CL2015001861A1 - Derivados de 1-(sustituidos)-5-fluoro-4-imino-3-metil-3, 4-dihidropirimidin-2 (1h) - Google Patents

Derivados de 1-(sustituidos)-5-fluoro-4-imino-3-metil-3, 4-dihidropirimidin-2 (1h)

Info

Publication number
CL2015001861A1
CL2015001861A1 CL2015001861A CL2015001861A CL2015001861A1 CL 2015001861 A1 CL2015001861 A1 CL 2015001861A1 CL 2015001861 A CL2015001861 A CL 2015001861A CL 2015001861 A CL2015001861 A CL 2015001861A CL 2015001861 A1 CL2015001861 A1 CL 2015001861A1
Authority
CL
Chile
Prior art keywords
imino
fluoro
dihydropyrimidin
derivatives
substituted
Prior art date
Application number
CL2015001861A
Other languages
English (en)
Spanish (es)
Inventor
Beth Lorsbach
Chenglin Yao
W John Owen
Lindsay Stelzer
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of CL2015001861A1 publication Critical patent/CL2015001861A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CL2015001861A 2012-12-28 2015-06-26 Derivados de 1-(sustituidos)-5-fluoro-4-imino-3-metil-3, 4-dihidropirimidin-2 (1h) CL2015001861A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261747128P 2012-12-28 2012-12-28

Publications (1)

Publication Number Publication Date
CL2015001861A1 true CL2015001861A1 (es) 2015-10-02

Family

ID=51022027

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2015001861A CL2015001861A1 (es) 2012-12-28 2015-06-26 Derivados de 1-(sustituidos)-5-fluoro-4-imino-3-metil-3, 4-dihidropirimidin-2 (1h)

Country Status (18)

Country Link
US (1) US9271497B2 (https=)
EP (2) EP2945635A4 (https=)
JP (1) JP6336480B2 (https=)
KR (1) KR20150103095A (https=)
CN (1) CN104994859B (https=)
AU (1) AU2013370470B2 (https=)
BR (1) BR102013033840B1 (https=)
CA (1) CA2893776A1 (https=)
CL (1) CL2015001861A1 (https=)
EC (1) ECSP15032926A (https=)
GT (1) GT201500196A (https=)
HK (1) HK1214518A1 (https=)
IL (1) IL239562B (https=)
MX (1) MX2015008443A (https=)
RU (2) RU2656101C2 (https=)
UA (1) UA117123C2 (https=)
WO (1) WO2014105821A1 (https=)
ZA (1) ZA201504195B (https=)

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RU2638556C2 (ru) 2012-12-28 2017-12-14 Адама Мактешим Лтд. Производные n-(замещенного)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксилата
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NZ722419A (en) 2013-12-31 2018-01-26 Adama Makhteshim Ltd Synergistic fungicidal mixtures and compositions for fungal control
CA2935594C (en) 2013-12-31 2022-05-03 Nakyen Choy 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
KR20170099928A (ko) 2014-12-30 2017-09-01 다우 아그로사이언시즈 엘엘씨 살진균 활성을 갖는 피콜린아미드
RU2687160C2 (ru) 2014-12-30 2019-05-07 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Пиколинамидные соединения с фунгицидной активностью
NZ732812A (en) 2014-12-30 2019-01-25 Dow Agrosciences Llc Use of picolinamides and other compounds as fungicides
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JP6687625B2 (ja) 2014-12-30 2020-04-22 ダウ アグロサイエンシィズ エルエルシー 殺真菌活性を有するピコリンアミド化合物
KR102659552B1 (ko) 2017-05-02 2024-04-23 코르테바 애그리사이언스 엘엘씨 잔디풀 상의 진균 질환에 대한 살진균제로서의 비고리형 피콜린아미드 화합물의 용도
TW201842851A (zh) 2017-05-02 2018-12-16 美商陶氏農業科學公司 用於穀類中的真菌防治之協同性混合物
TWI774761B (zh) 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於穀物中的真菌防治之協同性混合物
CN107192785B (zh) * 2017-06-09 2019-10-15 西南大学 放线菌jy-22抗真菌成分分离方法及其在复配剂中的应用
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
BR102019004480B1 (pt) 2018-03-08 2023-03-28 Dow Agrosciences Llc Picolinamidas como fungicidas
CA3115684A1 (en) 2018-10-15 2020-04-23 Dow Agrosciences Llc Methods for sythesis of oxypicolinamides
EP3876717A1 (en) 2018-11-05 2021-09-15 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
PY2057637A (es) 2019-09-23 2021-10-05 Adama Makhteshim Ltd Proceso para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto
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RU2638556C2 (ru) * 2012-12-28 2017-12-14 Адама Мактешим Лтд. Производные n-(замещенного)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксилата

Also Published As

Publication number Publication date
US9271497B2 (en) 2016-03-01
EP2945635A4 (en) 2016-05-25
RU2018118951A (ru) 2018-11-02
ECSP15032926A (es) 2015-11-30
HK1214518A1 (zh) 2016-07-29
JP6336480B2 (ja) 2018-06-06
EP2945635A1 (en) 2015-11-25
CN104994859A (zh) 2015-10-21
UA117123C2 (uk) 2018-06-25
ZA201504195B (en) 2017-08-30
GT201500196A (es) 2016-03-02
US20150342188A1 (en) 2015-12-03
HK1216147A1 (zh) 2016-10-21
EP3689142A1 (en) 2020-08-05
BR102013033840A2 (pt) 2015-10-06
RU2656101C2 (ru) 2018-05-31
BR102013033840B1 (pt) 2019-09-10
AU2013370470B2 (en) 2018-05-10
MX2015008443A (es) 2015-09-23
CN104994859B (zh) 2018-10-26
RU2018118951A3 (https=) 2019-02-26
AU2013370470A1 (en) 2015-07-02
CA2893776A1 (en) 2014-07-03
RU2015131110A (ru) 2017-02-03
KR20150103095A (ko) 2015-09-09
WO2014105821A1 (en) 2014-07-03
JP2016509589A (ja) 2016-03-31
IL239562A0 (en) 2015-08-31
IL239562B (en) 2018-02-28

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