CA2683461A1 - Novel vanilloid receptor ligands and the use thereof for the production of pharmaceuticals - Google Patents

Novel vanilloid receptor ligands and the use thereof for the production of pharmaceuticals Download PDF

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Publication number
CA2683461A1
CA2683461A1 CA002683461A CA2683461A CA2683461A1 CA 2683461 A1 CA2683461 A1 CA 2683461A1 CA 002683461 A CA002683461 A CA 002683461A CA 2683461 A CA2683461 A CA 2683461A CA 2683461 A1 CA2683461 A1 CA 2683461A1
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Prior art keywords
butyl
group
denotes
case
tert
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Abandoned
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CA002683461A
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English (en)
French (fr)
Inventor
Robert Frank
Gregor Bahrenberg
Thomas Christoph
Klaus Schiene
Jean De Vry
Derek John Saunders
Bernd Sundermann
Jeewoo Lee
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Gruenenthal GmbH
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Individual
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Priority claimed from DE102007018149A external-priority patent/DE102007018149A1/de
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Publication of CA2683461A1 publication Critical patent/CA2683461A1/en
Abandoned legal-status Critical Current

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    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D215/14—Radicals substituted by oxygen atoms
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    • C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
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  • Health & Medical Sciences (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
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  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Addiction (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Urology & Nephrology (AREA)
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  • Obesity (AREA)
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  • Diabetes (AREA)
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  • Ophthalmology & Optometry (AREA)
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  • Hospice & Palliative Care (AREA)
CA002683461A 2007-04-16 2008-04-16 Novel vanilloid receptor ligands and the use thereof for the production of pharmaceuticals Abandoned CA2683461A1 (en)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
DE102007018149A DE102007018149A1 (de) 2007-04-16 2007-04-16 Neue Vanilloid-Rezeptor Liganden und ihre Verwendung zur Herstellung von Arzneimitteln
DE102007018149.5 2007-04-16
EP2008002997 2008-04-15
US12/103,667 US8084484B2 (en) 2007-04-16 2008-04-15 Vanilloid receptor ligands, pharmaceutical compositions containing them, process for making them, and use thereof for treating pain and other conditions
US12/103,667 2008-04-15
EPPCT/EP2008/002997 2008-04-15
PCT/EP2008/003027 WO2008125342A2 (de) 2007-04-16 2008-04-16 Vanilloid-rezeptor-liganden und ihre verwendung zur herstellung von arzneimitteln

Publications (1)

Publication Number Publication Date
CA2683461A1 true CA2683461A1 (en) 2008-10-23

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ID=41360190

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Application Number Title Priority Date Filing Date
CA002683461A Abandoned CA2683461A1 (en) 2007-04-16 2008-04-16 Novel vanilloid receptor ligands and the use thereof for the production of pharmaceuticals

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JP (1) JP2010523727A (enrdf_load_stackoverflow)
KR (1) KR20100016593A (enrdf_load_stackoverflow)
CN (1) CN101679370A (enrdf_load_stackoverflow)
AU (1) AU2008238250B2 (enrdf_load_stackoverflow)
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ECSP099692A (es) 2009-11-30
CO6241154A2 (es) 2011-01-20
CN101679370A (zh) 2010-03-24
AU2008238250A1 (en) 2008-10-23
IL201505A0 (en) 2010-05-31
WO2008125342A3 (de) 2009-01-15
MX2009011149A (es) 2009-10-30
AU2008238250B2 (en) 2013-01-24
WO2008125342A2 (de) 2008-10-23
RU2009142023A (ru) 2011-05-27
ZA200907099B (en) 2013-03-27
JP2010523727A (ja) 2010-07-15
KR20100016593A (ko) 2010-02-12
BRPI0810035A2 (pt) 2016-07-26
RU2498982C2 (ru) 2013-11-20

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