RS55239B1 - N3-supstituisani derivati n1-sulfonil-5-fluorpirimidinona - Google Patents

N3-supstituisani derivati n1-sulfonil-5-fluorpirimidinona

Info

Publication number
RS55239B1
RS55239B1 RS20160719A RSP20160719A RS55239B1 RS 55239 B1 RS55239 B1 RS 55239B1 RS 20160719 A RS20160719 A RS 20160719A RS P20160719 A RSP20160719 A RS P20160719A RS 55239 B1 RS55239 B1 RS 55239B1
Authority
RS
Serbia
Prior art keywords
sulfonyl
substituted
fluoropyrimidinone
derivatives
fluoropyrimidinone derivatives
Prior art date
Application number
RS20160719A
Other languages
English (en)
Inventor
Timothy Boebel
Beth Lorsbach
Timothy Martin
W John Owen
Michael Sullenberger
Jeffery Webster
Chenglin Yao
Original Assignee
Adama Makhteshim Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adama Makhteshim Ltd filed Critical Adama Makhteshim Ltd
Publication of RS55239B1 publication Critical patent/RS55239B1/sr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim

Landscapes

  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Epidemiology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
RS20160719A 2010-04-26 2011-04-20 N3-supstituisani derivati n1-sulfonil-5-fluorpirimidinona RS55239B1 (sr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US32785510P 2010-04-26 2010-04-26
PCT/US2011/033203 WO2011137002A1 (en) 2010-04-26 2011-04-20 N3-substituted-n1-sulfonyl-5-fluoropyrimidinone derivatives
EP11775446.5A EP2563129B1 (en) 2010-04-26 2011-04-20 N3-substituted-n1-sulfonyl-5-fluoropyrimidinone derivatives

Publications (1)

Publication Number Publication Date
RS55239B1 true RS55239B1 (sr) 2017-02-28

Family

ID=44816310

Family Applications (1)

Application Number Title Priority Date Filing Date
RS20160719A RS55239B1 (sr) 2010-04-26 2011-04-20 N3-supstituisani derivati n1-sulfonil-5-fluorpirimidinona

Country Status (33)

Country Link
US (1) US8263603B2 (sr)
EP (1) EP2563129B1 (sr)
JP (1) JP5784705B2 (sr)
KR (1) KR101793766B1 (sr)
CN (1) CN102946730B (sr)
AU (1) AU2011245544B2 (sr)
BR (1) BR112012027439B1 (sr)
CA (1) CA2797226C (sr)
CL (1) CL2012002979A1 (sr)
CO (1) CO6592042A2 (sr)
CR (1) CR20120584A (sr)
CY (1) CY1117956T1 (sr)
DK (1) DK2563129T3 (sr)
EC (1) ECSP12012302A (sr)
ES (1) ES2588742T3 (sr)
GT (1) GT201200289A (sr)
HK (1) HK1182594A1 (sr)
HN (1) HN2012002272A (sr)
HR (1) HRP20161107T1 (sr)
HU (1) HUE029489T2 (sr)
IL (1) IL222646A (sr)
LT (1) LT2563129T (sr)
ME (1) ME02530B (sr)
MX (1) MX2012012530A (sr)
NZ (1) NZ603151A (sr)
PL (1) PL2563129T3 (sr)
PT (1) PT2563129T (sr)
RS (1) RS55239B1 (sr)
RU (1) RU2562840C2 (sr)
SI (1) SI2563129T1 (sr)
SM (1) SMT201600298B (sr)
UA (1) UA108101C2 (sr)
WO (1) WO2011137002A1 (sr)

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KR101743791B1 (ko) * 2009-08-07 2017-06-05 다우 아그로사이언시즈 엘엘씨 N1-술포닐-5-플루오로피리미디논 유도체
KR20150100869A (ko) * 2012-12-28 2015-09-02 다우 아그로사이언시즈 엘엘씨 N-(치환된)-5-플루오로-4-이미노-3-메틸-2-옥소-3,4-디히드로피리미딘-1(2h)-카르복스아미드 유도체
WO2014105844A1 (en) * 2012-12-28 2014-07-03 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxylate derivatives
UA117123C2 (uk) * 2012-12-28 2018-06-25 Адама Махтешім Лтд. Похідні 1-(заміщений бензоїл)-5-фтор-4-іміно-3-метил-3,4-дигідропіримідин-2(1h)-ону
WO2014105845A1 (en) * 2012-12-31 2014-07-03 Dow Agrosciences Llc 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
CN106061262A (zh) * 2013-12-31 2016-10-26 阿达玛马克西姆股份有限公司 用防治谷类中真菌的协同杀真菌混合物
NZ722439A (en) * 2013-12-31 2018-01-26 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
MA41272A (fr) * 2014-12-23 2017-10-31 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences
JP6862939B2 (ja) * 2016-03-11 2021-04-21 住友化学株式会社 植物病害防除組成物及び植物病害防除方法
JP7037507B2 (ja) * 2017-01-26 2022-03-16 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
WO2018190351A1 (ja) 2017-04-10 2018-10-18 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
WO2018190350A1 (ja) 2017-04-10 2018-10-18 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
TWI771402B (zh) 2017-04-11 2022-07-21 日商三井化學Agro股份有限公司 吡啶酮化合物及以吡啶酮化合物作為有效成分的農園藝用殺菌劑
JP7157738B2 (ja) 2017-06-08 2022-10-20 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
WO2019038583A1 (en) 2017-07-17 2019-02-28 Adama Makhteshim Ltd. 5-FLUORO-4-IMINO-3-METHYL-1-TOSYL-3,4-DIHYDROPYRIMIDIN-2-ONE POLYMORPHS
EP3828177B1 (en) 2018-07-25 2023-11-29 Mitsui Chemicals Crop & Life Solutions, Inc. Pyridone compound and agricultural and horticultural fungicide having this as active component
BR112021008755A2 (pt) 2018-11-05 2021-08-10 Adama Makhteshim Ltd. misturas e composições contendo 5-fluoro-4-imino-3- metil-1-tosil-3,4-dihidropirimidina-2-ona, e métodos de uso.
EP4003017A1 (en) 2019-07-22 2022-06-01 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
MX2022011088A (es) * 2020-03-09 2022-09-29 Adama Makhteshim Ltd Procedimiento para preparar 5-fluoro-4-imino-3-metil-1-(tolueno-4- sulfonil)-3,4-dihidro-1h-pirimidin-2-ona.
JP2023523655A (ja) 2020-05-04 2023-06-06 アダマ・マクテシム・リミテッド 5-フルオロ-4-イミノ-3-メチル-1-トシル-3,4-ジヒドロピリミジン-2-オンを含む混合物および組成物ならびにその使用方法
CA3185119A1 (en) 2020-07-08 2022-01-13 Matteo CERNUSCHI Fungicidal mixtures
US20240172750A1 (en) 2021-01-27 2024-05-30 Adama Makhteshim Ltd. 5-Fluoro-4-Imino-3-Methyl-1-Tosyl-3,4-Dihydropyrimidin-2(1H)-One for Controlling Plant Diseases
EP4334291A1 (en) 2021-05-04 2024-03-13 Adama Makhteshim Ltd. Crystalline forms of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4- dihydropyrimidin-2-one, and mixtures, compositions and methods of use thereof
WO2023042126A1 (en) * 2021-09-15 2023-03-23 Adama Makhteshim Ltd. Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one
WO2023135535A1 (en) * 2022-01-12 2023-07-20 Adama Makhteshim Ltd. Fungicidal mixtures comprising combination containing phthalimide fungicides
TW202400019A (zh) 2022-03-03 2024-01-01 以色列商亞達瑪馬克天辛有限公司 殺真菌組合、混合物、組合物及其用途
WO2023228148A1 (en) 2022-05-26 2023-11-30 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HRP970239B1 (en) * 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
EP1952689A4 (en) * 2005-11-22 2012-12-12 Ishihara Sangyo Kaisha GERMICIDAL COMPOSITION FOR AGRICULTURAL AND GARDENING APPLICATIONS AND METHOD FOR CONTROLLING PLANT DISEASES
JP5749017B2 (ja) * 2008-01-22 2015-07-15 ダウ アグロサイエンシィズ エルエルシー 5−フルオロピリミジン誘導体
EP2317851B1 (en) * 2008-08-01 2014-01-15 Dow AgroSciences LLC Use of 5-fluorocytosine as a fungicide
UA112284C2 (uk) * 2009-08-07 2016-08-25 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні 5-фторпіримідинону
KR101743791B1 (ko) 2009-08-07 2017-06-05 다우 아그로사이언시즈 엘엘씨 N1-술포닐-5-플루오로피리미디논 유도체

Also Published As

Publication number Publication date
HN2012002272A (es) 2015-04-27
LT2563129T (lt) 2016-10-25
CO6592042A2 (es) 2013-01-02
MX2012012530A (es) 2012-12-17
JP2013525434A (ja) 2013-06-20
IL222646A (en) 2017-01-31
CR20120584A (es) 2013-01-03
US8263603B2 (en) 2012-09-11
AU2011245544A1 (en) 2012-11-15
US20110263627A1 (en) 2011-10-27
BR112012027439B1 (pt) 2018-01-16
CN102946730B (zh) 2015-02-04
NZ603151A (en) 2013-10-25
CA2797226C (en) 2019-02-26
HUE029489T2 (en) 2017-02-28
EP2563129A1 (en) 2013-03-06
WO2011137002A1 (en) 2011-11-03
RU2562840C2 (ru) 2015-09-10
PT2563129T (pt) 2016-09-05
AU2011245544B2 (en) 2015-04-16
ME02530B (me) 2017-02-20
GT201200289A (es) 2014-04-08
BR112012027439A2 (pt) 2015-09-15
JP5784705B2 (ja) 2015-09-24
CN102946730A (zh) 2013-02-27
UA108101C2 (xx) 2015-03-25
HK1182594A1 (en) 2013-12-06
RU2012150293A (ru) 2014-06-10
PL2563129T3 (pl) 2017-08-31
KR20130093000A (ko) 2013-08-21
HRP20161107T1 (hr) 2016-12-30
CL2012002979A1 (es) 2013-01-25
ECSP12012302A (es) 2012-12-28
DK2563129T3 (en) 2016-09-12
SMT201600298B (it) 2016-11-10
SI2563129T1 (sl) 2016-12-30
EP2563129A4 (en) 2013-08-07
BR112012027439A8 (pt) 2017-07-11
EP2563129B1 (en) 2016-06-01
CA2797226A1 (en) 2011-11-03
ES2588742T3 (es) 2016-11-04
CY1117956T1 (el) 2017-05-17
IL222646A0 (en) 2012-12-31
KR101793766B1 (ko) 2017-11-03

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