AU659506B2 - Method for making steroidal peracyl glycosides - Google Patents

Method for making steroidal peracyl glycosides Download PDF

Info

Publication number
AU659506B2
AU659506B2 AU27758/92A AU2775892A AU659506B2 AU 659506 B2 AU659506 B2 AU 659506B2 AU 27758/92 A AU27758/92 A AU 27758/92A AU 2775892 A AU2775892 A AU 2775892A AU 659506 B2 AU659506 B2 AU 659506B2
Authority
AU
Australia
Prior art keywords
zinc
tigogenin
recited
cellobioside
international
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU27758/92A
Other languages
English (en)
Other versions
AU2775892A (en
Inventor
Douglas John M Allen
Frank Robert Busch
John Francis Lambert
Russell James Shine
Stanley Walter Walinsky
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp SRL
Original Assignee
Pfizer Corp Belgium
Pfizer Corp SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp Belgium, Pfizer Corp SRL filed Critical Pfizer Corp Belgium
Publication of AU2775892A publication Critical patent/AU2775892A/en
Application granted granted Critical
Publication of AU659506B2 publication Critical patent/AU659506B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005Oxygen-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AU27758/92A 1991-11-25 1992-10-15 Method for making steroidal peracyl glycosides Ceased AU659506B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US79757491A 1991-11-25 1991-11-25
US797574 1991-11-25
PCT/US1992/008638 WO1993011150A1 (en) 1991-11-25 1992-10-15 Method for making steroidal peracyl glycosides

Publications (2)

Publication Number Publication Date
AU2775892A AU2775892A (en) 1993-06-28
AU659506B2 true AU659506B2 (en) 1995-05-18

Family

ID=25171219

Family Applications (1)

Application Number Title Priority Date Filing Date
AU27758/92A Ceased AU659506B2 (en) 1991-11-25 1992-10-15 Method for making steroidal peracyl glycosides

Country Status (13)

Country Link
EP (1) EP0619822A1 (cs)
JP (1) JPH0826064B2 (cs)
AU (1) AU659506B2 (cs)
CA (1) CA2123684A1 (cs)
FI (1) FI942394L (cs)
HU (1) HUT67035A (cs)
IL (1) IL103797A0 (cs)
MX (1) MX9206761A (cs)
NZ (1) NZ245244A (cs)
PT (1) PT101088A (cs)
TW (1) TW232699B (cs)
WO (1) WO1993011150A1 (cs)
ZA (1) ZA929081B (cs)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5563259A (en) * 1992-06-26 1996-10-08 Pfizer Inc. Process for making β-O-cellobiosyl steroid derivatives and trimethyl silyl steroid intermediates used therein
US5606041A (en) * 1992-06-26 1997-02-25 Pfizer Inc. Process for steroidal peracyl glycosides
JPH07504921A (ja) * 1992-06-26 1995-06-01 フアイザー・インコーポレイテツド 高コレステロール血症を治療するためのステロイドグリコシド
JPH08504830A (ja) * 1993-04-28 1996-05-28 フアイザー・インコーポレイテツド スピロスタニルグリコシド結晶質一水塩
US5502038A (en) * 1993-06-21 1996-03-26 Medical Research Foundation Of Oregon Cholesterol sequestrant glycosides that inhibit intestinal cholesterol absorption
CA2180148A1 (en) * 1993-12-28 1995-07-06 Michael Paul Deninno Hypocholesterolemic agents
WO1996038466A1 (en) * 1995-05-29 1996-12-05 Pfizer Inc. Steroidal glycosides
US5756470A (en) * 1996-10-29 1998-05-26 Schering Corporation Sugar-substituted 2-azetidinones useful as hypocholesterolemic agents
US6982251B2 (en) 2000-12-20 2006-01-03 Schering Corporation Substituted 2-azetidinones useful as hypocholesterolemic agents
BR0206654A (pt) 2001-01-26 2004-02-25 Schering Corp Combinações de ativador(es) de receptor ativado por proliferação de peroxisoma (ppar) e inibidor(es) de absorção de esterol e tratamentos para indicações vasculares
WO2002058696A2 (en) 2001-01-26 2002-08-01 Schering Corporation The use of substituted azetidinone compounds for the treatment of sitosterolemia
US7071181B2 (en) 2001-01-26 2006-07-04 Schering Corporation Methods and therapeutic combinations for the treatment of diabetes using sterol absorption inhibitors
DE60216300T2 (de) 2001-09-21 2007-06-28 Schering Corp. Behandlung von xanthom mittels azetidinon-derivate als hemmer der sterol absorption
US7053080B2 (en) 2001-09-21 2006-05-30 Schering Corporation Methods and therapeutic combinations for the treatment of obesity using sterol absorption inhibitors
US7056906B2 (en) 2001-09-21 2006-06-06 Schering Corporation Combinations of hormone replacement therapy composition(s) and sterol absorption inhibitor(s) and treatments for vascular conditions in post-menopausal women
US7560449B2 (en) 2002-11-06 2009-07-14 Schering Corporation Methods and therapeutic combinations for the treatment of demyelination
ES2311806T3 (es) 2003-03-07 2009-02-16 Schering Corporation Compuesto de azetidinona sustituidos, fornulaciones y usos de los mismos para el tratamiento de hipercolesterolemia.
US7459442B2 (en) 2003-03-07 2008-12-02 Schering Corporation Substituted azetidinone compounds, processes for preparing the same, formulations and uses thereof
ES2318274T3 (es) 2003-03-07 2009-05-01 Schering Corporation Compuestos de azetidinona sustituida, formulaciones y uso de los mismos para el tratamiento de hipercolesterolemia.
MXPA05009502A (es) 2003-03-07 2005-10-18 Schering Corp Compuestos de azetidinona sustituidos, formulaciones y usos de los mismos para el tratamiento de hipercolesterolemia.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4602003A (en) * 1982-05-17 1986-07-22 Medical Research Foundation Of Oregon Synthetic compounds to inhibit intestinal absorption of cholesterol in the treatment of hypercholesterolemia
US4602005A (en) * 1982-05-17 1986-07-22 Medical Research Foundation Of Oregon Tigogenin cellobioside for treating hypercholesterolemia and atherosclerosis

Also Published As

Publication number Publication date
EP0619822A1 (en) 1994-10-19
CA2123684A1 (en) 1993-06-10
HUT67035A (en) 1995-01-30
MX9206761A (es) 1995-01-31
WO1993011150A1 (en) 1993-06-10
TW232699B (cs) 1994-10-21
FI942394A7 (fi) 1994-05-24
NZ245244A (en) 1995-04-27
IL103797A0 (en) 1993-04-04
JPH0826064B2 (ja) 1996-03-13
PT101088A (pt) 1994-02-28
ZA929081B (en) 1994-05-24
FI942394A0 (fi) 1994-05-24
AU2775892A (en) 1993-06-28
JPH06510794A (ja) 1994-12-01
FI942394L (fi) 1994-05-24
HU9401374D0 (en) 1994-08-29

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