CN108026045B - 用作RORγ调节剂的经过取代的四氢喹啉酮化合物 - Google Patents

用作RORγ调节剂的经过取代的四氢喹啉酮化合物 Download PDF

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CN108026045B
CN108026045B CN201680036585.XA CN201680036585A CN108026045B CN 108026045 B CN108026045 B CN 108026045B CN 201680036585 A CN201680036585 A CN 201680036585A CN 108026045 B CN108026045 B CN 108026045B
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compound
pharmaceutically acceptable
stereoisomer
mmol
acceptable salt
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CN108026045A (zh
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拉维·科特劳巴塞阿乌伊娜玛诺达
凯坦·潘迪特
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Aurigene Oncology Ltd
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Aurigene Discovery Technologies Ltd
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CN201680036585.XA 2015-05-15 2016-05-13 用作RORγ调节剂的经过取代的四氢喹啉酮化合物 Active CN108026045B (zh)

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IN2448/CHE/2015 2015-05-15
IN2448CH2015 2015-05-15
PCT/IB2016/052773 WO2016185342A1 (en) 2015-05-15 2016-05-13 Substituted tetrahydroquinolinone compounds as ror gamma modulators

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JP6448867B2 (ja) 2015-12-15 2019-01-09 アストラゼネカ・アクチエボラーグＡｓｔｒａｚｅｎｅｃａ Ａｋｔｉｅｂｏｌａｇ イソインドール化合物
TWI705958B (zh) 2016-12-05 2020-10-01 荷蘭商領導醫藥控股責任有限公司 ＲＯＲγ調節子
CN108218845B (zh) * 2016-12-21 2022-11-29 江苏柯菲平医药股份有限公司 一类色满-6-磺酰胺RORγ调节剂及其用途
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CN113121463A (zh) * 2019-12-31 2021-07-16 广东东阳光药业有限公司 具有双环结构的酰胺类化合物及其在药物中的应用
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