CN1142817A - 1n-烷基-n-芳基嘧啶胺及其衍生物 - Google Patents
1n-烷基-n-芳基嘧啶胺及其衍生物 Download PDFInfo
- Publication number
- CN1142817A CN1142817A CN94194465A CN94194465A CN1142817A CN 1142817 A CN1142817 A CN 1142817A CN 94194465 A CN94194465 A CN 94194465A CN 94194465 A CN94194465 A CN 94194465A CN 1142817 A CN1142817 A CN 1142817A
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- alkyl
- methyl
- ethyl
- bromo
- phenyl
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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- Chemical & Material Sciences (AREA)
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- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
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- Neurology (AREA)
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- Immunology (AREA)
- Addiction (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Pain & Pain Management (AREA)
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- Obesity (AREA)
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- Child & Adolescent Psychology (AREA)
- Toxicology (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US13420993A | 1993-10-12 | 1993-10-12 | |
| US08/134,209 | 1993-10-12 | ||
| US29727494A | 1994-08-26 | 1994-08-26 | |
| US08/297,274 | 1994-08-26 | ||
| US08/315,660 | 1994-09-29 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN1142817A true CN1142817A (zh) | 1997-02-12 |
Family
ID=26832075
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN94194465A Pending CN1142817A (zh) | 1993-10-12 | 1994-10-06 | 1n-烷基-n-芳基嘧啶胺及其衍生物 |
Country Status (6)
| Country | Link |
|---|---|
| JP (1) | JP3398152B2 (enExample) |
| CN (1) | CN1142817A (enExample) |
| FI (1) | FI961599A7 (enExample) |
| RU (1) | RU2153494C2 (enExample) |
| TW (1) | TW286316B (enExample) |
| WO (1) | WO1995010506A1 (enExample) |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1925859B (zh) * | 2004-03-02 | 2010-11-24 | 弗·哈夫曼-拉罗切有限公司 | 用于治疗焦虑、抑郁和癫痫的作为gaba受体配体的4-(硫基-嘧啶-4-基甲基)-吗啉衍生物和相关的化合物 |
| CN1926117B (zh) * | 2004-01-14 | 2011-12-07 | 泊灵格英格尔海姆国际有限公司 | 用于改进感知、注意力、学习效率、和/或记忆力的6-氨基-5-氰基-嘧啶-4-酮类化合物 |
| CN107573333A (zh) * | 2013-04-10 | 2018-01-12 | 江苏恒瑞医药股份有限公司 | 替格瑞洛的中间体及其制备方法和替格瑞洛的制备方法 |
Families Citing this family (112)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
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| CN1926117B (zh) * | 2004-01-14 | 2011-12-07 | 泊灵格英格尔海姆国际有限公司 | 用于改进感知、注意力、学习效率、和/或记忆力的6-氨基-5-氰基-嘧啶-4-酮类化合物 |
| CN102382063A (zh) * | 2004-01-14 | 2012-03-21 | 泊灵格英格尔海姆国际有限公司 | 用于改进感知、注意力、学习效率、和/或记忆力的6-氨基-5-氰基-嘧啶-4-酮类化合物 |
| CN1925859B (zh) * | 2004-03-02 | 2010-11-24 | 弗·哈夫曼-拉罗切有限公司 | 用于治疗焦虑、抑郁和癫痫的作为gaba受体配体的4-(硫基-嘧啶-4-基甲基)-吗啉衍生物和相关的化合物 |
| CN107573333A (zh) * | 2013-04-10 | 2018-01-12 | 江苏恒瑞医药股份有限公司 | 替格瑞洛的中间体及其制备方法和替格瑞洛的制备方法 |
| CN107573333B (zh) * | 2013-04-10 | 2019-10-18 | 江苏恒瑞医药股份有限公司 | 替格瑞洛的中间体及其制备方法和替格瑞洛的制备方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| FI961599A7 (fi) | 1996-06-07 |
| TW286316B (enExample) | 1996-09-21 |
| RU2153494C2 (ru) | 2000-07-27 |
| JP3398152B2 (ja) | 2003-04-21 |
| JPH09504520A (ja) | 1997-05-06 |
| FI961599A0 (fi) | 1996-04-11 |
| WO1995010506A1 (en) | 1995-04-20 |
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