ECSP099692A - Ligandos de receptor de vainilloide novedosos y su uso de los mismos para la produccion de sustancias farmaceuticas - Google Patents

Ligandos de receptor de vainilloide novedosos y su uso de los mismos para la produccion de sustancias farmaceuticas

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Publication number
ECSP099692A
ECSP099692A EC2009009692A ECSP099692A ECSP099692A EC SP099692 A ECSP099692 A EC SP099692A EC 2009009692 A EC2009009692 A EC 2009009692A EC SP099692 A ECSP099692 A EC SP099692A EC SP099692 A ECSP099692 A EC SP099692A
Authority
EC
Ecuador
Prior art keywords
production
pharmaceutical substances
vinylloid
new
receiver links
Prior art date
Application number
EC2009009692A
Other languages
English (en)
Inventor
Jee Woo Lee
Vry Jean Marie Victor De
Thomas Christoph
Robert Frank
Gregor Bahrenberg
Klaus Schiene
Derek John Sauders
Bernd Saudermann
Original Assignee
Gruenenthal Chemie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE102007018149A external-priority patent/DE102007018149A1/de
Application filed by Gruenenthal Chemie filed Critical Gruenenthal Chemie
Publication of ECSP099692A publication Critical patent/ECSP099692A/es

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    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D215/14—Radicals substituted by oxygen atoms
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Abstract

La presente invención se relaciona con ligandos de receptor vainilloide novedosos, un método para la producción de los mismos, sustancias farmacéuticas que contienen dichos compuestos y el uso de tales compuestos para la producción de sustancias farmacéuticas.
EC2009009692A 2007-04-16 2009-10-16 Ligandos de receptor de vainilloide novedosos y su uso de los mismos para la produccion de sustancias farmaceuticas ECSP099692A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE102007018149A DE102007018149A1 (de) 2007-04-16 2007-04-16 Neue Vanilloid-Rezeptor Liganden und ihre Verwendung zur Herstellung von Arzneimitteln
US12/103,667 US8084484B2 (en) 2007-04-16 2008-04-15 Vanilloid receptor ligands, pharmaceutical compositions containing them, process for making them, and use thereof for treating pain and other conditions
EP2008002997 2008-04-15

Publications (1)

Publication Number Publication Date
ECSP099692A true ECSP099692A (es) 2009-11-30

Family

ID=41360190

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2009009692A ECSP099692A (es) 2007-04-16 2009-10-16 Ligandos de receptor de vainilloide novedosos y su uso de los mismos para la produccion de sustancias farmaceuticas

Country Status (14)

Country Link
JP (1) JP2010523727A (es)
KR (1) KR20100016593A (es)
CN (1) CN101679370A (es)
AU (1) AU2008238250B2 (es)
BR (1) BRPI0810035A2 (es)
CA (1) CA2683461A1 (es)
CO (1) CO6241154A2 (es)
EC (1) ECSP099692A (es)
IL (1) IL201505A0 (es)
MX (1) MX2009011149A (es)
NZ (1) NZ580411A (es)
RU (1) RU2498982C2 (es)
WO (1) WO2008125342A2 (es)
ZA (1) ZA200907099B (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102007018149A1 (de) 2007-04-16 2008-10-23 Grünenthal GmbH Neue Vanilloid-Rezeptor Liganden und ihre Verwendung zur Herstellung von Arzneimitteln
MX2011011797A (es) 2009-05-07 2011-11-29 Gruenenthal Gmbh Fenilureas y fenilamidas sustituidas como ligandos del receptor de vanilloides.
US8946204B2 (en) 2009-05-07 2015-02-03 Gruenenthal Gmbh Substituted phenylureas and phenylamides as vanilloid receptor ligands
MX2014000964A (es) 2011-07-26 2014-03-27 Gruenenthal Gmbh Derivados aza heterociclicos sustituidos.
BR112014001714A2 (pt) 2011-07-26 2017-02-14 Gruenenthal Gmbh derivados de carboxamida e ureia aromáticos bicíclicos substituídos como ligantes de receptor vaniloide
AR088701A1 (es) * 2011-11-09 2014-06-25 Gruenenthal Gmbh Derivados de carboxamida y urea basados en pirazolilo, sustituidos, que contienen una porcion fenilo sustituida con un grupo que contiene n como ligandos del receptor de vanilloide
AU2013230425B2 (en) * 2012-03-05 2017-05-25 Dr.Reddy's Laboratories Ltd. Substituted heterocyclic acetamides as kappa opioid receptor (kor) agonists
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