CA2123684A1 - Method for making steroidal peracyl glycosides - Google Patents
Method for making steroidal peracyl glycosidesInfo
- Publication number
- CA2123684A1 CA2123684A1 CA002123684A CA2123684A CA2123684A1 CA 2123684 A1 CA2123684 A1 CA 2123684A1 CA 002123684 A CA002123684 A CA 002123684A CA 2123684 A CA2123684 A CA 2123684A CA 2123684 A1 CA2123684 A1 CA 2123684A1
- Authority
- CA
- Canada
- Prior art keywords
- beta
- zinc
- recited
- tigogenin
- cellobioside
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Steroid Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US79757491A | 1991-11-25 | 1991-11-25 | |
| US07/797,574 | 1991-11-25 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2123684A1 true CA2123684A1 (en) | 1993-06-10 |
Family
ID=25171219
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002123684A Abandoned CA2123684A1 (en) | 1991-11-25 | 1992-10-15 | Method for making steroidal peracyl glycosides |
Country Status (13)
| Country | Link |
|---|---|
| EP (1) | EP0619822A1 (cs) |
| JP (1) | JPH0826064B2 (cs) |
| AU (1) | AU659506B2 (cs) |
| CA (1) | CA2123684A1 (cs) |
| FI (1) | FI942394L (cs) |
| HU (1) | HUT67035A (cs) |
| IL (1) | IL103797A0 (cs) |
| MX (1) | MX9206761A (cs) |
| NZ (1) | NZ245244A (cs) |
| PT (1) | PT101088A (cs) |
| TW (1) | TW232699B (cs) |
| WO (1) | WO1993011150A1 (cs) |
| ZA (1) | ZA929081B (cs) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5563259A (en) * | 1992-06-26 | 1996-10-08 | Pfizer Inc. | Process for making β-O-cellobiosyl steroid derivatives and trimethyl silyl steroid intermediates used therein |
| US5606041A (en) * | 1992-06-26 | 1997-02-25 | Pfizer Inc. | Process for steroidal peracyl glycosides |
| JPH07504921A (ja) * | 1992-06-26 | 1995-06-01 | フアイザー・インコーポレイテツド | 高コレステロール血症を治療するためのステロイドグリコシド |
| JPH08504830A (ja) * | 1993-04-28 | 1996-05-28 | フアイザー・インコーポレイテツド | スピロスタニルグリコシド結晶質一水塩 |
| US5502038A (en) * | 1993-06-21 | 1996-03-26 | Medical Research Foundation Of Oregon | Cholesterol sequestrant glycosides that inhibit intestinal cholesterol absorption |
| CA2180148A1 (en) * | 1993-12-28 | 1995-07-06 | Michael Paul Deninno | Hypocholesterolemic agents |
| WO1996038466A1 (en) * | 1995-05-29 | 1996-12-05 | Pfizer Inc. | Steroidal glycosides |
| US5756470A (en) * | 1996-10-29 | 1998-05-26 | Schering Corporation | Sugar-substituted 2-azetidinones useful as hypocholesterolemic agents |
| US6982251B2 (en) | 2000-12-20 | 2006-01-03 | Schering Corporation | Substituted 2-azetidinones useful as hypocholesterolemic agents |
| BR0206654A (pt) | 2001-01-26 | 2004-02-25 | Schering Corp | Combinações de ativador(es) de receptor ativado por proliferação de peroxisoma (ppar) e inibidor(es) de absorção de esterol e tratamentos para indicações vasculares |
| WO2002058696A2 (en) | 2001-01-26 | 2002-08-01 | Schering Corporation | The use of substituted azetidinone compounds for the treatment of sitosterolemia |
| US7071181B2 (en) | 2001-01-26 | 2006-07-04 | Schering Corporation | Methods and therapeutic combinations for the treatment of diabetes using sterol absorption inhibitors |
| DE60216300T2 (de) | 2001-09-21 | 2007-06-28 | Schering Corp. | Behandlung von xanthom mittels azetidinon-derivate als hemmer der sterol absorption |
| US7053080B2 (en) | 2001-09-21 | 2006-05-30 | Schering Corporation | Methods and therapeutic combinations for the treatment of obesity using sterol absorption inhibitors |
| US7056906B2 (en) | 2001-09-21 | 2006-06-06 | Schering Corporation | Combinations of hormone replacement therapy composition(s) and sterol absorption inhibitor(s) and treatments for vascular conditions in post-menopausal women |
| US7560449B2 (en) | 2002-11-06 | 2009-07-14 | Schering Corporation | Methods and therapeutic combinations for the treatment of demyelination |
| ES2311806T3 (es) | 2003-03-07 | 2009-02-16 | Schering Corporation | Compuesto de azetidinona sustituidos, fornulaciones y usos de los mismos para el tratamiento de hipercolesterolemia. |
| US7459442B2 (en) | 2003-03-07 | 2008-12-02 | Schering Corporation | Substituted azetidinone compounds, processes for preparing the same, formulations and uses thereof |
| ES2318274T3 (es) | 2003-03-07 | 2009-05-01 | Schering Corporation | Compuestos de azetidinona sustituida, formulaciones y uso de los mismos para el tratamiento de hipercolesterolemia. |
| MXPA05009502A (es) | 2003-03-07 | 2005-10-18 | Schering Corp | Compuestos de azetidinona sustituidos, formulaciones y usos de los mismos para el tratamiento de hipercolesterolemia. |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4602003A (en) * | 1982-05-17 | 1986-07-22 | Medical Research Foundation Of Oregon | Synthetic compounds to inhibit intestinal absorption of cholesterol in the treatment of hypercholesterolemia |
| US4602005A (en) * | 1982-05-17 | 1986-07-22 | Medical Research Foundation Of Oregon | Tigogenin cellobioside for treating hypercholesterolemia and atherosclerosis |
-
1992
- 1992-10-15 JP JP5510090A patent/JPH0826064B2/ja not_active Expired - Lifetime
- 1992-10-15 AU AU27758/92A patent/AU659506B2/en not_active Ceased
- 1992-10-15 CA CA002123684A patent/CA2123684A1/en not_active Abandoned
- 1992-10-15 EP EP92921860A patent/EP0619822A1/en not_active Withdrawn
- 1992-10-15 HU HU9401374A patent/HUT67035A/hu unknown
- 1992-10-15 WO PCT/US1992/008638 patent/WO1993011150A1/en not_active Application Discontinuation
- 1992-10-15 FI FI942394A patent/FI942394L/fi not_active Application Discontinuation
- 1992-10-20 TW TW081108325A patent/TW232699B/zh active
- 1992-11-19 IL IL103797A patent/IL103797A0/xx unknown
- 1992-11-23 PT PT101088A patent/PT101088A/pt not_active Application Discontinuation
- 1992-11-24 NZ NZ245244A patent/NZ245244A/en unknown
- 1992-11-24 MX MX9206761A patent/MX9206761A/es not_active IP Right Cessation
- 1992-11-24 ZA ZA929081A patent/ZA929081B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP0619822A1 (en) | 1994-10-19 |
| HUT67035A (en) | 1995-01-30 |
| MX9206761A (es) | 1995-01-31 |
| WO1993011150A1 (en) | 1993-06-10 |
| TW232699B (cs) | 1994-10-21 |
| FI942394A7 (fi) | 1994-05-24 |
| NZ245244A (en) | 1995-04-27 |
| IL103797A0 (en) | 1993-04-04 |
| JPH0826064B2 (ja) | 1996-03-13 |
| PT101088A (pt) | 1994-02-28 |
| ZA929081B (en) | 1994-05-24 |
| FI942394A0 (fi) | 1994-05-24 |
| AU2775892A (en) | 1993-06-28 |
| AU659506B2 (en) | 1995-05-18 |
| JPH06510794A (ja) | 1994-12-01 |
| FI942394L (fi) | 1994-05-24 |
| HU9401374D0 (en) | 1994-08-29 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request | ||
| FZDE | Discontinued |