CN102727458B - 涂层组合物、涂布有该涂层组合物的固体制剂以及制备该固体制剂的方法 - Google Patents
涂层组合物、涂布有该涂层组合物的固体制剂以及制备该固体制剂的方法 Download PDFInfo
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A61K31/525—Isoalloxazines, e.g. riboflavins, vitamin B2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/02—Nutrients, e.g. vitamins, minerals
-
- C—CHEMISTRY; METALLURGY
- C09—DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
- C09D—COATING COMPOSITIONS, e.g. PAINTS, VARNISHES OR LACQUERS; FILLING PASTES; CHEMICAL PAINT OR INK REMOVERS; INKS; CORRECTING FLUIDS; WOODSTAINS; PASTES OR SOLIDS FOR COLOURING OR PRINTING; USE OF MATERIALS THEREFOR
- C09D101/00—Coating compositions based on cellulose, modified cellulose, or cellulose derivatives
- C09D101/08—Cellulose derivatives
- C09D101/26—Cellulose ethers
- C09D101/28—Alkyl ethers
- C09D101/284—Alkyl ethers with hydroxylated hydrocarbon radicals
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- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
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- Veterinary Medicine (AREA)
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- Epidemiology (AREA)
- Materials Engineering (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
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- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Nutrition Science (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| JP5836980B2 (ja) | 2013-01-11 | 2015-12-24 | 信越化学工業株式会社 | 薬物含有粒子、固形製剤及び薬物含有粒子の製造方法 |
| JP6267239B2 (ja) * | 2013-03-07 | 2018-01-24 | ダウ グローバル テクノロジーズ エルエルシー | 極めて低粘度の新規エステル化セルロースエーテル |
| US10646573B2 (en) * | 2013-06-03 | 2020-05-12 | Shin-Etsu Chemical Co., Ltd. | Composition for hot melt extrusion and method for producing hot melt extrudate by using same |
| JP6203702B2 (ja) * | 2014-11-18 | 2017-09-27 | 信越化学工業株式会社 | ヒプロメロース酢酸エステルコハク酸エステルを用いたスプレードライ用溶液及び固体分散体の製造方法 |
| BR112018010354A2 (pt) * | 2015-12-08 | 2018-12-04 | Dow Global Technologies Llc | composições compreendendo éteres de celulose e éteres de celulose esterificados solúveis em água |
| US9884922B2 (en) * | 2016-03-11 | 2018-02-06 | Shin-Etsu Chemical Co., Ltd. | Hypromellose acetate succinate, method for producing the same and composition containing the same |
| CN106138003A (zh) * | 2016-07-11 | 2016-11-23 | 成都中牧生物药业有限公司 | 一种稳定型薄膜包衣预混剂及制备方法 |
| CN105999286A (zh) * | 2016-07-11 | 2016-10-12 | 成都中牧生物药业有限公司 | 一种防潮薄膜包衣预混剂及制备方法 |
| CN106075461A (zh) * | 2016-07-11 | 2016-11-09 | 成都中牧生物药业有限公司 | 一种遮盖异味的薄膜包衣预混剂及制备方法 |
| JP7050714B2 (ja) * | 2019-04-04 | 2022-04-08 | 信越化学工業株式会社 | 腸溶性コーティング用組成物及び固形製剤の製造方法 |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| JPS62120315A (ja) * | 1985-11-20 | 1987-06-01 | Shin Etsu Chem Co Ltd | 経口投与型徐放性錠剤の製造方法 |
| US4789549A (en) * | 1987-03-09 | 1988-12-06 | Warner-Lambert Company | Sustained release dosage forms |
| CA2007181C (en) * | 1989-01-06 | 1998-11-24 | Angelo Mario Morella | Sustained release pharmaceutical composition |
| JPH04202124A (ja) * | 1990-11-29 | 1992-07-22 | Fuji Kagaku Kogyo Kk | 噴霧乾燥造粒法による薬物放出の制御された製剤の製造法 |
| JPH08143476A (ja) | 1994-11-18 | 1996-06-04 | Japan Tobacco Inc | 薬物放出制御膜及び固形製剤 |
| JP2000128779A (ja) | 1998-10-20 | 2000-05-09 | Mitsui Chemicals Inc | 薬物放出制御型製剤 |
| JP4181738B2 (ja) * | 2000-08-25 | 2008-11-19 | 信越化学工業株式会社 | 腸溶性コーティング製剤の製造方法 |
| AU2003284942A1 (en) | 2002-10-30 | 2004-06-07 | Pharmacia Corporation | Oral extended release tablets and methods of making and using the same |
| DE60309565T3 (de) * | 2003-05-02 | 2015-01-15 | Dexcel Ltd. | Tablettenzubereitung mit verlängerter Freisetzung von Venlafaxin |
| US7294347B2 (en) * | 2004-06-21 | 2007-11-13 | Council Of Scientific And Industrial Research | Coating compositions for bitterness inhibition |
| GB0517205D0 (en) * | 2005-08-22 | 2005-09-28 | Novartis Ag | Organic compounds |
| KR100888131B1 (ko) | 2006-10-10 | 2009-03-11 | 한올제약주식회사 | 시간차 투약 원리를 이용한 심혈관계 질환 치료용 복합제제 |
| JP2009191034A (ja) | 2008-02-15 | 2009-08-27 | Ss Pharmaceut Co Ltd | 時限放出製剤 |
| EP2281557A4 (en) * | 2008-04-29 | 2011-08-31 | Hanall Biopharma Co Ltd | PHARMACEUTICAL FORMULATION CONTAINING AN ANGIOTENSIN II RECEPTOR BLOCKING AGENT |
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- 2012-03-28 JP JP2012073410A patent/JP5667113B2/ja active Active
- 2012-03-29 CN CN201210087493.8A patent/CN102727458B/zh active Active
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| CN101917978A (zh) * | 2007-11-08 | 2010-12-15 | 葛兰素集团有限公司 | 药物制剂 |
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| JP2012214461A (ja) | 2012-11-08 |
| CN102727458A (zh) | 2012-10-17 |
| EP2510923A1 (en) | 2012-10-17 |
| US20120251588A1 (en) | 2012-10-04 |
| JP5667113B2 (ja) | 2015-02-12 |
| IN2012DE00868A (enExample) | 2015-09-04 |
| EP2510923B1 (en) | 2014-12-31 |
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