LT3371190T - Heterocikliniai junginiai, kaip pi3k-gama inhibitoriai - Google Patents
Heterocikliniai junginiai, kaip pi3k-gama inhibitoriaiInfo
- Publication number
- LT3371190T LT3371190T LTEPPCT/US2016/060468T LT16060468T LT3371190T LT 3371190 T LT3371190 T LT 3371190T LT 16060468 T LT16060468 T LT 16060468T LT 3371190 T LT3371190 T LT 3371190T
- Authority
- LT
- Lithuania
- Prior art keywords
- pi3k
- heterocyclic compounds
- gamma inhibitors
- gamma
- inhibitors
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
- Oncology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Epidemiology (AREA)
- Hematology (AREA)
- Dermatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Transplantation (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201562252050P | 2015-11-06 | 2015-11-06 | |
PCT/US2016/060468 WO2017079519A1 (en) | 2015-11-06 | 2016-11-04 | Heterocyclic compounds as pi3k-gamma inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
LT3371190T true LT3371190T (lt) | 2022-08-10 |
Family
ID=57460598
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
LTEPPCT/US2016/060468T LT3371190T (lt) | 2015-11-06 | 2016-11-04 | Heterocikliniai junginiai, kaip pi3k-gama inhibitoriai |
Country Status (17)
Country | Link |
---|---|
US (4) | US10065963B2 (lt) |
EP (2) | EP4086259A1 (lt) |
JP (1) | JP6854817B2 (lt) |
AR (1) | AR106595A1 (lt) |
DK (1) | DK3371190T3 (lt) |
ES (1) | ES2915550T3 (lt) |
HR (1) | HRP20220599T1 (lt) |
HU (1) | HUE059324T2 (lt) |
LT (1) | LT3371190T (lt) |
MA (1) | MA43169B1 (lt) |
MD (1) | MD3371190T2 (lt) |
PL (1) | PL3371190T3 (lt) |
PT (1) | PT3371190T (lt) |
RS (1) | RS63359B1 (lt) |
SI (1) | SI3371190T1 (lt) |
TW (2) | TWI744256B (lt) |
WO (1) | WO2017079519A1 (lt) |
Families Citing this family (21)
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US20180185368A1 (en) | 2014-11-06 | 2018-07-05 | Lysosomal Therapeutics Inc. | Substituted pyrrolo[1,2-a]pyrimidines and their use in the treatment of medical disorders |
US20170333435A1 (en) | 2014-11-06 | 2017-11-23 | Lysosomal Therapeutics Inc. | Substituted imidazo[1,5-a]pyrimidines and their use in the treatment of medical disorders |
DK3215511T3 (da) | 2014-11-06 | 2024-05-13 | Bial R&D Invest S A | Substituerede pyrazolo(1,5-a)pyrimidiner og deres anvendelse i behandlingen af medicinske lidelser |
WO2016130501A1 (en) | 2015-02-09 | 2016-08-18 | Incyte Corporation | Aza-heteroaryl compounds as pi3k-gamma inhibitors |
AR106595A1 (es) | 2015-11-06 | 2018-01-31 | Incyte Corp | COMPUESTOS HETEROCÍCLICOS COMO INHIBIDORES DE PI3K-g |
MA54567A (fr) | 2016-01-05 | 2021-10-27 | Incyte Corp | Pyridine et composés de pyridimine en tant qu'inhibiteurs de pi3k-gamma |
KR20180132629A (ko) * | 2016-02-25 | 2018-12-12 | 아셰뉴론 에스아 | 글리코시다제 저해제 |
SG11201808830YA (en) | 2016-04-06 | 2018-11-29 | Lysosomal Therapeutics Inc | Pyrazolo[1,5-a]pyrimidinyl carboxamide compounds and their use in the treatment of medical disorders |
US10787454B2 (en) | 2016-04-06 | 2020-09-29 | BIAL—BioTech Investments, Inc. | Imidazo[1,5-a]pyrimidinyl carboxamide compounds and their use in the treatment of medical disorders |
MX2018012207A (es) | 2016-04-06 | 2019-03-28 | Lysosomal Therapeutics Inc | Compuestos de pirrol[1,2-a]pirimidinil carboxamida y su uso en el tratamiento de trastornos médicos. |
WO2017192931A1 (en) | 2016-05-05 | 2017-11-09 | Lysosomal Therapeutics Inc. | SUBSTITUTED IMDAZO[1,2-α]PYRIDINES, SUBSTITUTED IMIDAZO[1,2-α]PYRAZINES, RELATED COMPOUNDS, AND THEIR USE IN THE TREATMENT OF MEDICAL DISORDERS |
MX2018013529A (es) | 2016-05-05 | 2019-07-04 | Lysosomal Therapeutics Inc | Imidazo[1,2-b]piridazinas sustituidas, imidazo[1,5-b]piridazinas sustituidas, compuestos relacionados y su uso en el tratamiento de trastornos médicos. |
AR108875A1 (es) | 2016-06-24 | 2018-10-03 | Incyte Corp | COMPUESTOS HETEROCÍCLICOS COMO INHIBIDORES DE PI3K-g |
SG11202003428VA (en) | 2017-10-18 | 2020-05-28 | Incyte Corp | Condensed imidazole derivatives substituted by tertiary hydroxy groups as pi3k-gamma inhibitors |
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CR20210165A (es) | 2018-09-05 | 2021-10-01 | Incyte Corp | Formas cristalinas de un inhibidor de fosfoinositida 3-quinasa (pi3k) campo técnico |
SG11202110523XA (en) | 2019-03-26 | 2021-10-28 | Ventyx Biosciences Inc | Tyk2 pseudokinase ligands |
CA3131856A1 (en) * | 2019-04-11 | 2020-10-15 | Janssen Pharmaceutica N.V. | Pyridine rings containing derivatives as malt1 inhibitors |
AU2020289537A1 (en) * | 2019-06-06 | 2021-11-25 | Aligos Therapeutics, Inc. | Heterocyclic compounds |
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WO2016130501A1 (en) | 2015-02-09 | 2016-08-18 | Incyte Corporation | Aza-heteroaryl compounds as pi3k-gamma inhibitors |
AR106595A1 (es) | 2015-11-06 | 2018-01-31 | Incyte Corp | COMPUESTOS HETEROCÍCLICOS COMO INHIBIDORES DE PI3K-g |
MA54567A (fr) | 2016-01-05 | 2021-10-27 | Incyte Corp | Pyridine et composés de pyridimine en tant qu'inhibiteurs de pi3k-gamma |
AR108875A1 (es) | 2016-06-24 | 2018-10-03 | Incyte Corp | COMPUESTOS HETEROCÍCLICOS COMO INHIBIDORES DE PI3K-g |
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2016
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- 2016-11-04 MA MA43169A patent/MA43169B1/fr unknown
- 2016-11-04 RS RS20220521A patent/RS63359B1/sr unknown
- 2016-11-04 EP EP22162035.4A patent/EP4086259A1/en not_active Withdrawn
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- 2016-11-04 HR HRP20220599TT patent/HRP20220599T1/hr unknown
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- 2016-11-04 SI SI201631549T patent/SI3371190T1/sl unknown
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- 2016-11-04 PT PT168052389T patent/PT3371190T/pt unknown
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2018
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2019
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US20200031837A1 (en) | 2020-01-30 |
HUE059324T2 (hu) | 2022-11-28 |
JP6854817B2 (ja) | 2021-04-07 |
US11091491B2 (en) | 2021-08-17 |
HRP20220599T1 (hr) | 2022-06-24 |
EP3371190A1 (en) | 2018-09-12 |
DK3371190T3 (da) | 2022-05-23 |
TWI824309B (zh) | 2023-12-01 |
MD3371190T2 (ro) | 2022-09-30 |
RS63359B1 (sr) | 2022-07-29 |
US20190062336A1 (en) | 2019-02-28 |
ES2915550T3 (es) | 2022-06-23 |
TWI744256B (zh) | 2021-11-01 |
US20230009843A1 (en) | 2023-01-12 |
US20170129899A1 (en) | 2017-05-11 |
US10065963B2 (en) | 2018-09-04 |
SI3371190T1 (sl) | 2022-08-31 |
AR106595A1 (es) | 2018-01-31 |
TW202204362A (zh) | 2022-02-01 |
PL3371190T3 (pl) | 2022-11-07 |
WO2017079519A1 (en) | 2017-05-11 |
JP2018532760A (ja) | 2018-11-08 |
EP3371190B1 (en) | 2022-03-30 |
MA43169A (fr) | 2018-09-12 |
PT3371190T (pt) | 2022-07-08 |
TW201726679A (zh) | 2017-08-01 |
EP4086259A1 (en) | 2022-11-09 |
US10472368B2 (en) | 2019-11-12 |
US11773102B2 (en) | 2023-10-03 |
MA43169B1 (fr) | 2022-05-31 |
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