CA2642738A1 - Pi-3 kinase inhibitors and methods of their use - Google Patents
Pi-3 kinase inhibitors and methods of their use Download PDFInfo
- Publication number
- CA2642738A1 CA2642738A1 CA002642738A CA2642738A CA2642738A1 CA 2642738 A1 CA2642738 A1 CA 2642738A1 CA 002642738 A CA002642738 A CA 002642738A CA 2642738 A CA2642738 A CA 2642738A CA 2642738 A1 CA2642738 A1 CA 2642738A1
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- Prior art keywords
- substituted
- alkyl
- amino
- compound
- hydrogen
- Prior art date
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- Abandoned
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Classifications
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- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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Landscapes
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Applications Claiming Priority (5)
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| US77347606P | 2006-02-14 | 2006-02-14 | |
| US60/773,476 | 2006-02-14 | ||
| US87672906P | 2006-12-22 | 2006-12-22 | |
| US60/876,729 | 2006-12-22 | ||
| PCT/US2007/062157 WO2007095588A1 (en) | 2006-02-14 | 2007-02-14 | Pi-3 kinase inhibitors and methods of their use |
Publications (1)
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| CA2642738A1 true CA2642738A1 (en) | 2007-08-23 |
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| CA002642738A Abandoned CA2642738A1 (en) | 2006-02-14 | 2007-02-14 | Pi-3 kinase inhibitors and methods of their use |
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| US (1) | US20100075965A1 (https=) |
| EP (1) | EP1989201A1 (https=) |
| JP (1) | JP2009530233A (https=) |
| KR (1) | KR20080112202A (https=) |
| AR (1) | AR059506A1 (https=) |
| AU (1) | AU2007214462A1 (https=) |
| BR (1) | BRPI0707816A2 (https=) |
| CA (1) | CA2642738A1 (https=) |
| MX (1) | MX2008010397A (https=) |
| PE (1) | PE20070978A1 (https=) |
| RU (1) | RU2008136783A (https=) |
| TW (1) | TW200804379A (https=) |
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| EP2058309A4 (en) * | 2006-08-04 | 2010-12-22 | Takeda Pharmaceutical | CONDENSED HETEROCYCLIC COMPOUND |
| BRPI0716239A2 (pt) | 2006-08-30 | 2013-08-13 | Cellzome Ltd | derivados de triazol como inibidores de cinase |
| CA2672494A1 (en) | 2006-12-14 | 2008-06-19 | Nps Pharmaceuticals, Inc. | Use of d-serine derivatives for the treatment of anxiety disorders |
| US8263585B2 (en) | 2007-05-04 | 2012-09-11 | Novartis Ag | Organic compounds |
| TW200911798A (en) * | 2007-08-02 | 2009-03-16 | Amgen Inc | PI3 kinase modulators and methods of use |
| WO2009021990A1 (en) * | 2007-08-14 | 2009-02-19 | Bayer Schering Pharma Aktiengesellschaft | Fused imidazoles for cancer treatment |
| EP2062893A1 (en) * | 2007-10-18 | 2009-05-27 | Bayer Schering Pharma AG | Fused imidazoles for cancer treatment |
| ES2400604T3 (es) * | 2007-08-17 | 2013-04-11 | Icagen, Inc. | Heterociclos como moduladores del canal de potasio |
| US8431608B2 (en) | 2007-08-17 | 2013-04-30 | Icagen Inc. | Heterocycles as potassium channel modulators |
| CA2691448A1 (en) | 2007-08-31 | 2009-03-05 | Dominique Swinnen | Triazolopyridine compounds and their use as ask inhibitors |
| AU2008328882A1 (en) * | 2007-11-27 | 2009-06-04 | Cellzome Limited | Amino triazoles as PI3K inhibitors |
| AU2008343813B2 (en) * | 2007-12-19 | 2012-04-12 | Amgen Inc. | Inhibitors of PI3 kinase |
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| WO2009126635A1 (en) * | 2008-04-09 | 2009-10-15 | Abbott Laboratories | 2-amino-benzothiazole derivates useful as inhibitors of rock kinases |
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| KR20020084116A (ko) * | 2000-02-07 | 2002-11-04 | 애보트 게엠베하 운트 콤파니 카게 | 2-벤조티아졸릴 우레아 유도체 및 이의 단백질 키나제억제제로서의 용도 |
| DE60115069T2 (de) * | 2000-09-11 | 2006-08-03 | Chiron Corp., Emeryville | Chinolinonderivate als tyrosin-kinase inhibitoren |
| DE60131015T2 (de) * | 2000-12-15 | 2008-07-10 | Vertex Pharmaceuticals Inc., Cambridge | Bakterielle gyrase-hemmer und deren verwendung |
| US20030134846A1 (en) * | 2001-10-09 | 2003-07-17 | Schering Corporation | Treatment of trypanosoma brucei with farnesyl protein transferase inhibitors |
| AU2002316231A1 (en) * | 2002-02-19 | 2003-09-29 | Xenoport, Inc. | Methods for synthesis of prodrugs from 1-acyl-alkyl derivatives and compositions thereof |
| US6900342B2 (en) * | 2002-05-10 | 2005-05-31 | Dabur India Limited | Anticancer taxanes such as paclitaxel, docetaxel and their structural analogs, and a method for the preparation thereof |
| DK1603570T5 (da) * | 2003-02-26 | 2013-12-09 | Sugen Inc | Aminoheteroarylforbindelser som proteinkinaseinhibitorer |
| WO2005035526A1 (en) * | 2003-10-09 | 2005-04-21 | Argenta Discovery Ltd. | Bicyclic compounds and their therapeutic use |
| ES2328047T3 (es) * | 2004-03-19 | 2009-11-06 | Warner-Lambert Company Llc | Derivados de imidazopiridina e imidazopirimidina como agentes antibacterianos. |
| EP2058309A4 (en) * | 2006-08-04 | 2010-12-22 | Takeda Pharmaceutical | CONDENSED HETEROCYCLIC COMPOUND |
-
2007
- 2007-02-12 PE PE2007000145A patent/PE20070978A1/es not_active Application Discontinuation
- 2007-02-13 TW TW096105314A patent/TW200804379A/zh unknown
- 2007-02-14 JP JP2008555474A patent/JP2009530233A/ja active Pending
- 2007-02-14 EP EP07757005A patent/EP1989201A1/en not_active Withdrawn
- 2007-02-14 RU RU2008136783/04A patent/RU2008136783A/ru not_active Application Discontinuation
- 2007-02-14 MX MX2008010397A patent/MX2008010397A/es active IP Right Grant
- 2007-02-14 CA CA002642738A patent/CA2642738A1/en not_active Abandoned
- 2007-02-14 US US12/279,148 patent/US20100075965A1/en not_active Abandoned
- 2007-02-14 AU AU2007214462A patent/AU2007214462A1/en not_active Abandoned
- 2007-02-14 KR KR1020087020573A patent/KR20080112202A/ko not_active Ceased
- 2007-02-14 WO PCT/US2007/062157 patent/WO2007095588A1/en not_active Ceased
- 2007-02-14 BR BRPI0707816-1A patent/BRPI0707816A2/pt not_active IP Right Cessation
- 2007-02-14 AR ARP070100634A patent/AR059506A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JP2009530233A (ja) | 2009-08-27 |
| PE20070978A1 (es) | 2007-11-15 |
| WO2007095588A1 (en) | 2007-08-23 |
| US20100075965A1 (en) | 2010-03-25 |
| AR059506A1 (es) | 2008-04-09 |
| KR20080112202A (ko) | 2008-12-24 |
| BRPI0707816A2 (pt) | 2011-05-10 |
| EP1989201A1 (en) | 2008-11-12 |
| MX2008010397A (es) | 2008-10-27 |
| TW200804379A (en) | 2008-01-16 |
| RU2008136783A (ru) | 2010-03-20 |
| AU2007214462A1 (en) | 2007-08-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request | ||
| FZDE | Discontinued |
Effective date: 20140214 |