FI942394L - Menetelmä steroidiperasyyliglykosidien valmistamiseksi - Google Patents

Menetelmä steroidiperasyyliglykosidien valmistamiseksi Download PDF

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Publication number
FI942394L
FI942394L FI942394A FI942394A FI942394L FI 942394 L FI942394 L FI 942394L FI 942394 A FI942394 A FI 942394A FI 942394 A FI942394 A FI 942394A FI 942394 L FI942394 L FI 942394L
Authority
FI
Finland
Prior art keywords
steroid
preparation
peracyl
glycosides
peracyl glycosides
Prior art date
Application number
FI942394A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI942394A7 (fi
FI942394A0 (fi
Inventor
Douglas John M Allen
Frank Robert Busch
John Francis Lambert
Russell James Shine
Stanley Walter Walinsky
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI942394A7 publication Critical patent/FI942394A7/fi
Publication of FI942394A0 publication Critical patent/FI942394A0/fi
Publication of FI942394L publication Critical patent/FI942394L/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005Oxygen-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
FI942394A 1991-11-25 1992-10-15 Menetelmä steroidiperasyyliglykosidien valmistamiseksi FI942394L (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US79757491A 1991-11-25 1991-11-25
PCT/US1992/008638 WO1993011150A1 (en) 1991-11-25 1992-10-15 Method for making steroidal peracyl glycosides

Publications (3)

Publication Number Publication Date
FI942394A7 FI942394A7 (fi) 1994-05-24
FI942394A0 FI942394A0 (fi) 1994-05-24
FI942394L true FI942394L (fi) 1994-05-24

Family

ID=25171219

Family Applications (1)

Application Number Title Priority Date Filing Date
FI942394A FI942394L (fi) 1991-11-25 1992-10-15 Menetelmä steroidiperasyyliglykosidien valmistamiseksi

Country Status (13)

Country Link
EP (1) EP0619822A1 (cs)
JP (1) JPH0826064B2 (cs)
AU (1) AU659506B2 (cs)
CA (1) CA2123684A1 (cs)
FI (1) FI942394L (cs)
HU (1) HUT67035A (cs)
IL (1) IL103797A0 (cs)
MX (1) MX9206761A (cs)
NZ (1) NZ245244A (cs)
PT (1) PT101088A (cs)
TW (1) TW232699B (cs)
WO (1) WO1993011150A1 (cs)
ZA (1) ZA929081B (cs)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5563259A (en) * 1992-06-26 1996-10-08 Pfizer Inc. Process for making β-O-cellobiosyl steroid derivatives and trimethyl silyl steroid intermediates used therein
US5606041A (en) * 1992-06-26 1997-02-25 Pfizer Inc. Process for steroidal peracyl glycosides
JPH07504921A (ja) * 1992-06-26 1995-06-01 フアイザー・インコーポレイテツド 高コレステロール血症を治療するためのステロイドグリコシド
JPH08504830A (ja) * 1993-04-28 1996-05-28 フアイザー・インコーポレイテツド スピロスタニルグリコシド結晶質一水塩
US5502038A (en) * 1993-06-21 1996-03-26 Medical Research Foundation Of Oregon Cholesterol sequestrant glycosides that inhibit intestinal cholesterol absorption
CA2180148A1 (en) * 1993-12-28 1995-07-06 Michael Paul Deninno Hypocholesterolemic agents
WO1996038466A1 (en) * 1995-05-29 1996-12-05 Pfizer Inc. Steroidal glycosides
US5756470A (en) * 1996-10-29 1998-05-26 Schering Corporation Sugar-substituted 2-azetidinones useful as hypocholesterolemic agents
US6982251B2 (en) 2000-12-20 2006-01-03 Schering Corporation Substituted 2-azetidinones useful as hypocholesterolemic agents
BR0206654A (pt) 2001-01-26 2004-02-25 Schering Corp Combinações de ativador(es) de receptor ativado por proliferação de peroxisoma (ppar) e inibidor(es) de absorção de esterol e tratamentos para indicações vasculares
WO2002058696A2 (en) 2001-01-26 2002-08-01 Schering Corporation The use of substituted azetidinone compounds for the treatment of sitosterolemia
US7071181B2 (en) 2001-01-26 2006-07-04 Schering Corporation Methods and therapeutic combinations for the treatment of diabetes using sterol absorption inhibitors
DE60216300T2 (de) 2001-09-21 2007-06-28 Schering Corp. Behandlung von xanthom mittels azetidinon-derivate als hemmer der sterol absorption
US7053080B2 (en) 2001-09-21 2006-05-30 Schering Corporation Methods and therapeutic combinations for the treatment of obesity using sterol absorption inhibitors
US7056906B2 (en) 2001-09-21 2006-06-06 Schering Corporation Combinations of hormone replacement therapy composition(s) and sterol absorption inhibitor(s) and treatments for vascular conditions in post-menopausal women
US7560449B2 (en) 2002-11-06 2009-07-14 Schering Corporation Methods and therapeutic combinations for the treatment of demyelination
ES2311806T3 (es) 2003-03-07 2009-02-16 Schering Corporation Compuesto de azetidinona sustituidos, fornulaciones y usos de los mismos para el tratamiento de hipercolesterolemia.
US7459442B2 (en) 2003-03-07 2008-12-02 Schering Corporation Substituted azetidinone compounds, processes for preparing the same, formulations and uses thereof
ES2318274T3 (es) 2003-03-07 2009-05-01 Schering Corporation Compuestos de azetidinona sustituida, formulaciones y uso de los mismos para el tratamiento de hipercolesterolemia.
MXPA05009502A (es) 2003-03-07 2005-10-18 Schering Corp Compuestos de azetidinona sustituidos, formulaciones y usos de los mismos para el tratamiento de hipercolesterolemia.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4602003A (en) * 1982-05-17 1986-07-22 Medical Research Foundation Of Oregon Synthetic compounds to inhibit intestinal absorption of cholesterol in the treatment of hypercholesterolemia
US4602005A (en) * 1982-05-17 1986-07-22 Medical Research Foundation Of Oregon Tigogenin cellobioside for treating hypercholesterolemia and atherosclerosis

Also Published As

Publication number Publication date
EP0619822A1 (en) 1994-10-19
CA2123684A1 (en) 1993-06-10
HUT67035A (en) 1995-01-30
MX9206761A (es) 1995-01-31
WO1993011150A1 (en) 1993-06-10
TW232699B (cs) 1994-10-21
FI942394A7 (fi) 1994-05-24
NZ245244A (en) 1995-04-27
IL103797A0 (en) 1993-04-04
JPH0826064B2 (ja) 1996-03-13
PT101088A (pt) 1994-02-28
ZA929081B (en) 1994-05-24
FI942394A0 (fi) 1994-05-24
AU2775892A (en) 1993-06-28
AU659506B2 (en) 1995-05-18
JPH06510794A (ja) 1994-12-01
HU9401374D0 (en) 1994-08-29

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Legal Events

Date Code Title Description
FD Application lapsed