BR112012027439A2 - derivados de n1-sulfonil-5-flúor-pirimidinona n3-substituídos - Google Patents

derivados de n1-sulfonil-5-flúor-pirimidinona n3-substituídos

Info

Publication number
BR112012027439A2
BR112012027439A2 BR112012027439A BR112012027439A BR112012027439A2 BR 112012027439 A2 BR112012027439 A2 BR 112012027439A2 BR 112012027439 A BR112012027439 A BR 112012027439A BR 112012027439 A BR112012027439 A BR 112012027439A BR 112012027439 A2 BR112012027439 A2 BR 112012027439A2
Authority
BR
Brazil
Prior art keywords
sulfonyl
fluoro
unsubstituted
pyrimidinone derivatives
derivatives
Prior art date
Application number
BR112012027439A
Other languages
English (en)
Other versions
BR112012027439A8 (pt
BR112012027439B1 (pt
Inventor
Beth Lorsbach
Chenglin Yao
Jeffery Webster
Michael Sullenberger
Timothy Boebel
Timothy Martin
W John Owen
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of BR112012027439A2 publication Critical patent/BR112012027439A2/pt
Publication of BR112012027439A8 publication Critical patent/BR112012027439A8/pt
Publication of BR112012027439B1 publication Critical patent/BR112012027439B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim

Landscapes

  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Epidemiology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

derivados de n1-sulfonil-5-flúor-pirimidinona n3-substituídos. a presente invenção refere-se ao campo de n1-sulfonil-5-flúor-primidinomas n3-substituídos e seus derivados e ao uso destes compostos como fungicidas.
BR112012027439-2A 2010-04-26 2011-04-20 N3-Substituted N1-Sulfonyl-5-Fluoro-Pyrimidinone Derivatives BR112012027439B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US32785510P 2010-04-26 2010-04-26
US61327855 2010-04-26
PCT/US2011/033203 WO2011137002A1 (en) 2010-04-26 2011-04-20 N3-substituted-n1-sulfonyl-5-fluoropyrimidinone derivatives

Publications (3)

Publication Number Publication Date
BR112012027439A2 true BR112012027439A2 (pt) 2015-09-15
BR112012027439A8 BR112012027439A8 (pt) 2017-07-11
BR112012027439B1 BR112012027439B1 (pt) 2018-01-16

Family

ID=44816310

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112012027439-2A BR112012027439B1 (pt) 2010-04-26 2011-04-20 N3-Substituted N1-Sulfonyl-5-Fluoro-Pyrimidinone Derivatives

Country Status (33)

Country Link
US (1) US8263603B2 (pt)
EP (1) EP2563129B1 (pt)
JP (1) JP5784705B2 (pt)
KR (1) KR101793766B1 (pt)
CN (1) CN102946730B (pt)
AU (1) AU2011245544B2 (pt)
BR (1) BR112012027439B1 (pt)
CA (1) CA2797226C (pt)
CL (1) CL2012002979A1 (pt)
CO (1) CO6592042A2 (pt)
CR (1) CR20120584A (pt)
CY (1) CY1117956T1 (pt)
DK (1) DK2563129T3 (pt)
EC (1) ECSP12012302A (pt)
ES (1) ES2588742T3 (pt)
GT (1) GT201200289A (pt)
HK (1) HK1182594A1 (pt)
HN (1) HN2012002272A (pt)
HR (1) HRP20161107T1 (pt)
HU (1) HUE029489T2 (pt)
IL (1) IL222646A (pt)
LT (1) LT2563129T (pt)
ME (1) ME02530B (pt)
MX (1) MX2012012530A (pt)
NZ (1) NZ603151A (pt)
PL (1) PL2563129T3 (pt)
PT (1) PT2563129T (pt)
RS (1) RS55239B1 (pt)
RU (1) RU2562840C2 (pt)
SI (1) SI2563129T1 (pt)
SM (1) SMT201600298B (pt)
UA (1) UA108101C2 (pt)
WO (1) WO2011137002A1 (pt)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
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BR112012002830B1 (pt) * 2009-08-07 2019-05-28 Adama Makhteshim Ltd. Derivados de n1-sulfonil-5-fluoropiri-midinona, composição para controle de um patógeno fúngico, e método para controle ou prevenção de ataque de fungos em uma planta
CN104994859B (zh) * 2012-12-28 2018-10-26 阿达玛马克西姆股份有限公司 1-(取代的苯甲酰基)-5-氟-4-亚氨基-3-甲基-3,4-二氢嘧啶-2(1h)-酮衍生物
MX2015008444A (es) * 2012-12-28 2015-09-23 Dow Agrosciences Llc Derivados de n-(sustituido)-5-flouro-4-imino-3-metil-2-oxo-3,4-dih idropirimidin-1 (2h)-carboximida.
WO2014105844A1 (en) * 2012-12-28 2014-07-03 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxylate derivatives
CN112094262A (zh) * 2012-12-31 2020-12-18 阿达玛马克西姆股份有限公司 作为杀真菌剂的化合物
EA030030B1 (ru) * 2013-12-31 2018-06-29 Адама Мактешим Лтд. Синергетические фунгицидные смеси и синергетические фунгицидные композиции для борьбы с грибами
MX2016008758A (es) * 2013-12-31 2017-05-09 Adama Makhteshim Ltd 5-fluor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4 -dihidropirimidin-2(1h)-ona y los procesos para su preparacion.
MA41272A (fr) * 2014-12-23 2017-10-31 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences
JP6862939B2 (ja) * 2016-03-11 2021-04-21 住友化学株式会社 植物病害防除組成物及び植物病害防除方法
US11051513B2 (en) * 2017-01-26 2021-07-06 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients
WO2018190350A1 (ja) 2017-04-10 2018-10-18 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
JP7134946B2 (ja) 2017-04-10 2022-09-12 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
CN110234627B (zh) 2017-04-11 2023-09-01 三井化学植保株式会社 吡啶酮化合物及以吡啶酮化合物作为有效成分的农园艺用杀菌剂
EP3636636B1 (en) 2017-06-08 2022-07-06 Mitsui Chemicals Agro, Inc. Pyridone compound and agricultural and horticultural fungicide
IL309708A (en) 2017-07-17 2024-02-01 Adama Makhteshim Ltd Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one
TWI828725B (zh) 2018-07-25 2024-01-11 日商三井化學植保股份有限公司 吡啶酮化合物及以吡啶酮化合物作為有效成分的農園藝用殺菌劑
CR20210270A (es) 2018-11-05 2021-07-20 Adama Makhteshim Ltd Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de los mismos
BR112022001191A2 (pt) * 2019-07-22 2022-03-15 Adama Makhteshim Ltd Combinações fungicidas, misturas e composições e usos das mesmas
IL296178A (en) * 2020-03-09 2022-11-01 Adama Makhteshim Ltd Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-4,3-dihydro-1h-pyrimidin-2-one
CN116113623A (zh) 2020-05-04 2023-05-12 阿达玛马克西姆有限公司 包含5-氟-4-亚氨基-3-甲基-1-甲苯磺酰基-3,4-二氢嘧啶-2-酮的混合物及组合物，及其使用方法
PE20230375A1 (es) 2020-07-08 2023-03-06 Adama Makhteshim Ltd Mezclas fungicidas
CU20230035A7 (es) 2021-01-27 2024-04-08 Adama Makhteshim Ltd 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2(1h)-ona para control de enfermedades de las plantas
BR112023023105A2 (pt) 2021-05-04 2024-01-30 Adama Makhteshim Ltd Formas cristalinas de 5-fluoro-4-imino-3-metil-1-tosil-3,4-di-hidropirimidin-2-ona, e misturas, composições e métodos de uso das mesmas
WO2023042126A1 (en) * 2021-09-15 2023-03-23 Adama Makhteshim Ltd. Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one
WO2023135535A1 (en) * 2022-01-12 2023-07-20 Adama Makhteshim Ltd. Fungicidal mixtures comprising combination containing phthalimide fungicides
WO2023166485A1 (en) 2022-03-03 2023-09-07 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
WO2023228148A1 (en) 2022-05-26 2023-11-30 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof

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Publication number Priority date Publication date Assignee Title
HRP970239B1 (en) * 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
EP2617287A1 (en) * 2005-11-22 2013-07-24 Ishihara Sangyo Kaisha, Ltd. Germicide composition for agricultural and gardening applications and method for controlling plant disease
ES2549379T3 (es) * 2008-01-22 2015-10-27 Dow Agrosciences Llc Derivados de 4-amino5-fluoropirimidina como fungicidas
UA107651C2 (en) * 2008-08-01 2015-02-10 Dow Agrosciences Llc Use of 5-fluorocytosine as a fungicide
UA112284C2 (uk) * 2009-08-07 2016-08-25 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні 5-фторпіримідинону
BR112012002830B1 (pt) * 2009-08-07 2019-05-28 Adama Makhteshim Ltd. Derivados de n1-sulfonil-5-fluoropiri-midinona, composição para controle de um patógeno fúngico, e método para controle ou prevenção de ataque de fungos em uma planta

Also Published As

Publication number Publication date
HN2012002272A (es) 2015-04-27
EP2563129A1 (en) 2013-03-06
MX2012012530A (es) 2012-12-17
BR112012027439A8 (pt) 2017-07-11
KR101793766B1 (ko) 2017-11-03
ME02530B (me) 2017-02-20
HK1182594A1 (en) 2013-12-06
AU2011245544A1 (en) 2012-11-15
CA2797226C (en) 2019-02-26
KR20130093000A (ko) 2013-08-21
LT2563129T (lt) 2016-10-25
PL2563129T3 (pl) 2017-08-31
EP2563129B1 (en) 2016-06-01
HUE029489T2 (en) 2017-02-28
CR20120584A (es) 2013-01-03
IL222646A (en) 2017-01-31
GT201200289A (es) 2014-04-08
US8263603B2 (en) 2012-09-11
PT2563129T (pt) 2016-09-05
JP2013525434A (ja) 2013-06-20
DK2563129T3 (en) 2016-09-12
CN102946730A (zh) 2013-02-27
CA2797226A1 (en) 2011-11-03
EP2563129A4 (en) 2013-08-07
AU2011245544B2 (en) 2015-04-16
BR112012027439B1 (pt) 2018-01-16
SI2563129T1 (sl) 2016-12-30
US20110263627A1 (en) 2011-10-27
UA108101C2 (xx) 2015-03-25
RU2012150293A (ru) 2014-06-10
RU2562840C2 (ru) 2015-09-10
CO6592042A2 (es) 2013-01-02
CY1117956T1 (el) 2017-05-17
ECSP12012302A (es) 2012-12-28
RS55239B1 (sr) 2017-02-28
HRP20161107T1 (hr) 2016-12-30
JP5784705B2 (ja) 2015-09-24
CN102946730B (zh) 2015-02-04
ES2588742T3 (es) 2016-11-04
IL222646A0 (en) 2012-12-31
CL2012002979A1 (es) 2013-01-25
NZ603151A (en) 2013-10-25
WO2011137002A1 (en) 2011-11-03
SMT201600298B (it) 2016-11-10

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B25A Requested transfer of rights approved

Owner name: ADAMA MAKHTESHIM LTD. (IL)

B15K Others concerning applications: alteration of classification

Ipc: A01N 43/54 (2006.01), C07D 239/47 (2006.01), A01P

B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]
B25G Requested change of headquarter approved