AU2013370470B2 - 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one derivatives - Google Patents

1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one derivatives Download PDF

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Publication number
AU2013370470B2
AU2013370470B2 AU2013370470A AU2013370470A AU2013370470B2 AU 2013370470 B2 AU2013370470 B2 AU 2013370470B2 AU 2013370470 A AU2013370470 A AU 2013370470A AU 2013370470 A AU2013370470 A AU 2013370470A AU 2013370470 B2 AU2013370470 B2 AU 2013370470B2
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AU
Australia
Prior art keywords
compound
plant
compounds
methyl
phenyl
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Ceased
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AU2013370470A
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AU2013370470A1 (en
Inventor
Beth Lorsbach
W. John Owen
Lindsay Stelzer
Chenglin Yao
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Adama Makhteshim Ltd
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Adama Makhteshim Ltd
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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine

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  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2013370470A 2012-12-28 2013-12-23 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one derivatives Ceased AU2013370470B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261747128P 2012-12-28 2012-12-28
US61/747,128 2012-12-28
PCT/US2013/077478 WO2014105821A1 (en) 2012-12-28 2013-12-23 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives

Publications (2)

Publication Number Publication Date
AU2013370470A1 AU2013370470A1 (en) 2015-07-02
AU2013370470B2 true AU2013370470B2 (en) 2018-05-10

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AU2013370470A Ceased AU2013370470B2 (en) 2012-12-28 2013-12-23 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one derivatives

Country Status (18)

Country Link
US (1) US9271497B2 (https=)
EP (2) EP2945635A4 (https=)
JP (1) JP6336480B2 (https=)
KR (1) KR20150103095A (https=)
CN (1) CN104994859B (https=)
AU (1) AU2013370470B2 (https=)
BR (1) BR102013033840B1 (https=)
CA (1) CA2893776A1 (https=)
CL (1) CL2015001861A1 (https=)
EC (1) ECSP15032926A (https=)
GT (1) GT201500196A (https=)
HK (1) HK1214518A1 (https=)
IL (1) IL239562B (https=)
MX (1) MX2015008443A (https=)
RU (2) RU2656101C2 (https=)
UA (1) UA117123C2 (https=)
WO (1) WO2014105821A1 (https=)
ZA (1) ZA201504195B (https=)

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RU2638556C2 (ru) 2012-12-28 2017-12-14 Адама Мактешим Лтд. Производные n-(замещенного)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксилата
AU2013370494B2 (en) 2012-12-31 2017-08-17 Adama Makhteshim Ltd. 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides
NZ722419A (en) 2013-12-31 2018-01-26 Adama Makhteshim Ltd Synergistic fungicidal mixtures and compositions for fungal control
CA2935594C (en) 2013-12-31 2022-05-03 Nakyen Choy 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
KR20170099928A (ko) 2014-12-30 2017-09-01 다우 아그로사이언시즈 엘엘씨 살진균 활성을 갖는 피콜린아미드
RU2687160C2 (ru) 2014-12-30 2019-05-07 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Пиколинамидные соединения с фунгицидной активностью
NZ732812A (en) 2014-12-30 2019-01-25 Dow Agrosciences Llc Use of picolinamides and other compounds as fungicides
US20180000084A1 (en) 2014-12-30 2018-01-04 Dow Agrosciences Llc Use of picolinamide compounds with fungicidal activity
JP6687625B2 (ja) 2014-12-30 2020-04-22 ダウ アグロサイエンシィズ エルエルシー 殺真菌活性を有するピコリンアミド化合物
KR102659552B1 (ko) 2017-05-02 2024-04-23 코르테바 애그리사이언스 엘엘씨 잔디풀 상의 진균 질환에 대한 살진균제로서의 비고리형 피콜린아미드 화합물의 용도
TW201842851A (zh) 2017-05-02 2018-12-16 美商陶氏農業科學公司 用於穀類中的真菌防治之協同性混合物
TWI774761B (zh) 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於穀物中的真菌防治之協同性混合物
CN107192785B (zh) * 2017-06-09 2019-10-15 西南大学 放线菌jy-22抗真菌成分分离方法及其在复配剂中的应用
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
BR102019004480B1 (pt) 2018-03-08 2023-03-28 Dow Agrosciences Llc Picolinamidas como fungicidas
CA3115684A1 (en) 2018-10-15 2020-04-23 Dow Agrosciences Llc Methods for sythesis of oxypicolinamides
EP3876717A1 (en) 2018-11-05 2021-09-15 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
PY2057637A (es) 2019-09-23 2021-10-05 Adama Makhteshim Ltd Proceso para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto
US12281076B2 (en) 2019-10-18 2025-04-22 Corteva Agriscience Llc Process for synthesis of picolinamides

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US20110263627A1 (en) * 2010-04-26 2011-10-27 Dow Agrosciences Llc N3-substituted-n1-sulfonyl-5-fluoropyrimidinone derivatives

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Also Published As

Publication number Publication date
US9271497B2 (en) 2016-03-01
EP2945635A4 (en) 2016-05-25
RU2018118951A (ru) 2018-11-02
ECSP15032926A (es) 2015-11-30
HK1214518A1 (zh) 2016-07-29
JP6336480B2 (ja) 2018-06-06
EP2945635A1 (en) 2015-11-25
CN104994859A (zh) 2015-10-21
UA117123C2 (uk) 2018-06-25
ZA201504195B (en) 2017-08-30
GT201500196A (es) 2016-03-02
US20150342188A1 (en) 2015-12-03
HK1216147A1 (zh) 2016-10-21
CL2015001861A1 (es) 2015-10-02
EP3689142A1 (en) 2020-08-05
BR102013033840A2 (pt) 2015-10-06
RU2656101C2 (ru) 2018-05-31
BR102013033840B1 (pt) 2019-09-10
MX2015008443A (es) 2015-09-23
CN104994859B (zh) 2018-10-26
RU2018118951A3 (https=) 2019-02-26
AU2013370470A1 (en) 2015-07-02
CA2893776A1 (en) 2014-07-03
RU2015131110A (ru) 2017-02-03
KR20150103095A (ko) 2015-09-09
WO2014105821A1 (en) 2014-07-03
JP2016509589A (ja) 2016-03-31
IL239562A0 (en) 2015-08-31
IL239562B (en) 2018-02-28

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