ECSP15032926A - Derivados de 1-(benzoílo-sustituido)-5-fluoro-4-imino-3-metil-3,4-dihidropirimidin-2(1h)-ona - Google Patents

Derivados de 1-(benzoílo-sustituido)-5-fluoro-4-imino-3-metil-3,4-dihidropirimidin-2(1h)-ona

Info

Publication number
ECSP15032926A
ECSP15032926A ECIEPI201532926A ECPI201532926A ECSP15032926A EC SP15032926 A ECSP15032926 A EC SP15032926A EC IEPI201532926 A ECIEPI201532926 A EC IEPI201532926A EC PI201532926 A ECPI201532926 A EC PI201532926A EC SP15032926 A ECSP15032926 A EC SP15032926A
Authority
EC
Ecuador
Prior art keywords
compounds
fungicides
dihydropyrimidin
imino
fluoro
Prior art date
Application number
ECIEPI201532926A
Other languages
English (en)
Spanish (es)
Inventor
W Owen
Beth Lorsbach
Chenglin Yao
Lindsay Stelzer
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of ECSP15032926A publication Critical patent/ECSP15032926A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ECIEPI201532926A 2012-12-28 2015-07-28 Derivados de 1-(benzoílo-sustituido)-5-fluoro-4-imino-3-metil-3,4-dihidropirimidin-2(1h)-ona ECSP15032926A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261747128P 2012-12-28 2012-12-28

Publications (1)

Publication Number Publication Date
ECSP15032926A true ECSP15032926A (es) 2015-11-30

Family

ID=51022027

Family Applications (1)

Application Number Title Priority Date Filing Date
ECIEPI201532926A ECSP15032926A (es) 2012-12-28 2015-07-28 Derivados de 1-(benzoílo-sustituido)-5-fluoro-4-imino-3-metil-3,4-dihidropirimidin-2(1h)-ona

Country Status (18)

Country Link
US (1) US9271497B2 (https=)
EP (2) EP2945635A4 (https=)
JP (1) JP6336480B2 (https=)
KR (1) KR20150103095A (https=)
CN (1) CN104994859B (https=)
AU (1) AU2013370470B2 (https=)
BR (1) BR102013033840B1 (https=)
CA (1) CA2893776A1 (https=)
CL (1) CL2015001861A1 (https=)
EC (1) ECSP15032926A (https=)
GT (1) GT201500196A (https=)
HK (1) HK1214518A1 (https=)
IL (1) IL239562B (https=)
MX (1) MX2015008443A (https=)
RU (2) RU2656101C2 (https=)
UA (1) UA117123C2 (https=)
WO (1) WO2014105821A1 (https=)
ZA (1) ZA201504195B (https=)

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RU2638556C2 (ru) 2012-12-28 2017-12-14 Адама Мактешим Лтд. Производные n-(замещенного)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксилата
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NZ722419A (en) 2013-12-31 2018-01-26 Adama Makhteshim Ltd Synergistic fungicidal mixtures and compositions for fungal control
CA2935594C (en) 2013-12-31 2022-05-03 Nakyen Choy 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
KR20170099928A (ko) 2014-12-30 2017-09-01 다우 아그로사이언시즈 엘엘씨 살진균 활성을 갖는 피콜린아미드
RU2687160C2 (ru) 2014-12-30 2019-05-07 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Пиколинамидные соединения с фунгицидной активностью
NZ732812A (en) 2014-12-30 2019-01-25 Dow Agrosciences Llc Use of picolinamides and other compounds as fungicides
US20180000084A1 (en) 2014-12-30 2018-01-04 Dow Agrosciences Llc Use of picolinamide compounds with fungicidal activity
JP6687625B2 (ja) 2014-12-30 2020-04-22 ダウ アグロサイエンシィズ エルエルシー 殺真菌活性を有するピコリンアミド化合物
KR102659552B1 (ko) 2017-05-02 2024-04-23 코르테바 애그리사이언스 엘엘씨 잔디풀 상의 진균 질환에 대한 살진균제로서의 비고리형 피콜린아미드 화합물의 용도
TW201842851A (zh) 2017-05-02 2018-12-16 美商陶氏農業科學公司 用於穀類中的真菌防治之協同性混合物
TWI774761B (zh) 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於穀物中的真菌防治之協同性混合物
CN107192785B (zh) * 2017-06-09 2019-10-15 西南大学 放线菌jy-22抗真菌成分分离方法及其在复配剂中的应用
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
BR102019004480B1 (pt) 2018-03-08 2023-03-28 Dow Agrosciences Llc Picolinamidas como fungicidas
CA3115684A1 (en) 2018-10-15 2020-04-23 Dow Agrosciences Llc Methods for sythesis of oxypicolinamides
EP3876717A1 (en) 2018-11-05 2021-09-15 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
PY2057637A (es) 2019-09-23 2021-10-05 Adama Makhteshim Ltd Proceso para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto
US12281076B2 (en) 2019-10-18 2025-04-22 Corteva Agriscience Llc Process for synthesis of picolinamides

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CA2894510A1 (en) * 2012-12-28 2014-07-03 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2h)-carboxamide derivatives
RU2638556C2 (ru) * 2012-12-28 2017-12-14 Адама Мактешим Лтд. Производные n-(замещенного)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксилата

Also Published As

Publication number Publication date
US9271497B2 (en) 2016-03-01
EP2945635A4 (en) 2016-05-25
RU2018118951A (ru) 2018-11-02
HK1214518A1 (zh) 2016-07-29
JP6336480B2 (ja) 2018-06-06
EP2945635A1 (en) 2015-11-25
CN104994859A (zh) 2015-10-21
UA117123C2 (uk) 2018-06-25
ZA201504195B (en) 2017-08-30
GT201500196A (es) 2016-03-02
US20150342188A1 (en) 2015-12-03
HK1216147A1 (zh) 2016-10-21
CL2015001861A1 (es) 2015-10-02
EP3689142A1 (en) 2020-08-05
BR102013033840A2 (pt) 2015-10-06
RU2656101C2 (ru) 2018-05-31
BR102013033840B1 (pt) 2019-09-10
AU2013370470B2 (en) 2018-05-10
MX2015008443A (es) 2015-09-23
CN104994859B (zh) 2018-10-26
RU2018118951A3 (https=) 2019-02-26
AU2013370470A1 (en) 2015-07-02
CA2893776A1 (en) 2014-07-03
RU2015131110A (ru) 2017-02-03
KR20150103095A (ko) 2015-09-09
WO2014105821A1 (en) 2014-07-03
JP2016509589A (ja) 2016-03-31
IL239562A0 (en) 2015-08-31
IL239562B (en) 2018-02-28

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