CA2898000A1 - Solid solution compositions and use in severe pain - Google Patents

Solid solution compositions and use in severe pain Download PDF

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Publication number
CA2898000A1
CA2898000A1 CA2898000A CA2898000A CA2898000A1 CA 2898000 A1 CA2898000 A1 CA 2898000A1 CA 2898000 A CA2898000 A CA 2898000A CA 2898000 A CA2898000 A CA 2898000A CA 2898000 A1 CA2898000 A1 CA 2898000A1
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CA
Canada
Prior art keywords
weight
pharmaceutical composition
pain
solid solution
therapeutic compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA2898000A
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English (en)
French (fr)
Inventor
Robin Mark Bannister
John Brew
Richard Robert REILEY
Wilson Caparros-Wanderley
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Infirst Healthcare Ltd
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Infirst Healthcare Ltd
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Publication of CA2898000A1 publication Critical patent/CA2898000A1/en
Abandoned legal-status Critical Current

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    • A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
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    • A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
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