CY1117956T1 - N3-αντικατεστημενα-n1-sulfonyl-5-fluoropyrimidinone παραγωγα - Google Patents

N3-αντικατεστημενα-n1-sulfonyl-5-fluoropyrimidinone παραγωγα

Info

Publication number
CY1117956T1
CY1117956T1 CY20161100852T CY161100852T CY1117956T1 CY 1117956 T1 CY1117956 T1 CY 1117956T1 CY 20161100852 T CY20161100852 T CY 20161100852T CY 161100852 T CY161100852 T CY 161100852T CY 1117956 T1 CY1117956 T1 CY 1117956T1
Authority
CY
Cyprus
Prior art keywords
sulfonyl
fluoropyrimidinone
replaced
product
fluoropyrimidinones
Prior art date
Application number
CY20161100852T
Other languages
English (en)
Inventor
Timothy Boebel
Beth Lorsbach
Timothy Martin
W John Owen
Michael Sullenberger
Jeffery Webster
Chenglin Yao
Original Assignee
Adama Makhteshim Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adama Makhteshim Ltd filed Critical Adama Makhteshim Ltd
Publication of CY1117956T1 publication Critical patent/CY1117956T1/el

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim

Abstract

Αυτή η παρούσα κοινοποίηση σχετίζεται με το πεδίο των Ν3-αντικατεστημένων-Ν1-sulfonyl-S-fluoropyrimidinones και τα παράγωγα τους και την χρήση αυτών των ενώσεων σαν μυκητοκτόνων.
CY20161100852T 2010-04-26 2016-08-31 N3-αντικατεστημενα-n1-sulfonyl-5-fluoropyrimidinone παραγωγα CY1117956T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32785510P 2010-04-26 2010-04-26
PCT/US2011/033203 WO2011137002A1 (en) 2010-04-26 2011-04-20 N3-substituted-n1-sulfonyl-5-fluoropyrimidinone derivatives

Publications (1)

Publication Number Publication Date
CY1117956T1 true CY1117956T1 (el) 2017-05-17

Family

ID=44816310

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20161100852T CY1117956T1 (el) 2010-04-26 2016-08-31 N3-αντικατεστημενα-n1-sulfonyl-5-fluoropyrimidinone παραγωγα

Country Status (33)

Country Link
US (1) US8263603B2 (el)
EP (1) EP2563129B1 (el)
JP (1) JP5784705B2 (el)
KR (1) KR101793766B1 (el)
CN (1) CN102946730B (el)
AU (1) AU2011245544B2 (el)
BR (1) BR112012027439B1 (el)
CA (1) CA2797226C (el)
CL (1) CL2012002979A1 (el)
CO (1) CO6592042A2 (el)
CR (1) CR20120584A (el)
CY (1) CY1117956T1 (el)
DK (1) DK2563129T3 (el)
EC (1) ECSP12012302A (el)
ES (1) ES2588742T3 (el)
GT (1) GT201200289A (el)
HK (1) HK1182594A1 (el)
HN (1) HN2012002272A (el)
HR (1) HRP20161107T1 (el)
HU (1) HUE029489T2 (el)
IL (1) IL222646A (el)
LT (1) LT2563129T (el)
ME (1) ME02530B (el)
MX (1) MX2012012530A (el)
NZ (1) NZ603151A (el)
PL (1) PL2563129T3 (el)
PT (1) PT2563129T (el)
RS (1) RS55239B1 (el)
RU (1) RU2562840C2 (el)
SI (1) SI2563129T1 (el)
SM (1) SMT201600298B (el)
UA (1) UA108101C2 (el)
WO (1) WO2011137002A1 (el)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ597644A (en) * 2009-08-07 2014-05-30 Dow Agrosciences Llc N1-sulfonyl-5-fluoropyrimidinone derivatives
CA2893776A1 (en) * 2012-12-28 2014-07-03 Dow Agrosciences Llc 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives
CA2893778A1 (en) * 2012-12-28 2014-07-03 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2h)-carboxylate derivatives
AU2013370490B2 (en) 2012-12-28 2018-05-10 Adama Makhteshim Ltd. N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2H)-carboxamide derivatives
CA2894553C (en) * 2012-12-31 2021-03-02 Dow Agrosciences Llc 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
EA029457B1 (ru) * 2013-12-31 2018-03-30 Адама Мактешим Лтд. Синергетические фунгицидные смеси и композиции для борьбы с грибами
AP2016009342A0 (en) * 2013-12-31 2016-07-31 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
MA41272A (fr) * 2014-12-23 2017-10-31 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences
JP6862939B2 (ja) * 2016-03-11 2021-04-21 住友化学株式会社 植物病害防除組成物及び植物病害防除方法
US11051513B2 (en) * 2017-01-26 2021-07-06 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients
EP3611166B1 (en) 2017-04-10 2022-09-21 Mitsui Chemicals Agro, Inc. Pyridone compound, and agricultural and horticultural fungicide having this as active component
JP7168556B2 (ja) 2017-04-10 2022-11-09 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
CN110234627B (zh) 2017-04-11 2023-09-01 三井化学植保株式会社 吡啶酮化合物及以吡啶酮化合物作为有效成分的农园艺用杀菌剂
US11117863B2 (en) 2017-06-08 2021-09-14 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients
MA49639A (fr) 2017-07-17 2020-05-27 Adama Makhteshim Ltd Polymorphes de 5-fluoro-4-imino-3-méthyl-1-tosyl-3,4-dihydropyrimidin-2-one
TWI828725B (zh) 2018-07-25 2024-01-11 日商三井化學植保股份有限公司 吡啶酮化合物及以吡啶酮化合物作為有效成分的農園藝用殺菌劑
PE20212103A1 (es) 2018-11-05 2021-11-04 Adama Makhteshim Ltd Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y metodos de uso de los mismos
UY38798A (es) 2019-07-22 2021-02-26 Adama Makhteshim Ltd Combinaciones, mezclas y composiciones fungicidas y usos de las mismas
MX2022011088A (es) * 2020-03-09 2022-09-29 Adama Makhteshim Ltd Procedimiento para preparar 5-fluoro-4-imino-3-metil-1-(tolueno-4- sulfonil)-3,4-dihidro-1h-pirimidin-2-ona.
UY39197A (es) 2020-05-04 2021-11-30 Adama Makhteshim Ltd Mezclas y composiciones que comprenden 5-fluoro-4-imino-3- metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de las mismas
CA3185119A1 (en) 2020-07-08 2022-01-13 Matteo CERNUSCHI Fungicidal mixtures
WO2022162591A1 (en) 2021-01-27 2022-08-04 Adama Makhteshim Ltd. 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1 h)-one for controlling plant diseases
AU2022268726A1 (en) 2021-05-04 2023-11-23 Adama Makhteshim Ltd. Crystalline forms of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4- dihydropyrimidin-2-one, and mixtures, compositions and methods of use thereof
AR127068A1 (es) * 2021-09-15 2023-12-13 Adama Makhteshim Ltd Procedimiento para preparar 5-fluoro-4-imino-3-metil-1(tolueno-4-sulfonil)-3,4-dihidro-1h-pirimidin-2-ona
WO2023135535A1 (en) * 2022-01-12 2023-07-20 Adama Makhteshim Ltd. Fungicidal mixtures comprising combination containing phthalimide fungicides
TW202400019A (zh) 2022-03-03 2024-01-01 以色列商亞達瑪馬克天辛有限公司 殺真菌組合、混合物、組合物及其用途
WO2023228148A1 (en) 2022-05-26 2023-11-30 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HRP970239B1 (en) * 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
EP2617287A1 (en) * 2005-11-22 2013-07-24 Ishihara Sangyo Kaisha, Ltd. Germicide composition for agricultural and gardening applications and method for controlling plant disease
ES2549046T3 (es) * 2008-01-22 2015-10-22 Dow Agrosciences, Llc Derivados de N-ciano-4-amino-5-fluoro-pirimidina como fungicidas
EP2647287A1 (en) * 2008-08-01 2013-10-09 Dow AgroSciences LLC Use of 5-fluorocytosine and its derivatives as fungicides
UA112284C2 (uk) * 2009-08-07 2016-08-25 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні 5-фторпіримідинону
NZ597644A (en) * 2009-08-07 2014-05-30 Dow Agrosciences Llc N1-sulfonyl-5-fluoropyrimidinone derivatives

Also Published As

Publication number Publication date
KR20130093000A (ko) 2013-08-21
CA2797226C (en) 2019-02-26
CR20120584A (es) 2013-01-03
IL222646A (en) 2017-01-31
ECSP12012302A (es) 2012-12-28
IL222646A0 (en) 2012-12-31
PT2563129T (pt) 2016-09-05
KR101793766B1 (ko) 2017-11-03
CO6592042A2 (es) 2013-01-02
DK2563129T3 (en) 2016-09-12
HRP20161107T1 (hr) 2016-12-30
GT201200289A (es) 2014-04-08
CN102946730B (zh) 2015-02-04
BR112012027439A2 (pt) 2015-09-15
US8263603B2 (en) 2012-09-11
NZ603151A (en) 2013-10-25
CA2797226A1 (en) 2011-11-03
WO2011137002A1 (en) 2011-11-03
RS55239B1 (sr) 2017-02-28
RU2012150293A (ru) 2014-06-10
EP2563129A4 (en) 2013-08-07
RU2562840C2 (ru) 2015-09-10
LT2563129T (lt) 2016-10-25
SMT201600298B (it) 2016-11-10
HK1182594A1 (en) 2013-12-06
UA108101C2 (xx) 2015-03-25
JP5784705B2 (ja) 2015-09-24
BR112012027439B1 (pt) 2018-01-16
PL2563129T3 (pl) 2017-08-31
CL2012002979A1 (es) 2013-01-25
HUE029489T2 (en) 2017-02-28
SI2563129T1 (sl) 2016-12-30
EP2563129B1 (en) 2016-06-01
ME02530B (me) 2017-02-20
ES2588742T3 (es) 2016-11-04
MX2012012530A (es) 2012-12-17
BR112012027439A8 (pt) 2017-07-11
EP2563129A1 (en) 2013-03-06
AU2011245544A1 (en) 2012-11-15
JP2013525434A (ja) 2013-06-20
CN102946730A (zh) 2013-02-27
US20110263627A1 (en) 2011-10-27
HN2012002272A (es) 2015-04-27
AU2011245544B2 (en) 2015-04-16

Similar Documents

Publication Publication Date Title
CY1117956T1 (el) N3-αντικατεστημενα-n1-sulfonyl-5-fluoropyrimidinone παραγωγα
CY1123958T1 (el) Μεθοδος παρασκευης παραγωγων και ενδιαμεσων καρβαμοϋλπυριδονης
CY1121299T1 (el) Υποκατεστημενες τρικυκλικες ενωσεις ως αναστολεις fgfr
CY1121862T1 (el) Αντισωματα anti-phf-tau και χρησεις αυτων
CY1119060T1 (el) Ρυθμιστες ενζυμων μεθυλικης τροποποιησης, συνθεσεις και χρησεις αυτων
CY1122115T1 (el) Παραγωγα ν1-ακυλο-5-φθοροπυριμιδινονης
CY1121129T1 (el) Αναστολεις toy fgfr4 πυριμιδινης
CY1115945T1 (el) Παραγωγα πυραζολοκινολινονης, η παρασκευη τους και η θεραπευτικη τους χρηση
CY1117878T1 (el) Πυριδινo-2-αμιδια χρησιμα ως αγωνιστες του cb2
EA201270257A1 (ru) Производные n1-сульфонил-5-фторпиримидинона
CY1118950T1 (el) Νεα παραγωγα πυραζολιου
CY1118885T1 (el) Συνθετικες πεπτιδογλυκανες που δεσμευουν υαλουρονικο οξυ, παρασκευη, και μεθοδοι χρησης
CY1120460T1 (el) Παραγωγο πυραζολοπυριμιδινης με υποκατεστημενη τη θεση 4, και χρηση αυτου στην παρασκευη φαρμακων
EA201270254A1 (ru) Производные 5-фторпиримидинона
UY34602A (es) ?Derivados de bencimidazolil- e imidazopiridinil-metilamina?
CR20140468A (es) Inhibidores de diacilglicerol aciltransferasa 2
UY34472A (es) Derivados modificados de 4-fenil-piridina
BR112016029333A2 (pt) síntese de compostos de carbamoilpiridona policíclico
CR20150470A (es) Derivados de triazolona de piridinilo y piridinilo fusionado
CY1120204T1 (el) Αμορφη στερεα διασπορα για χρηση σε θεραπεια καρκινου του εγκεφαλο
EA201591728A1 (ru) Гетероциклические соединения и способы их применения
FI20115758A (fi) Uusia viljatuotteita, niiden valmistus ja käyttö, ja niitä sisältäviä kosmeettisia formulaatioita
CY1120759T1 (el) Παρασκευη διγλυκοζιτη (s,s)-σεκοϊσολαρικιρεσινολης και διγλυκοζιτη (r,r)-σεκοϊσολαρικιρεσινολης
EA201591451A1 (ru) Модуляторы flap
CR20110403A (es) Derivados de tiadiazoles y oxadiazoles, su preparación y su aplicación en terapia