CA1300133C - Benzimidazoles et imidazopyridines sulfonamides, leur preparation et leurapplication en tant que medicaments - Google Patents
Benzimidazoles et imidazopyridines sulfonamides, leur preparation et leurapplication en tant que medicamentsInfo
- Publication number
- CA1300133C CA1300133C CA000534593A CA534593A CA1300133C CA 1300133 C CA1300133 C CA 1300133C CA 000534593 A CA000534593 A CA 000534593A CA 534593 A CA534593 A CA 534593A CA 1300133 C CA1300133 C CA 1300133C
- Authority
- CA
- Canada
- Prior art keywords
- radical
- benzimidazole
- dioxide
- nitro
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/28—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
- C07D513/14—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8605721A FR2597478B1 (fr) | 1986-04-21 | 1986-04-21 | Benzimidazoles et imidazopyridines sulfonamides, leur preparation et leur application en tant que medicaments. |
| FR8605721 | 1986-04-21 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA1300133C true CA1300133C (fr) | 1992-05-05 |
Family
ID=9334440
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA000534593A Expired - Lifetime CA1300133C (fr) | 1986-04-21 | 1987-04-13 | Benzimidazoles et imidazopyridines sulfonamides, leur preparation et leurapplication en tant que medicaments |
Country Status (20)
| Country | Link |
|---|---|
| US (2) | US4933338A (forum.php) |
| EP (1) | EP0246126A1 (forum.php) |
| JP (1) | JPH0643404B2 (forum.php) |
| KR (1) | KR930003613B1 (forum.php) |
| CN (1) | CN87102916A (forum.php) |
| AU (1) | AU608511B2 (forum.php) |
| BR (1) | BR8701897A (forum.php) |
| CA (1) | CA1300133C (forum.php) |
| DD (1) | DD297817A5 (forum.php) |
| DK (1) | DK185487A (forum.php) |
| ES (1) | ES2005158A6 (forum.php) |
| FR (1) | FR2597478B1 (forum.php) |
| HU (1) | HUT63151A (forum.php) |
| IN (1) | IN167204B (forum.php) |
| NO (1) | NO871643L (forum.php) |
| PL (1) | PL156736B1 (forum.php) |
| PT (1) | PT84724B (forum.php) |
| RU (1) | RU1813087C (forum.php) |
| YU (1) | YU46193B (forum.php) |
| ZA (1) | ZA872739B (forum.php) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL71664A (en) * | 1983-05-03 | 1987-11-30 | Byk Gulden Lomberg Chem Fab | Fluoroalkoxy compounds,process for their preparation and pharmaceutical compositions containing the same |
| KR950001015B1 (ko) * | 1986-01-10 | 1995-02-07 | 닛뽕 케미화 가부시끼가이샤 | 술폭시드 유도체의 제조방법 |
| US5162317A (en) * | 1988-05-12 | 1992-11-10 | Esai Co., Ltd. | Pyridinium salt and pharmacological composition containing the same |
| NZ270985A (en) | 1994-04-29 | 1997-06-24 | Lilly Co Eli | Substituted benzimidazole derivatives; medicaments and preparation of medicaments |
| EP1086094A1 (en) * | 1998-05-23 | 2001-03-28 | Byk Gulden Lomberg Chemische Fabrik GmbH | Quinoline-aminomethyl-pyridyl derivatives with anti-helicobacter activity |
| CN1295561A (zh) | 1998-06-03 | 2001-05-16 | Gpinil控股公司 | N－杂环羧酸或羧酸等排物的n－结合氨磺酰 |
| WO2004032861A2 (en) * | 2002-10-11 | 2004-04-22 | Bristol-Myers Squibb Company | Hexahydro-benzimidazolone compounds useful as anti-inflammatory agents |
| CN101497616B (zh) * | 2008-01-30 | 2011-05-18 | 山东轩竹医药科技有限公司 | 含有氨基氧基取代的吡啶的咪唑并吡啶的化合物 |
| CN110551145B (zh) * | 2019-10-24 | 2022-08-05 | 江苏师范大学 | 一类呋喃并香豆素-Tröger’s Base衍生物及其合成方法与应用 |
| KR20250134151A (ko) * | 2022-12-16 | 2025-09-09 | 텐비 테라퓨틱스, 인크. | 화합물, 조성물 및 방법 |
| CN118373826A (zh) * | 2024-04-19 | 2024-07-23 | 常州大学 | 一种合成吲哚并1,4-二氮八元杂环类化合物的方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE502319A (forum.php) * | 1950-04-04 | |||
| US2603649A (en) * | 1950-04-04 | 1952-07-15 | American Cyanamid Co | Heterocyclic sulfonamides and method of preparing the same |
| GB833049A (en) * | 1957-04-04 | 1960-04-21 | Omikron Gagliardi Soc Di Fatto | Improvements in the preparation of heterocyclic sulfonamides |
| DE2726625A1 (de) * | 1976-06-25 | 1977-12-29 | Ciba Geigy Ag | Verfahren zum flammfestmachen von polyesterfasermaterialien |
| GB8316645D0 (en) * | 1983-06-18 | 1983-07-20 | Wyeth John & Brother Ltd | Heterocyclic compounds |
-
1986
- 1986-04-21 FR FR8605721A patent/FR2597478B1/fr not_active Expired
-
1987
- 1987-04-09 IN IN305/DEL/87A patent/IN167204B/en unknown
- 1987-04-10 DK DK185487A patent/DK185487A/da not_active Application Discontinuation
- 1987-04-13 AU AU71438/87A patent/AU608511B2/en not_active Ceased
- 1987-04-13 CA CA000534593A patent/CA1300133C/fr not_active Expired - Lifetime
- 1987-04-14 ES ES8701081A patent/ES2005158A6/es not_active Expired
- 1987-04-15 US US07/038,874 patent/US4933338A/en not_active Expired - Fee Related
- 1987-04-16 ZA ZA872739A patent/ZA872739B/xx unknown
- 1987-04-16 EP EP87400875A patent/EP0246126A1/fr not_active Withdrawn
- 1987-04-17 HU HU871716A patent/HUT63151A/hu unknown
- 1987-04-20 RU SU874202461A patent/RU1813087C/ru active
- 1987-04-20 DD DD87301968A patent/DD297817A5/de not_active IP Right Cessation
- 1987-04-20 PT PT84724A patent/PT84724B/pt not_active IP Right Cessation
- 1987-04-21 YU YU72387A patent/YU46193B/sh unknown
- 1987-04-21 JP JP62098483A patent/JPH0643404B2/ja not_active Expired - Lifetime
- 1987-04-21 BR BR8701897A patent/BR8701897A/pt unknown
- 1987-04-21 KR KR1019870003936A patent/KR930003613B1/ko not_active Expired - Fee Related
- 1987-04-21 CN CN87102916A patent/CN87102916A/zh active Pending
- 1987-04-21 NO NO871643A patent/NO871643L/no unknown
- 1987-04-21 PL PL1987265299A patent/PL156736B1/pl unknown
-
1989
- 1989-04-28 US US07/344,966 patent/US4943570A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| NO871643D0 (no) | 1987-04-21 |
| JPS62289568A (ja) | 1987-12-16 |
| EP0246126A1 (fr) | 1987-11-19 |
| DD297817A5 (de) | 1992-01-23 |
| YU46193B (sh) | 1993-05-28 |
| BR8701897A (pt) | 1988-02-02 |
| CN87102916A (zh) | 1988-04-27 |
| YU72387A (en) | 1989-02-28 |
| PL156736B1 (pl) | 1992-04-30 |
| US4943570A (en) | 1990-07-24 |
| RU1813087C (ru) | 1993-04-30 |
| US4933338A (en) | 1990-06-12 |
| FR2597478A1 (fr) | 1987-10-23 |
| HUT63151A (en) | 1993-07-28 |
| ZA872739B (en) | 1987-12-30 |
| JPH0643404B2 (ja) | 1994-06-08 |
| PT84724A (fr) | 1987-05-01 |
| DK185487A (da) | 1987-10-22 |
| NO871643L (no) | 1987-10-22 |
| KR930003613B1 (ko) | 1993-05-08 |
| AU608511B2 (en) | 1991-04-11 |
| KR870010050A (ko) | 1987-11-30 |
| IN167204B (forum.php) | 1990-09-22 |
| DK185487D0 (da) | 1987-04-10 |
| AU7143887A (en) | 1987-10-22 |
| PT84724B (pt) | 1989-12-29 |
| FR2597478B1 (fr) | 1988-12-16 |
| PL265299A1 (en) | 1988-07-21 |
| ES2005158A6 (es) | 1989-03-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MKLA | Lapsed |