BR112014017799A8 - Compostos inibidores de metaloenzima - Google Patents

Compostos inibidores de metaloenzima

Info

Publication number
BR112014017799A8
BR112014017799A8 BR112014017799A BR112014017799A BR112014017799A8 BR 112014017799 A8 BR112014017799 A8 BR 112014017799A8 BR 112014017799 A BR112014017799 A BR 112014017799A BR 112014017799 A BR112014017799 A BR 112014017799A BR 112014017799 A8 BR112014017799 A8 BR 112014017799A8
Authority
BR
Brazil
Prior art keywords
metalloenzyme inhibitors
metalloenzyme
inhibitors
compounds
fungicidal activity
Prior art date
Application number
BR112014017799A
Other languages
English (en)
Other versions
BR112014017799A2 (pt
Inventor
J Hoekstra William
J Schotzinger Robert
W Rafferty Stephen
Original Assignee
Viamet Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Viamet Pharmaceuticals Inc filed Critical Viamet Pharmaceuticals Inc
Publication of BR112014017799A2 publication Critical patent/BR112014017799A2/pt
Publication of BR112014017799A8 publication Critical patent/BR112014017799A8/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/713—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with four or more nitrogen atoms as the only ring hetero atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N57/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds
    • A01N57/10—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-oxygen bonds or phosphorus-to-sulfur bonds
    • A01N57/16—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-oxygen bonds or phosphorus-to-sulfur bonds containing heterocyclic radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

COMPOSTOS INIBIDORES DE METALOENZIMA. Trata-se de compostos que têm atividade fungicida agrícola.
BR112014017799A 2012-01-20 2013-01-18 Compostos inibidores de metaloenzima BR112014017799A8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261589064P 2012-01-20 2012-01-20
PCT/US2013/022317 WO2013110002A1 (en) 2012-01-20 2013-01-18 Metalloenzyme inhibitor compounds

Publications (2)

Publication Number Publication Date
BR112014017799A2 BR112014017799A2 (pt) 2017-06-20
BR112014017799A8 true BR112014017799A8 (pt) 2017-07-11

Family

ID=48799720

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112014017799A BR112014017799A8 (pt) 2012-01-20 2013-01-18 Compostos inibidores de metaloenzima

Country Status (17)

Country Link
US (1) US9414596B2 (pt)
EP (1) EP2804479A4 (pt)
JP (3) JP2015505538A (pt)
KR (1) KR20140116515A (pt)
CN (1) CN104135861A (pt)
AU (1) AU2013209520A1 (pt)
BR (1) BR112014017799A8 (pt)
CA (1) CA2861341A1 (pt)
CL (1) CL2014001892A1 (pt)
CO (1) CO7111289A2 (pt)
CR (1) CR20140387A (pt)
EA (1) EA201491386A1 (pt)
EC (1) ECSP14014530A (pt)
IN (1) IN2014DN06812A (pt)
MX (1) MX2014008729A (pt)
PH (1) PH12014501653A1 (pt)
WO (1) WO2013110002A1 (pt)

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HUE029892T2 (en) 2009-10-07 2017-04-28 Dow Agrosciences Llc Synergistic fungicidal preparations for fungi in cereals
EP2723731B1 (en) 2011-06-23 2017-10-25 Viamet Pharmaceuticals, Inc. Metalloenzyme inhibitor compounds
ES2774267T3 (es) 2012-01-20 2020-07-20 Mycovia Pharmaceuticals Inc Compuestos inhibidores de metaloenzimas
KR102148190B1 (ko) 2012-12-28 2020-08-26 다우 아그로사이언시즈 엘엘씨 곡류에서의 진균 방제를 위한 상승작용적 살진균 혼합물
RU2015131840A (ru) 2012-12-31 2017-02-03 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Макроциклические пиколинамиды в качестве фунгицидов
US9974304B2 (en) 2013-12-26 2018-05-22 Dow Agrosciences Llc Use of macrocyclic picolinamides as fungicides
CN106061257A (zh) 2013-12-26 2016-10-26 美国陶氏益农公司 大环吡啶酰胺作为杀真菌剂的用途
WO2015143192A1 (en) * 2014-03-19 2015-09-24 Viamet Pharmaceuticals, Inc. 2-(2,4-difluorophenyl)-1,1-difluoro-1-(5-substituted-pyridin-2-yl)-3-(1h-tetrazol-1-yl)propan-2-ols and processes for their preparation
JP6613391B2 (ja) * 2014-03-19 2019-12-04 ブイピーエス‐３，インコーポレイテッド ２−（２，４−ジフルオロフェニル）−１，１−ジフルオロ−１−（５−置換ピリジン−２−イル）−３−（１ｈ−テトラゾール−１−イル）プロパン−２−オールおよびその調製工程
BR112016020937B1 (pt) * 2014-03-19 2022-09-20 The United States Of America, As Represented By The Secretary, Department Of Health & Human Services Processo de preparação de compostos antifúngicos
JP2017507991A (ja) * 2014-03-19 2017-03-23 ヴィアメット ファーマスーティカルズ，インコーポレイテッド 抗真菌化合物の調製方法
JP6518683B2 (ja) 2014-03-19 2019-05-22 ヴィアメット ファーマスーティカルズ（エヌシー），インコーポレイテッド 抗真菌化合物の調製方法
JP6572234B2 (ja) * 2014-03-19 2019-09-04 ヴィアメット ファーマスーティカルズ（エヌシー），インコーポレイテッド 抗真菌化合物の調製方法
WO2015143137A1 (en) * 2014-03-19 2015-09-24 Viamet Pharmaceuticals, Inc. Antifungal compound process
CA2942930A1 (en) 2014-03-19 2015-09-24 Viamet Pharmaceuticals, Inc. Antifungal compound process
JP2017514790A (ja) * 2014-03-19 2017-06-08 ヴィアメット ファーマスーティカルズ，インコーポレイテッド 抗真菌化合物の調製方法
CA2942972A1 (en) * 2014-03-19 2015-09-24 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Antifungal compound process
JP2017513848A (ja) 2014-04-15 2017-06-01 ダウ アグロサイエンシィズ エルエルシー 殺真菌剤としての金属酵素阻害剤化合物
WO2015160664A1 (en) * 2014-04-15 2015-10-22 Dow Agrosciences Llc Metalloenzyme inhibitor compounds as fungicides
EP3139916A4 (en) 2014-05-06 2017-11-15 Dow AgroSciences LLC Macrocyclic picolinamides as fungicides
TW201625577A (zh) 2014-07-08 2016-07-16 陶氏農業科學公司 作爲殺真菌劑之巨環吡啶醯胺（二）
CN106470982A (zh) 2014-07-08 2017-03-01 美国陶氏益农公司 作为杀真菌剂的大环吡啶酰胺
US9936697B2 (en) 2014-12-30 2018-04-10 Dow Agrosciences Llc Fungicidal compositions
BR112017013608B8 (pt) 2014-12-30 2022-08-23 Dow Agrosciences Llc Picolinamidas como fungicidas
NZ732573A (en) 2014-12-30 2019-01-25 Dow Agrosciences Llc Use of picolinamide compounds with fungicidal activity
KR20170100549A (ko) 2014-12-30 2017-09-04 다우 아그로사이언시즈 엘엘씨 살진균 활성을 갖는 피콜린아미드 화합물
CN107205386B (zh) 2014-12-30 2021-07-23 美国陶氏益农公司 具有杀真菌活性的吡啶酰胺
WO2016122802A1 (en) 2014-12-30 2016-08-04 Dow Agrosciences Llc Picolinamide compounds with fungicidal activity
BR112017018823A2 (pt) 2015-03-19 2018-04-24 Viamet Pharmaceuticals, Inc. compostos antifúngicos e processos para a fabricação
EA038214B1 (ru) 2015-09-18 2021-07-23 Майковиа Фармасьютикалс, Инк. Способ получения противогрибковых соединений
WO2017117393A1 (en) 2015-12-30 2017-07-06 Viamet Pharmaceuticals, Inc. Metalloenzyme inhibitor compounds
WO2018045010A1 (en) 2016-08-30 2018-03-08 Dow Agrosciences Llc Pyrido-1,3-oxazine-2,4-dione compounds with fungicidal activity
WO2018044996A1 (en) 2016-08-30 2018-03-08 Dow Agrosciences Llc Picolinamides as fungicides
US10244754B2 (en) 2016-08-30 2019-04-02 Dow Agrosciences Llc Picolinamide N-oxide compounds with fungicidal activity
WO2018044987A1 (en) 2016-08-30 2018-03-08 Dow Agrosciences Llc Thiopicolinamide compounds with fungicidal activity
BR102018000183B1 (pt) 2017-01-05 2023-04-25 Dow Agrosciences Llc Picolinamidas, composição para controle de um patógeno fúngico, e método para controle e prevenção de um ataque por fungos em uma planta
EP3580218A1 (en) * 2017-02-08 2019-12-18 Bayer CropScience Aktiengesellschaft Novel triazole derivatives
US11191269B2 (en) 2017-05-02 2021-12-07 Dow Agrosciences Llc Use of an acyclic picolinamide compound as a fungicide for fungal diseases on turfgrasses
TWI774761B (zh) 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於穀物中的真菌防治之協同性混合物
TW201842851A (zh) 2017-05-02 2018-12-16 美商陶氏農業科學公司 用於穀類中的真菌防治之協同性混合物
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Also Published As

Publication number Publication date
CN104135861A (zh) 2014-11-05
CO7111289A2 (es) 2014-11-10
EP2804479A4 (en) 2015-07-22
JP2015505538A (ja) 2015-02-23
IN2014DN06812A (pt) 2015-05-22
MX2014008729A (es) 2015-02-04
US9414596B2 (en) 2016-08-16
JP2019116476A (ja) 2019-07-18
US20150024938A1 (en) 2015-01-22
WO2013110002A1 (en) 2013-07-25
EA201491386A1 (ru) 2014-11-28
EP2804479A1 (en) 2014-11-26
KR20140116515A (ko) 2014-10-02
JP2017110004A (ja) 2017-06-22
AU2013209520A1 (en) 2014-08-28
ECSP14014530A (es) 2015-06-30
CA2861341A1 (en) 2013-07-25
CR20140387A (es) 2014-11-27
PH12014501653A1 (en) 2014-10-13
BR112014017799A2 (pt) 2017-06-20
CL2014001892A1 (es) 2014-11-14

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]
B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]