CN1019972C - 制备5，6-二羟基吲哚及其3-烷基衍生物和中间体化合物的方法 - Google Patents

制备5，6-二羟基吲哚及其3-烷基衍生物和中间体化合物的方法 Download PDF

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Publication number
CN1019972C
CN1019972C CN87107372A CN87107372A CN1019972C CN 1019972 C CN1019972 C CN 1019972C CN 87107372 A CN87107372 A CN 87107372A CN 87107372 A CN87107372 A CN 87107372A CN 1019972 C CN1019972 C CN 1019972C
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China
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formula
compound
hydrogen
reaction
benzyl
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Expired - Fee Related
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CN87107372A
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English (en)
Chinese (zh)
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CN87107372A (zh
Inventor
阿莱克斯·米尼诺
简·扎奎斯·万单伯斯彻
格拉德·兰格
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LOreal SA
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LOreal SA
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/32—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring
    • C07C255/37—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by etherified hydroxy groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/32—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring
    • C07C255/42—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being further bound to other hetero atoms
    • C07C255/43—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being further bound to other hetero atoms the carbon skeleton being further substituted by singly-bound oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A61K8/4906—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom
    • A61K8/4913—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom having five membered rings, e.g. pyrrolidone carboxylic acid
    • A61K8/492—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom having five membered rings, e.g. pyrrolidone carboxylic acid having condensed rings, e.g. indol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q5/00—Preparations for care of the hair
    • A61Q5/10—Preparations for permanently dyeing the hair
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/32—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring
    • C07C255/36—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by hydroxy groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
    • D—TEXTILES; PAPER
    • D06—TREATMENT OF TEXTILES OR THE LIKE; LAUNDERING; FLEXIBLE MATERIALS NOT OTHERWISE PROVIDED FOR
    • D06P—DYEING OR PRINTING TEXTILES; DYEING LEATHER, FURS OR SOLID MACROMOLECULAR SUBSTANCES IN ANY FORM
    • D06P3/00—Special processes of dyeing or printing textiles, or dyeing leather, furs, or solid macromolecular substances in any form, classified according to the material treated
    • D06P3/02—Material containing basic nitrogen
    • D06P3/04—Material containing basic nitrogen containing amide groups
    • D06P3/08—Material containing basic nitrogen containing amide groups using oxidation dyes
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10T—TECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
    • Y10T428/00—Stock material or miscellaneous articles
    • Y10T428/14—Layer or component removable to expose adhesive
    • Y10T428/1476—Release layer

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Birds (AREA)
  • Epidemiology (AREA)
  • Textile Engineering (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Coloring (AREA)
  • Catalysts (AREA)
  • Cosmetics (AREA)
CN87107372A 1986-11-07 1987-11-06 制备5，6-二羟基吲哚及其3-烷基衍生物和中间体化合物的方法 Expired - Fee Related CN1019972C (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US92772386A 1986-11-07 1986-11-07
US927.723 1986-11-07

Publications (2)

Publication Number Publication Date
CN87107372A CN87107372A (zh) 1988-08-03
CN1019972C true CN1019972C (zh) 1993-03-03

Family

ID=25455154

Family Applications (1)

Application Number Title Priority Date Filing Date
CN87107372A Expired - Fee Related CN1019972C (zh) 1986-11-07 1987-11-06 制备5，6-二羟基吲哚及其3-烷基衍生物和中间体化合物的方法

Country Status (20)

Country Link
US (4) US5410067A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
JP (1) JP2553108B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
KR (1) KR970002746B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CN (1) CN1019972C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AR (1) AR245695A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AT (1) AT390950B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AU (1) AU604780B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BE (1) BE1000762A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BR (1) BR8705980A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (2) CA1300633C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CH (2) CH676845A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DE (1) DE3737825A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ES (1) ES2007747A6 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FR (1) FR2606405B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GB (1) GB2198128B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GR (1) GR871701B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IT (1) IT1211506B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NL (1) NL8702660A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PT (1) PT86088B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ZA (1) ZA878313B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GR871701B (en) * 1986-11-07 1988-03-04 Oreal Method for preparing 5,6 - dihydrixyindol, and its 3 - alkylated derivative and intermediates
US5283352A (en) * 1986-11-28 1994-02-01 Orion-Yhtyma Oy Pharmacologically active compounds, methods for the preparation thereof and compositions containing the same
YU213587A (en) * 1986-11-28 1989-06-30 Orion Yhtymae Oy Process for obtaining new pharmacologic active cateholic derivatives
FI864875A0 (fi) * 1986-11-28 1986-11-28 Orion Yhtymae Oy Nya farmakologiskt aktiva foereningar, dessa innehaollande kompositioner samt foerfarande och mellanprodukter foer anvaendning vid framstaellning av dessa.
US5489614A (en) * 1987-11-27 1996-02-06 Orion-Yhtyma Oy Catechol derivatives, their physiologically acceptable salts, esters and use
DE4204089A1 (de) * 1992-02-12 1993-08-19 Henkel Kgaa Synthese von indolen durch dehydrierung von indolinen
US5262546A (en) * 1992-11-17 1993-11-16 Clairol, Inc. Process for the preparation of 5,6-diacetoxyindole
FR2742162B1 (fr) 1995-12-06 1998-01-16 Oreal Procede de preparation de composes indoliques
US6160127A (en) * 1998-07-15 2000-12-12 Bristol-Myers Squibb Company Process for the preparation of substituted indoles
CA2341711A1 (en) * 1998-08-28 2000-03-09 Smithkline Beecham Corporation Process for making 2-amino-5-cyanophenol
US6384263B1 (en) * 2000-08-04 2002-05-07 E. I. Du Pont De Nemours And Company Process for making 3-hydroxyalkanelnitriles and conversion of the 3-hydroxyalkanelnitrile to an hydroxyaminoalkane
CN102976957A (zh) * 2012-11-30 2013-03-20 四川大学 一种制备4-氨基邻苯二酚的方法
CN103073495B (zh) * 2013-02-06 2015-08-05 苏州立新制药有限公司 一种ent-3-甲氧基吗喃的制备方法
CN111247124B (zh) * 2017-11-01 2023-10-13 花王株式会社 二羟基吲哚类化合物的制造方法
CN114805126B (zh) * 2022-05-03 2024-06-18 浙江荣耀生物科技股份有限公司 2-硝基-4,5-二苄氧基苯乙腈的制备方法

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT199319B (de) * 1955-07-29 1958-08-25 Oreal Mittel zum Färben von keratinhaltigen Fasern, insbesondere von menschlichem Haar
NL254075A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * 1959-07-24
US3370063A (en) * 1964-10-05 1968-02-20 Mcneilab Inc Substituted dimethoxy indoles and method of making the same
US3976695A (en) * 1970-01-13 1976-08-24 Smithkline Corporation Halogen substituted α-(aminoalkyl)-3,4-dihydroxybenzyl alcohols
US3995041A (en) * 1975-10-30 1976-11-30 Miles Laboratories, Inc. Derivatives of 2-substituted-hydroxyanilino-hexahydro-2H-benzo[α]quinolizines
DE2604838A1 (de) * 1976-02-07 1977-08-11 Knoll Ag Alkylendioxypiperazinderivate
JPS5562061A (en) * 1978-10-31 1980-05-10 Ihara Chem Ind Co Ltd Production of indoles
JPS5576859A (en) * 1978-12-01 1980-06-10 Fujimoto Seiyaku Kk Novel preparation of 4-hydroxyindole
CA1201067A (en) * 1982-12-07 1986-02-25 Keith Brown Hair dyeing process and composition
ES532455A0 (es) * 1983-05-13 1985-06-16 Yamanouchi Pharma Co Ltd Un procedimiento para la produccion de un derivado de catecol
LU86256A1 (fr) * 1986-01-20 1988-01-20 Oreal Procede de teinture des fibres keratiniques avec du 5,6-dihydroxyindole associe avec un iodure
LU86314A1 (fr) * 1986-02-20 1987-09-10 Oreal Procede de teinture des fibres keratiniques humaines avec le 5,6-dihydroxyindole et un anion metallique
GR871701B (en) * 1986-11-07 1988-03-04 Oreal Method for preparing 5,6 - dihydrixyindol, and its 3 - alkylated derivative and intermediates
DE3642331A1 (de) * 1986-12-11 1988-06-23 Basf Ag Basisch substituierte phenylacetonitrile, ihre herstellung und diese enthaltende arzneimittel

Also Published As

Publication number Publication date
AU604780B2 (en) 1991-01-03
IT1211506B (it) 1989-11-03
ATA294087A (de) 1990-01-15
AU8087087A (en) 1988-06-02
CA1300643C (fr) 1992-05-12
GB2198128B (en) 1990-11-07
JP2553108B2 (ja) 1996-11-13
DE3737825C2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1990-05-31
IT8767951A0 (it) 1987-11-06
US5508464A (en) 1996-04-16
ES2007747A6 (es) 1989-07-01
US5410067A (en) 1995-04-25
AT390950B (de) 1990-07-25
PT86088A (fr) 1987-12-01
AR245695A1 (es) 1994-02-28
CH679150A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1991-12-31
CN87107372A (zh) 1988-08-03
CA1300633C (fr) 1992-05-12
FR2606405A1 (fr) 1988-05-13
GB2198128A (en) 1988-06-08
FR2606405B1 (fr) 1995-06-23
GR871701B (en) 1988-03-04
KR880006168A (ko) 1988-07-21
BR8705980A (pt) 1988-06-14
CH676845A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1991-03-15
US5536865A (en) 1996-07-16
PT86088B (pt) 1990-11-20
US5498746A (en) 1996-03-12
JPS63135365A (ja) 1988-06-07
GB8726173D0 (en) 1987-12-16
KR970002746B1 (en) 1997-03-10
NL8702660A (nl) 1988-06-01
BE1000762A5 (fr) 1989-03-28
DE3737825A1 (de) 1988-05-19
ZA878313B (en) 1989-07-26

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