CH646057A5 - Mittel zur behandlung von glaucoma. - Google Patents

Mittel zur behandlung von glaucoma. Download PDF

Info

Publication number
CH646057A5
CH646057A5 CH22080A CH22080A CH646057A5 CH 646057 A5 CH646057 A5 CH 646057A5 CH 22080 A CH22080 A CH 22080A CH 22080 A CH22080 A CH 22080A CH 646057 A5 CH646057 A5 CH 646057A5
Authority
CH
Switzerland
Prior art keywords
hydroxy
propoxy
dihydrocarbostyril
compound
compounds
Prior art date
Application number
CH22080A
Other languages
German (de)
English (en)
Inventor
Nobuyuku Tanaka
Yoichi Nishinakamura
Kazuyuku Nakagawa
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26345304&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CH646057(A5) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from JP54010108A external-priority patent/JPS5951927B2/ja
Priority claimed from JP54070361A external-priority patent/JPS5951928B2/ja
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of CH646057A5 publication Critical patent/CH646057A5/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CH22080A 1979-01-30 1980-01-11 Mittel zur behandlung von glaucoma. CH646057A5 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP54010108A JPS5951927B2 (ja) 1979-01-30 1979-01-30 緑内障治療剤
JP54070361A JPS5951928B2 (ja) 1979-06-04 1979-06-04 緑内障治療剤

Publications (1)

Publication Number Publication Date
CH646057A5 true CH646057A5 (de) 1984-11-15

Family

ID=26345304

Family Applications (1)

Application Number Title Priority Date Filing Date
CH22080A CH646057A5 (de) 1979-01-30 1980-01-11 Mittel zur behandlung von glaucoma.

Country Status (15)

Country Link
US (1) US4309432A (US20100268047A1-20101021-C00003.png)
AT (1) AT371340B (US20100268047A1-20101021-C00003.png)
AU (1) AU518814B2 (US20100268047A1-20101021-C00003.png)
CA (1) CA1139669A (US20100268047A1-20101021-C00003.png)
CH (1) CH646057A5 (US20100268047A1-20101021-C00003.png)
DE (1) DE3001011C2 (US20100268047A1-20101021-C00003.png)
DK (1) DK11580A (US20100268047A1-20101021-C00003.png)
ES (1) ES487642A0 (US20100268047A1-20101021-C00003.png)
FI (1) FI800089A (US20100268047A1-20101021-C00003.png)
FR (1) FR2447721A1 (US20100268047A1-20101021-C00003.png)
GB (1) GB2042338B (US20100268047A1-20101021-C00003.png)
IT (1) IT1141662B (US20100268047A1-20101021-C00003.png)
NL (1) NL191575C (US20100268047A1-20101021-C00003.png)
NO (1) NO800059L (US20100268047A1-20101021-C00003.png)
SE (1) SE451069B (US20100268047A1-20101021-C00003.png)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0056420A1 (en) * 1981-01-15 1982-07-28 Schering Corporation Ophthalmic gel
FR2539413A1 (fr) * 1983-01-17 1984-07-20 Pos Lab Carbostyriloximinopropanolamines utiles comme medicaments et procede pour leur preparation
US4792561A (en) * 1986-05-29 1988-12-20 Syntex (U.S.A.) Inc. Carbostyril derivatives as combined thromboxane synthetase and cyclic-AMP phosphodiesterase inhibitors
US4921862A (en) * 1986-05-29 1990-05-01 Syntex (U.S.A.) Inc. Carbostyril derivatives as combined thromboxane synthetase and cyclic-amp phosphodiesterase inhibitors
ES2070151T3 (es) * 1988-08-10 1995-06-01 Otsuka Pharma Co Ltd Agentes cardiotonicos.
US5198448A (en) * 1988-08-10 1993-03-30 Otsuka Pharmaceutical Company, Limited Cardiotonics
DK0389995T3 (da) * 1989-03-28 1995-07-03 Nisshin Flour Milling Co Isoquinolinderivater til behandling af glaukom eller okular hypertension
FR2676740B1 (fr) * 1991-05-23 1993-11-05 Roussel Uclaf Nouveaux derives sterouides du pregna-4,9(11),17(20)-trie-3-one, leur preparation, leur application a la preparation de composes sterouides de type pregna-4,9(11),16-triene-3,20-dione et nouveaux intermediaires.
US5629345A (en) * 1993-07-23 1997-05-13 Vide Pharmaceuticals Methods and compositions for ATP-sensitive K+ channel inhibition for lowering intraocular pressure
US5965620A (en) * 1993-07-23 1999-10-12 Vide Pharmaceuticals Methods and compositions for ATP-sensitive K+ channel inhibition for lowering intraocular pressure
US5776482A (en) * 1996-03-29 1998-07-07 University Of Iowa Research Foundation Tetrahydroquinoline analogues for use in glaucoma treatment
MY116782A (en) 1997-12-22 2004-03-31 Otsuka Pharma Co Ltd Water-soluble eye drop
EP2117344A4 (en) * 2006-12-06 2011-03-16 United States Borax Inc ANIMAL FEED

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3910924A (en) * 1972-04-13 1975-10-07 Otsuka Pharma Co Ltd 3,4-Dihydrocarbostyril derivatives and a process for preparing the same
JPS517672B2 (US20100268047A1-20101021-C00003.png) * 1972-04-13 1976-03-10
AR207554A1 (es) * 1972-12-02 1976-10-15 Otsuka Pharma Co Ltd Procedimiento para producir derivados de 3-alquil-5-((3,4-dihidro-5-carbostiril)oximetil)-oxazolidinona-(2)
JPS5239035B2 (US20100268047A1-20101021-C00003.png) * 1972-12-14 1977-10-03
US3975391A (en) * 1973-12-26 1976-08-17 Otsuka Pharmaceutical Company Limited 5-[1-Hydroxy-2-(substituted-amino)]ethyl-8-hydroxy-3,4-dihydrocarbostyril derivatives
US3953546A (en) * 1973-07-31 1976-04-27 Sumitomo Chemical Company, Limited Thio(dithio)phosphorates
JPS5082218A (US20100268047A1-20101021-C00003.png) * 1973-11-10 1975-07-03
US3994901A (en) * 1974-06-13 1976-11-30 Otsuka Pharmaceutical Company Limited 5-[1-Hydroxy-2-(substituted-amino)]alkyl-8-hydroxy-3,4-dihydrocarbostyril derivatives
US4081447A (en) * 1975-04-09 1978-03-28 Abbott Laboratories 5-[2-Hydroxy-3-(3,4-dimethoxy phenethylamino)]-propoxy-3,4-dihydro carbostyril and pharmaceutically acceptable salts thereof
US4210753A (en) * 1976-03-17 1980-07-01 Otsuka Pharmaceutical Co., Ltd. Carbostyril compounds
CH619453A5 (US20100268047A1-20101021-C00003.png) * 1976-03-17 1980-09-30 Otsuka Pharma Co Ltd
DE2719562C2 (de) * 1976-05-08 1986-05-07 Otsuka Pharmaceutical Co. Ltd., Tokio/Tokyo 3, 4-Dihydrocarbostyrilderivate, Verfahren zu deren Herstellung und Arzneimittel, welche diese enthalten
JPS552631A (en) * 1978-06-19 1980-01-10 Otsuka Pharmaceut Co Ltd 3,4-dihydrocarbostyril derivative
JPS5513241A (en) * 1978-07-14 1980-01-30 Otsuka Pharmaceut Co Ltd Remedy for glaucoma

Also Published As

Publication number Publication date
AU5426579A (en) 1980-08-07
NL191575B (nl) 1995-06-01
ATA14480A (de) 1982-11-15
IT1141662B (it) 1986-10-08
AU518814B2 (en) 1981-10-22
GB2042338A (en) 1980-09-24
FI800089A (fi) 1980-07-31
AT371340B (de) 1983-06-27
NL191575C (nl) 1995-10-03
FR2447721A1 (fr) 1980-08-29
DE3001011C2 (de) 1986-02-06
DK11580A (da) 1980-07-31
FR2447721B1 (US20100268047A1-20101021-C00003.png) 1983-03-11
SE8000245L (sv) 1980-07-31
IT8005106A0 (it) 1980-01-09
DE3001011A1 (de) 1980-08-28
GB2042338B (en) 1983-11-30
NO800059L (no) 1980-07-31
ES8100268A1 (es) 1980-11-01
SE451069B (sv) 1987-08-31
ES487642A0 (es) 1980-11-01
NL8000211A (nl) 1980-08-01
CA1139669A (en) 1983-01-18
US4309432A (en) 1982-01-05

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