acid
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30Hetero atoms other than halogen
    • C07D333/36Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D411/00Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D411/02Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D411/12Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
CNB001040979A 1999-03-16 2000-03-16 制备2-烷基-3-氨基噻吩衍生物的方法以及3-氨基噻吩衍生物 Expired - Lifetime CN1142929C (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP6938799 1999-03-16
JP69387/1999 1999-03-16

Related Child Applications (1)

Application Number Title Priority Date Filing Date
CNB031241263A Division CN1224622C (zh) 1999-03-16 2000-03-16 制备2-烷基-3-氨基噻吩衍生物的方法以及3-氨基噻吩衍生物

Publications (2)

Publication Number Publication Date
CN1267671A CN1267671A (zh) 2000-09-27
CN1142929C true CN1142929C (zh) 2004-03-24

Family

ID=13401143

Family Applications (2)

Application Number Title Priority Date Filing Date
CNB001040979A Expired - Lifetime CN1142929C (zh) 1999-03-16 2000-03-16 制备2-烷基-3-氨基噻吩衍生物的方法以及3-氨基噻吩衍生物
CNB031241263A Expired - Lifetime CN1224622C (zh) 1999-03-16 2000-03-16 制备2-烷基-3-氨基噻吩衍生物的方法以及3-氨基噻吩衍生物

Family Applications After (1)

Application Number Title Priority Date Filing Date
CNB031241263A Expired - Lifetime CN1224622C (zh) 1999-03-16 2000-03-16 制备2-烷基-3-氨基噻吩衍生物的方法以及3-氨基噻吩衍生物

Country Status (12)

Country Link
US (3) US6239282B1 (https=)
EP (2) EP1559714B1 (https=)
KR (1) KR100439255B1 (https=)
CN (2) CN1142929C (https=)
AT (2) ATE383353T1 (https=)
BR (1) BR0001744B1 (https=)
DE (2) DE60037766T2 (https=)
DK (2) DK1036793T3 (https=)
ES (2) ES2298648T3 (https=)
HU (2) HU228563B1 (https=)
IL (2) IL153681A (https=)
IN (1) IN190570B (https=)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2271109T3 (es) 2000-11-08 2007-04-16 Syngenta Participations Ag Pirrocarboxamidas y pirrolcarbotioamidas y sus usos agroquimicos.
GB0101996D0 (en) 2001-01-25 2001-03-14 Syngenta Participations Ag Organtic compounds
WO2004009581A1 (ja) * 2002-07-24 2004-01-29 Mitsui Chemicals, Inc. 2−アルキル−3−アミノチオフェン誘導体の製造法
IN2004DE01799A (https=) 2003-10-23 2007-01-12 Bayer Cropscience Ag
JP2008527119A (ja) 2005-01-13 2008-07-24 シンベンション アーゲー 炭素ナノ粒子を含有する複合材料
US20070092282A1 (en) * 2005-10-26 2007-04-26 Hideya Takenoshita Image forming device
US8153823B2 (en) * 2006-04-17 2012-04-10 Mitsui Chemicals, Inc. 2-alkenyl-3-aminothiophene derivative and process for producing thereof
JP2008120710A (ja) * 2006-11-10 2008-05-29 Mitsui Chemicals Inc 2−アルキル−3−アミノチオフェン誘導体の製造方法
US20130231303A1 (en) 2010-11-15 2013-09-05 Bayer Intellectual Property Gmbh 5-halogenopyrazole(thio)carboxamides
CN111732493B (zh) * 2017-01-16 2023-01-24 宜昌尚诺德生物医药科技有限公司 一种芳胺化合物的合成工艺

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3933573A1 (de) * 1989-10-07 1991-04-18 Basf Ag Carbonsaeureamide, verfahren zu ihrer herstellung und ihre verwendung als herbizide
JPH05345780A (ja) * 1991-12-24 1993-12-27 Kumiai Chem Ind Co Ltd ピリミジンまたはトリアジン誘導体及び除草剤
DE69618370T2 (de) 1995-04-11 2002-09-26 Mitsui Chemicals, Inc. Substituierte Thiophenderivate und diese als aktiver Bestandteil enthaltenden Fungizide für Land- und Gartenbauwirtschaft
RU2111982C1 (ru) 1996-05-20 1998-05-27 Общественное объединение "Евразийское физическое общество" Способ получения вспениваемых кремнийорганических композиций
US5869427A (en) * 1996-06-11 1999-02-09 Mitsui Chemicals, Inc. Substituted thiophene derivative and plant disease control agent comprising the same as active ingredient

Also Published As

Publication number Publication date
US6331634B1 (en) 2001-12-18
ATE304004T1 (de) 2005-09-15
US20010023295A1 (en) 2001-09-20
CN1267671A (zh) 2000-09-27
CN1495180A (zh) 2004-05-12
DE60022416T2 (de) 2006-06-29
EP1036793A3 (en) 2001-02-28
HU228563B1 (hu) 2013-04-29
US6331639B2 (en) 2001-12-18
ES2247968T3 (es) 2006-03-16
ES2298648T3 (es) 2008-05-16
IL153681A (en) 2006-08-20
ATE383353T1 (de) 2008-01-15
HUP0001129A3 (en) 2002-03-28
BR0001744B1 (pt) 2011-08-23
DE60037766D1 (de) 2008-02-21
EP1036793B1 (en) 2005-09-07
HU0001129D0 (en) 2000-05-28
US6239282B1 (en) 2001-05-29
KR100439255B1 (ko) 2004-07-05
EP1036793A2 (en) 2000-09-20
DE60037766T2 (de) 2009-01-15
BR0001744A (pt) 2000-10-31
DK1559714T3 (da) 2008-03-25
KR20010006815A (ko) 2001-01-26
IN190570B (https=) 2003-08-09
HUP0001129A2 (hu) 2001-01-29
CN1224622C (zh) 2005-10-26
DK1036793T3 (da) 2005-10-03
EP1559714B1 (en) 2008-01-09
IL134788A0 (en) 2001-04-30
DE60022416D1 (de) 2005-10-13
EP1559714A1 (en) 2005-08-03
HUS1600015I1 (hu) 2016-05-30

Similar Documents

Publication Publication Date Title
CN1053666C (zh) 苯并杂环化合物或其药用盐的制备方法
CN1040322C (zh) 嘧啶化合物
CN1136213C (zh) 新的苯并噻吩、苯并呋喃和吲哚化合物、其制备方法和含有它们的药物组合物
CN1221417A (zh) 具有抗糖尿病、降低血脂、抗高血压性能的噻唑烷二酮化合物,其制备方法及其药物组合物
CN1753884A (zh) 阿片类受体拮抗剂
CN1173497A (zh) 含杂环碳酸衍生物
CN1835923A (zh) 制备4-氨基-3-喹啉腈的方法
CN1062726A (zh) N-甲酰苯胺类杀节肢动物剂
CN1142929C (zh) 制备2-烷基-3-氨基噻吩衍生物的方法以及3-氨基噻吩衍生物
CN1042133C (zh) N-取代的氮杂双环庚烷衍生物及其用途
CN87103504A (zh) 杂环羧酰胺
CN1295563A (zh) 用作毒蕈碱性受体拮抗剂的2-芳基乙基-(哌啶-4-基甲基)胺衍生物
CN1332727A (zh) 3,3-二芳基哌啶和2,2-二芳基吗啉衍生物
CN1052478C (zh) 1,4-二取代-5(4h)-四唑啉酮类的制备方法
CN1821217A (zh) 反式-4-氨基-1-环己烷羧酸衍生物的制备方法
CN1440385A (zh) 用于治疗艾滋病的吡咯衍生物
CN87107226A (zh) 内酰胺衍生物及其制备
CN1245169A (zh) 新的硝酮化合物,其制备方法以及含有它们的药物组合物
CN1852907A (zh) 2-氨基-5-苯甲酰基噻唑npy拮抗剂
CN1798726A (zh) 取代吲哚及一种制备取代吲哚的方法
CN1218941C (zh) 乙磺酰哌啶衍生物的制备方法
CN1040105C (zh) 制备氨基酮衍生物的方法
CN1950362A (zh) 类胰蛋白酶抑制剂的制备方法
CN1173977C (zh) 制备噻吩并嘧啶衍生物的方法
CN1249043C (zh) 新的杂环化合物,其制备方法以及含有它们的药物组合物

Legal Events

Date Code Title Description
C10 Entry into substantive examination
SE01 Entry into force of request for substantive examination
C06 Publication
PB01 Publication
C14 Grant of patent or utility model
GR01 Patent grant
REG Reference to a national code

Ref country code: HK

Ref legal event code: GR

Ref document number: 1072095

Country of ref document: HK

CX01 Expiry of patent term

Granted publication date: 20040324

CX01 Expiry of patent term