PL2563129T3 - N3-podstawione pochodne n1-sulfonylo-5-fluoropirymidynonu - Google Patents

N3-podstawione pochodne n1-sulfonylo-5-fluoropirymidynonu

Info

Publication number
PL2563129T3
PL2563129T3 PL11775446T PL11775446T PL2563129T3 PL 2563129 T3 PL2563129 T3 PL 2563129T3 PL 11775446 T PL11775446 T PL 11775446T PL 11775446 T PL11775446 T PL 11775446T PL 2563129 T3 PL2563129 T3 PL 2563129T3
Authority
PL
Poland
Prior art keywords
sulfonyl
substituted
fluoropyrimidinone
derivatives
fluoropyrimidinone derivatives
Prior art date
Application number
PL11775446T
Other languages
English (en)
Inventor
Timothy Boebel
Beth Lorsbach
Timothy Martin
W. John Owen
Michael Sullenberger
Jeffery Webster
Chenglin Yao
Original Assignee
Adama Makhteshim Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adama Makhteshim Ltd filed Critical Adama Makhteshim Ltd
Publication of PL2563129T3 publication Critical patent/PL2563129T3/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim

Landscapes

  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PL11775446T 2010-04-26 2011-04-20 N3-podstawione pochodne n1-sulfonylo-5-fluoropirymidynonu PL2563129T3 (pl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US32785510P 2010-04-26 2010-04-26

Publications (1)

Publication Number Publication Date
PL2563129T3 true PL2563129T3 (pl) 2017-08-31

Family

ID=44816310

Family Applications (1)

Application Number Title Priority Date Filing Date
PL11775446T PL2563129T3 (pl) 2010-04-26 2011-04-20 N3-podstawione pochodne n1-sulfonylo-5-fluoropirymidynonu

Country Status (33)

Country Link
US (1) US8263603B2 (pl)
EP (1) EP2563129B1 (pl)
JP (1) JP5784705B2 (pl)
KR (1) KR101793766B1 (pl)
CN (1) CN102946730B (pl)
AU (1) AU2011245544B2 (pl)
BR (1) BR112012027439B1 (pl)
CA (1) CA2797226C (pl)
CL (1) CL2012002979A1 (pl)
CO (1) CO6592042A2 (pl)
CR (1) CR20120584A (pl)
CY (1) CY1117956T1 (pl)
DK (1) DK2563129T3 (pl)
EC (1) ECSP12012302A (pl)
ES (1) ES2588742T3 (pl)
GT (1) GT201200289A (pl)
HN (1) HN2012002272A (pl)
HR (1) HRP20161107T1 (pl)
HU (1) HUE029489T2 (pl)
IL (1) IL222646A (pl)
LT (1) LT2563129T (pl)
ME (1) ME02530B (pl)
MX (1) MX2012012530A (pl)
NZ (1) NZ603151A (pl)
PH (1) PH12012502138B1 (pl)
PL (1) PL2563129T3 (pl)
PT (1) PT2563129T (pl)
RS (1) RS55239B1 (pl)
RU (1) RU2562840C2 (pl)
SI (1) SI2563129T1 (pl)
SM (1) SMT201600298B (pl)
UA (1) UA108101C2 (pl)
WO (1) WO2011137002A1 (pl)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2012001622A (es) * 2009-08-07 2012-04-11 Dow Agrosciences Llc Derivados de n1-sulfonil-5-fluoropirimidinona.
JP6336480B2 (ja) * 2012-12-28 2018-06-06 アダマ・マクテシム・リミテッド 1−(置換ベンゾイル)−5−フルオロ−4−イミノ−3−メチル−3,4−ジヒドロピリミジン−2(1h)−オンの誘導体
MX2015008444A (es) * 2012-12-28 2015-09-23 Dow Agrosciences Llc Derivados de n-(sustituido)-5-flouro-4-imino-3-metil-2-oxo-3,4-dih idropirimidin-1 (2h)-carboximida.
AU2013370493B2 (en) * 2012-12-28 2017-08-17 Adama Makhteshim Ltd. N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2H)-carboxylate derivatives
KR102309245B1 (ko) * 2012-12-31 2021-10-06 아다마 마켓심 리미티드 살진균제로서의 3-알킬-5-플루오로-4-치환된-이미노-3,4-디히드로피리미딘-2(1h)-온 유도체
EA036389B1 (ru) * 2013-12-31 2020-11-03 Адама Мактешим Лтд. 5-фтор-4-имино-3-(алкил/замещенный алкил)-1-(арилсульфонил)-3,4-дигидропиримидин-2(1h)-он и способы их получения
FI3096619T3 (fi) * 2013-12-31 2025-09-03 Adama Makhteshim Ltd Synergistisiä sienituhoaineseoksia sienten torjuntaan viljakasveissa
MA41272A (fr) * 2014-12-23 2017-10-31 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences
JP6862939B2 (ja) * 2016-03-11 2021-04-21 住友化学株式会社 植物病害防除組成物及び植物病害防除方法
WO2018139560A1 (ja) 2017-01-26 2018-08-02 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
WO2018190350A1 (ja) 2017-04-10 2018-10-18 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
WO2018190351A1 (ja) 2017-04-10 2018-10-18 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
TWI771402B (zh) 2017-04-11 2022-07-21 日商三井化學Agro股份有限公司 吡啶酮化合物及以吡啶酮化合物作為有效成分的農園藝用殺菌劑
JP7157738B2 (ja) 2017-06-08 2022-10-20 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
WO2020022412A1 (ja) 2018-07-25 2020-01-30 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
US12414559B2 (en) 2018-11-05 2025-09-16 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
CA3295216A1 (en) * 2019-07-22 2026-03-02 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
WO2021059160A1 (en) 2019-09-23 2021-04-01 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine -(1h)-one
CN115776980A (zh) * 2020-03-09 2023-03-10 阿达玛马克西姆有限公司 用于制备5-氟-4-亚氨基-3-甲基-1-(甲苯-4-磺酰基)-3,4-二氢-1h-嘧啶-2-酮的方法
WO2021224802A1 (en) * 2020-05-04 2021-11-11 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
BR112023000205A2 (pt) 2020-07-08 2023-04-25 Adama Makhteshim Ltd Misturas fungicidas
PE20250069A1 (es) 2021-01-27 2025-01-13 Adama Makhteshim Ltd 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2(1h)-ona para control de enfermedades de plantas
AU2022268726A1 (en) 2021-05-04 2023-11-23 Adama Makhteshim Ltd. Crystalline forms of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4- dihydropyrimidin-2-one, and mixtures, compositions and methods of use thereof
CN118139845A (zh) * 2021-09-15 2024-06-04 安道麦马克西姆有限公司 用于制备5-氟-4-亚氨基-3-甲基-1-(甲苯-4-磺酰基)-3,4-二氢-1h-嘧啶-2-酮的方法
CA3248206A1 (en) * 2022-01-12 2023-07-20 Adama Makhteshim Ltd. FUNGICIDE MIXTURES COMPRISING A COMBINATION CONTAINING PHTALIMIDE FUNGICIDES
UY40172A (es) 2022-03-03 2023-10-13 Adama Makhteshim Ltd Combinaciones, mezclas y composiciones fungicidas y usos de las mismas
AU2023275068A1 (en) 2022-05-26 2024-11-28 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
CN120882310A (zh) 2023-03-09 2025-10-31 安道麦马克西姆有限公司 杀真菌组合、混合物及组合物以及其用途
EP4680029A1 (en) 2023-03-14 2026-01-21 Adama Makhteshim Ltd. Liquid compositions containing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1h)-one and derivatives thereof and a uv absorber
IL308593A (en) 2023-11-15 2025-06-01 Adama Makhteshim Ltd Reducing environmental impact of fungicidal enhancement
WO2025114931A1 (en) 2023-11-28 2025-06-05 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HRP970239B1 (en) * 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
CA2629295A1 (en) * 2005-11-22 2007-05-31 Ishihara Sangyo Kaisha, Ltd. Germicide composition for agricultural and gardening applications and method for controlling plant disease
ES2549379T3 (es) * 2008-01-22 2015-10-27 Dow Agrosciences Llc Derivados de 4-amino5-fluoropirimidina como fungicidas
PL2317851T3 (pl) * 2008-08-01 2014-06-30 Dow Agrosciences Llc Zastosowanie 5-fluorocytozyny jako fungicydu
MX2012001622A (es) * 2009-08-07 2012-04-11 Dow Agrosciences Llc Derivados de n1-sulfonil-5-fluoropirimidinona.
UA112284C2 (uk) * 2009-08-07 2016-08-25 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні 5-фторпіримідинону

Also Published As

Publication number Publication date
EP2563129A1 (en) 2013-03-06
JP5784705B2 (ja) 2015-09-24
CN102946730A (zh) 2013-02-27
DK2563129T3 (en) 2016-09-12
UA108101C2 (xx) 2015-03-25
WO2011137002A1 (en) 2011-11-03
PT2563129T (pt) 2016-09-05
LT2563129T (lt) 2016-10-25
MX2012012530A (es) 2012-12-17
NZ603151A (en) 2013-10-25
KR101793766B1 (ko) 2017-11-03
HK1182594A1 (en) 2013-12-06
EP2563129B1 (en) 2016-06-01
ECSP12012302A (es) 2012-12-28
JP2013525434A (ja) 2013-06-20
ES2588742T3 (es) 2016-11-04
HRP20161107T1 (hr) 2016-12-30
CO6592042A2 (es) 2013-01-02
BR112012027439A2 (pt) 2015-09-15
GT201200289A (es) 2014-04-08
US20110263627A1 (en) 2011-10-27
US8263603B2 (en) 2012-09-11
SMT201600298B (it) 2016-11-10
CY1117956T1 (el) 2017-05-17
AU2011245544A1 (en) 2012-11-15
RU2012150293A (ru) 2014-06-10
SI2563129T1 (sl) 2016-12-30
CL2012002979A1 (es) 2013-01-25
EP2563129A4 (en) 2013-08-07
CR20120584A (es) 2013-01-03
BR112012027439A8 (pt) 2017-07-11
PH12012502138B1 (en) 2019-09-25
HUE029489T2 (en) 2017-02-28
AU2011245544B2 (en) 2015-04-16
RU2562840C2 (ru) 2015-09-10
ME02530B (me) 2017-02-20
PH12012502138A1 (en) 2013-02-04
IL222646A (en) 2017-01-31
RS55239B1 (sr) 2017-02-28
KR20130093000A (ko) 2013-08-21
CA2797226A1 (en) 2011-11-03
BR112012027439B1 (pt) 2018-01-16
HN2012002272A (es) 2015-04-27
IL222646A0 (en) 2012-12-31
CN102946730B (zh) 2015-02-04
CA2797226C (en) 2019-02-26

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