CN101500570A - 新型带式制剂 - Google Patents
新型带式制剂 Download PDFInfo
- Publication number
- CN101500570A CN101500570A CNA2007800296920A CN200780029692A CN101500570A CN 101500570 A CN101500570 A CN 101500570A CN A2007800296920 A CNA2007800296920 A CN A2007800296920A CN 200780029692 A CN200780029692 A CN 200780029692A CN 101500570 A CN101500570 A CN 101500570A
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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- A—HUMAN NECESSITIES
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- A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
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- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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- A—HUMAN NECESSITIES
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Abstract
Description
经口给药(文献1) | 本发明实施例1的带式制剂 | |
N-氧化物形式/化合物A | 0.40 | 0.029 |
N-去乙基形式/化合物A | 0.10 | 0.043 |
渗透促进剂(在粘合剂层中的含量:重量%) | |
实施例7 | 月桂醇(10) |
实施例8 | 癸醇(10) |
实施例9 | 己二酸二异丙酯(10) |
实施例10 | 中链脂肪酸甘油三酯(10) |
实施例11 | 丙二醇(10) |
实施例12 | 油酸(10) |
实施例13 | 克罗米通(10) |
实施例14 | N-甲基-2-吡咯烷酮(NMP)(10) |
实施例15 | 橄榄油(10) |
实施例16 | 大豆油(10) |
实施例17 | 肉豆蔻酸(10) |
实施例18 | 甘油(10) |
实施例19 | 聚乙二醇200(10) |
实施例20 | 角鲨烷(10) |
实施例21 | 液态石蜡(10) |
实施例22 | 聚氧乙烯(160)聚氧丙烯(40)二醇(10) |
实施例23 | 聚氧乙烯-壬基苯基醚(10) |
实施例24 | 聚桂醇(10) |
实施例25 | α-单异硬脂基甘油醚(10) |
实施例26 | 聚氧乙烯氢化蓖麻油10(10) |
实施例27 | 肉豆蔻酸异丙酯(10) |
实施例28 | 癸二酸二乙酯(10) |
实施例29 | 失水山梨醇倍半油酸酯(10) |
实施例30 | 聚氧乙烯(40)硬脂酸酯(10) |
实施例31 | 单月桂酸聚乙二醇酯(10) |
实施例32 | 十六醇·聚乙二醇单硬脂酸酯混合蜡(10) |
实施例33 | 液态羊毛脂(10) |
实施例34 | 乳酸(10) |
实施例35 | 乙酸(10) |
实施例36 | 乳酸十六酯(10) |
实施例37 | 油酸油酯(10) |
实施例38 | 2-乙基己酸十六酯(10) |
实施例39 | 乙酸正丁酯(10) |
实施例40 | 1-薄荷醇(10) |
实施例41 | 甲基异丁基酮(10) |
实施例42 | 三乙酸甘油酯(10) |
Claims (8)
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2006161072 | 2006-06-09 | ||
JP161072/2006 | 2006-06-09 | ||
JP232926/2006 | 2006-08-30 | ||
JP2006232926 | 2006-08-30 | ||
PCT/JP2007/061538 WO2007142295A1 (ja) | 2006-06-09 | 2007-06-07 | 新規テープ製剤 |
Publications (2)
Publication Number | Publication Date |
---|---|
CN101500570A true CN101500570A (zh) | 2009-08-05 |
CN101500570B CN101500570B (zh) | 2012-07-04 |
Family
ID=38801541
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CN2007800296920A Active CN101500570B (zh) | 2006-06-09 | 2007-06-07 | 贴剂 |
Country Status (13)
Country | Link |
---|---|
US (1) | US8354121B2 (zh) |
EP (1) | EP2036559B1 (zh) |
JP (1) | JP5001271B2 (zh) |
KR (1) | KR101390012B1 (zh) |
CN (1) | CN101500570B (zh) |
AU (1) | AU2007255724B2 (zh) |
BR (1) | BRPI0713104A2 (zh) |
CA (1) | CA2653827C (zh) |
ES (1) | ES2456328T3 (zh) |
HK (1) | HK1137344A1 (zh) |
MX (1) | MX2008015794A (zh) |
RU (1) | RU2445959C2 (zh) |
WO (1) | WO2007142295A1 (zh) |
Cited By (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2012105715A1 (en) * | 2011-02-02 | 2012-08-09 | Dainippon Sumitomo Pharma Co., Ltd. | Novel external preparation |
CN103338771A (zh) * | 2011-02-02 | 2013-10-02 | 日东电工株式会社 | 贴剂 |
CN103347522A (zh) * | 2011-02-02 | 2013-10-09 | 大日本住友制药株式会社 | 透皮贴剂 |
CN103347541A (zh) * | 2011-02-02 | 2013-10-09 | 日东电工株式会社 | 贴片制剂的制造方法 |
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-
2007
- 2007-06-07 AU AU2007255724A patent/AU2007255724B2/en not_active Ceased
- 2007-06-07 MX MX2008015794A patent/MX2008015794A/es active IP Right Grant
- 2007-06-07 WO PCT/JP2007/061538 patent/WO2007142295A1/ja active Application Filing
- 2007-06-07 RU RU2008152758/15A patent/RU2445959C2/ru not_active IP Right Cessation
- 2007-06-07 US US12/308,099 patent/US8354121B2/en not_active Expired - Fee Related
- 2007-06-07 KR KR1020097000298A patent/KR101390012B1/ko active IP Right Grant
- 2007-06-07 CN CN2007800296920A patent/CN101500570B/zh active Active
- 2007-06-07 CA CA2653827A patent/CA2653827C/en not_active Expired - Fee Related
- 2007-06-07 JP JP2008520617A patent/JP5001271B2/ja active Active
- 2007-06-07 ES ES07744868.6T patent/ES2456328T3/es active Active
- 2007-06-07 BR BRPI0713104-6A patent/BRPI0713104A2/pt not_active IP Right Cessation
- 2007-06-07 EP EP07744868.6A patent/EP2036559B1/en not_active Not-in-force
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2010
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Cited By (7)
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WO2012105715A1 (en) * | 2011-02-02 | 2012-08-09 | Dainippon Sumitomo Pharma Co., Ltd. | Novel external preparation |
CN103338771A (zh) * | 2011-02-02 | 2013-10-02 | 日东电工株式会社 | 贴剂 |
CN103347522A (zh) * | 2011-02-02 | 2013-10-09 | 大日本住友制药株式会社 | 透皮贴剂 |
CN103347541A (zh) * | 2011-02-02 | 2013-10-09 | 日东电工株式会社 | 贴片制剂的制造方法 |
CN103347522B (zh) * | 2011-02-02 | 2015-09-02 | 大日本住友制药株式会社 | 透皮贴剂 |
CN109516953A (zh) * | 2017-09-18 | 2019-03-26 | 北京万全德众医药生物技术有限公司 | 布南色林工艺杂质的制备 |
CN115605206A (zh) * | 2020-05-14 | 2023-01-13 | 株式会社钟化(Jp) | 含布南色林贴剂及其制造方法 |
Also Published As
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CA2653827A1 (en) | 2007-12-13 |
RU2445959C2 (ru) | 2012-03-27 |
HK1137344A1 (en) | 2010-07-30 |
KR101390012B1 (ko) | 2014-04-29 |
MX2008015794A (es) | 2009-01-12 |
EP2036559B1 (en) | 2014-03-19 |
EP2036559A1 (en) | 2009-03-18 |
KR20090031407A (ko) | 2009-03-25 |
US20090169605A1 (en) | 2009-07-02 |
RU2008152758A (ru) | 2010-07-20 |
JPWO2007142295A1 (ja) | 2009-10-29 |
AU2007255724B2 (en) | 2012-05-10 |
AU2007255724A1 (en) | 2007-12-13 |
JP5001271B2 (ja) | 2012-08-15 |
US8354121B2 (en) | 2013-01-15 |
EP2036559A4 (en) | 2013-02-20 |
CN101500570B (zh) | 2012-07-04 |
BRPI0713104A2 (pt) | 2012-10-16 |
CA2653827C (en) | 2014-04-08 |
WO2007142295A1 (ja) | 2007-12-13 |
ES2456328T3 (es) | 2014-04-22 |
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Address after: No. 6-8, Doshucho 2-chome, Chuo-ku, Osaka City, Osaka Prefecture, Japan Patentee after: SUMITOMO PHARMACEUTICALS CO.,LTD. Address before: Osaka, Japan Patentee before: Dainippon Sumitomo Pharma Co.,Ltd. |