CN101263115A

CN101263115A - 经取代吲哚和其用途

经取代吲哚和其用途 Download PDF

Info

Publication number: CN101263115A
Authority: CN; China
Prior art keywords: indoles; amino; phenyl; benzyl; alkylsulfonyl
Prior art date: 2005-08-17
Legal status : Pending

Application number

CNA2006800298940A

Other languages

English (en)

Chinese (zh)

Inventor

胡白华

詹姆斯·W·耶特尔

Current Assignee

Wyeth LLC

Original Assignee

Wyeth LLC

Priority date

2005-08-17

Filing date

2006-08-16

Publication date

2008-09-10

2006-08-16 Application filed by Wyeth LLC filed Critical Wyeth LLC

2008-09-10 Publication of CN101263115A publication Critical patent/CN101263115A/zh

Status Pending legal-status Critical Current

Links

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125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims description 83
108010022233 Plasminogen Activator Inhibitor 1 Proteins 0.000 claims description 76
102100039418 Plasminogen activator inhibitor 1 Human genes 0.000 claims description 76
125000004390 alkyl sulfonyl group Chemical group 0.000 claims description 76
125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 claims description 55
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