CH624405A5 - - Google Patents

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Publication number
CH624405A5
CH624405A5 CH1385676A CH1385676A CH624405A5 CH 624405 A5 CH624405 A5 CH 624405A5 CH 1385676 A CH1385676 A CH 1385676A CH 1385676 A CH1385676 A CH 1385676A CH 624405 A5 CH624405 A5 CH 624405A5
Authority
CH
Switzerland
Prior art keywords
piperidino
propyl
adenine
phenoxymethyl
formula
Prior art date
Application number
CH1385676A
Other languages
German (de)
English (en)
Inventor
Walter-Gunar Dr Rer Nat Friebe
Max Dr Rer Nat Thiel
Kurt Dr Ing Stach
Otto-Henning Dr Rer N Wilhelms
Erika Von Dr Med Moellendorff
Vet Gisbert Dr Med Sponer
Original Assignee
Boehringer Mannheim Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Mannheim Gmbh filed Critical Boehringer Mannheim Gmbh
Publication of CH624405A5 publication Critical patent/CH624405A5/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/26Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32Nitrogen atom
    • C07D473/34Nitrogen atom attached in position 6, e.g. adenine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CH1385676A 1975-11-07 1976-11-03 CH624405A5 (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19752550000 DE2550000A1 (de) 1975-11-07 1975-11-07 Neue purin-derivate und verfahren zu ihrer herstellung

Publications (1)

Publication Number Publication Date
CH624405A5 true CH624405A5 (fi) 1981-07-31

Family

ID=5961168

Family Applications (1)

Application Number Title Priority Date Filing Date
CH1385676A CH624405A5 (fi) 1975-11-07 1976-11-03

Country Status (20)

Country Link
US (1) US4086347A (fi)
JP (1) JPS5259187A (fi)
AT (1) AT344726B (fi)
BE (1) BE847974A (fi)
CA (1) CA1062708A (fi)
CH (1) CH624405A5 (fi)
DD (1) DD126941A5 (fi)
DE (1) DE2550000A1 (fi)
DK (1) DK138077C (fi)
FI (1) FI763149A (fi)
FR (1) FR2330402A1 (fi)
GB (1) GB1510764A (fi)
HU (1) HU176481B (fi)
IE (1) IE43780B1 (fi)
IT (1) IT1063616B (fi)
LU (1) LU76142A1 (fi)
NL (1) NL7612287A (fi)
SE (1) SE423902B (fi)
SU (1) SU683623A3 (fi)
ZA (1) ZA766380B (fi)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2549999A1 (de) * 1975-11-07 1977-05-12 Boehringer Mannheim Gmbh Piperidin-derivate und verfahren zu ihrer herstellung
LU76148A1 (fi) * 1976-11-08 1978-07-10
DE2804416A1 (de) * 1978-02-02 1979-08-09 Boehringer Mannheim Gmbh Neue purin-derivate, verfahren zu deren herstellung sowie diese verbindungen enthaltende arzneimittel
DE2922159A1 (de) * 1979-05-31 1980-12-04 Boehringer Mannheim Gmbh Neue xanthin-derivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
CH648559A5 (de) * 1981-07-20 1985-03-29 Siegfried Ag Theophyllinderivate und verfahren zu deren herstellung.
GB8515934D0 (en) * 1985-06-24 1985-07-24 Janssen Pharmaceutica Nv (4-piperidinomethyl and-hetero)purines
US5258380A (en) * 1985-06-24 1993-11-02 Janssen Pharmaceutica N.V. (4-piperidinylmethyl and -hetero)purines
DE3529497A1 (de) * 1985-08-17 1987-02-26 Boehringer Mannheim Gmbh N(pfeil hoch)6(pfeil hoch)-disubstituierte purinderivate, verfahren zu deren herstellung sowie diese verbindungen enthaltende arzneimittel
FR2741881B1 (fr) * 1995-12-01 1999-07-30 Centre Nat Rech Scient Nouveaux derives de purine possedant notamment des prorietes anti-proliferatives et leurs applications biologiques
US9469644B2 (en) * 2013-03-05 2016-10-18 Hoffmann-La Roche Inc. Inhibitors of Bruton's tyrosine kinase

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2245061A1 (de) * 1972-09-14 1974-03-28 Boehringer Mannheim Gmbh Derivate des adenins
DE2401254A1 (de) * 1974-01-11 1975-11-27 Boehringer Mannheim Gmbh Neue derivate von n hoch 6-substituierten adeninen

Also Published As

Publication number Publication date
FR2330402B1 (fi) 1980-03-07
CA1062708A (en) 1979-09-18
ATA823876A (de) 1977-12-15
NL7612287A (nl) 1977-05-10
DD126941A5 (fi) 1977-08-24
SU683623A3 (ru) 1979-08-30
US4086347A (en) 1978-04-25
AT344726B (de) 1978-08-10
DK138077B (da) 1978-07-10
IE43780B1 (en) 1981-05-20
GB1510764A (en) 1978-05-17
DK494976A (da) 1977-05-08
HU176481B (en) 1981-03-28
IT1063616B (it) 1985-02-11
LU76142A1 (fi) 1977-05-18
DE2550000A1 (de) 1977-05-12
FR2330402A1 (fr) 1977-06-03
ZA766380B (en) 1977-11-30
BE847974A (fr) 1977-05-04
IE43780L (en) 1977-05-07
SE423902B (sv) 1982-06-14
DK138077C (da) 1978-11-27
FI763149A (fi) 1977-05-08
SE7612235L (sv) 1977-05-08
JPS5259187A (en) 1977-05-16

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Legal Events

Date Code Title Description
PL Patent ceased