CA1144919A - Derives de vinyl-3 cephalosporines, et leur preparation - Google Patents

Derives de vinyl-3 cephalosporines, et leur preparation

Info

Publication number
CA1144919A
CA1144919A CA000352324A CA352324A CA1144919A CA 1144919 A CA1144919 A CA 1144919A CA 000352324 A CA000352324 A CA 000352324A CA 352324 A CA352324 A CA 352324A CA 1144919 A CA1144919 A CA 1144919A
Authority
CA
Canada
Prior art keywords
radical
general formula
thia
aza
oxo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA000352324A
Other languages
English (en)
French (fr)
Inventor
Daniel Farge
Jean-Francois Peyronel
Claude Moutonnier
Pierre Le Roy
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Rhone Poulenc Industries SA
Original Assignee
Rhone Poulenc Industries SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Industries SA filed Critical Rhone Poulenc Industries SA
Application granted granted Critical
Publication of CA1144919A publication Critical patent/CA1144919A/fr
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/02Nutrients, e.g. vitamins, minerals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Nutrition Science (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CA000352324A 1979-05-23 1980-05-21 Derives de vinyl-3 cephalosporines, et leur preparation Expired CA1144919A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR7913096 1979-05-23
FR7913096A FR2457296A1 (fr) 1979-05-23 1979-05-23 Nouveaux derives de vinyl-3 cephalosporines et leur preparation

Publications (1)

Publication Number Publication Date
CA1144919A true CA1144919A (fr) 1983-04-19

Family

ID=9225762

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000352324A Expired CA1144919A (fr) 1979-05-23 1980-05-21 Derives de vinyl-3 cephalosporines, et leur preparation

Country Status (31)

Country Link
US (1) US4307233A (US20100170793A1-20100708-C00006.png)
JP (1) JPS55154981A (US20100170793A1-20100708-C00006.png)
AT (1) AT369375B (US20100170793A1-20100708-C00006.png)
AU (1) AU534806B2 (US20100170793A1-20100708-C00006.png)
BE (1) BE883416A (US20100170793A1-20100708-C00006.png)
CA (1) CA1144919A (US20100170793A1-20100708-C00006.png)
CH (1) CH645379A5 (US20100170793A1-20100708-C00006.png)
CS (1) CS244405B2 (US20100170793A1-20100708-C00006.png)
DD (1) DD150899A5 (US20100170793A1-20100708-C00006.png)
DE (1) DE3019462A1 (US20100170793A1-20100708-C00006.png)
DK (1) DK222080A (US20100170793A1-20100708-C00006.png)
ES (1) ES491687A0 (US20100170793A1-20100708-C00006.png)
FI (1) FI801641A (US20100170793A1-20100708-C00006.png)
FR (1) FR2457296A1 (US20100170793A1-20100708-C00006.png)
GB (1) GB2051062B (US20100170793A1-20100708-C00006.png)
GR (1) GR68426B (US20100170793A1-20100708-C00006.png)
HU (1) HU185890B (US20100170793A1-20100708-C00006.png)
IE (1) IE49814B1 (US20100170793A1-20100708-C00006.png)
IL (1) IL60139A (US20100170793A1-20100708-C00006.png)
IT (1) IT1140974B (US20100170793A1-20100708-C00006.png)
LU (1) LU82477A1 (US20100170793A1-20100708-C00006.png)
NL (1) NL8003023A (US20100170793A1-20100708-C00006.png)
NO (1) NO801502L (US20100170793A1-20100708-C00006.png)
NZ (1) NZ193799A (US20100170793A1-20100708-C00006.png)
PH (1) PH15946A (US20100170793A1-20100708-C00006.png)
PL (1) PL126481B1 (US20100170793A1-20100708-C00006.png)
PT (1) PT71276A (US20100170793A1-20100708-C00006.png)
SE (1) SE451072B (US20100170793A1-20100708-C00006.png)
SU (1) SU1031409A3 (US20100170793A1-20100708-C00006.png)
YU (1) YU136880A (US20100170793A1-20100708-C00006.png)
ZA (1) ZA803038B (US20100170793A1-20100708-C00006.png)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL58717A (en) * 1978-11-15 1983-05-15 Glaxo Group Ltd Derivatives of(6r,7r)-7-((z)-2-(2-aminothiazol-4-yl)-2-(carboxy-(lower alkyl or cycloalkyl)oxyimino)acetamido)-3-(2-alkyl-pyrazolium-1-ylmethyl)ceph-3-em-4-carboxylate,process for their preparation and pharmaceutical compositions comprising them
FR2494279A1 (fr) * 1980-11-20 1982-05-21 Rhone Poulenc Ind Nouvelles oxacephalosporines, leur preparation et les medicaments qui les contiennent
FR2494280A1 (fr) * 1980-11-20 1982-05-21 Rhone Poulenc Ind Nouveaux derives de la cephalosporine et leur preparation
FR2494275A2 (fr) * 1980-11-20 1982-05-21 Rhone Poulenc Ind Nouveaux derives de vinyl-3 cephalosporines et leur preparation
FR2505334A1 (fr) * 1981-05-11 1982-11-12 Rhone Poulenc Sante Nouvelles oxacephalosporines et leur preparation
FR2511372A1 (fr) * 1981-08-17 1983-02-18 Rhone Poulenc Sante Nouveaux derives de la cephalosporine et leur preparation
US4486586A (en) * 1983-02-10 1984-12-04 Bristol-Myers Company Cephalosporin derivatives
US4560749A (en) * 1983-11-18 1985-12-24 Eli Lilly And Company Cephem-3-imidates and 3-amidines
US4708955A (en) * 1985-06-24 1987-11-24 Bristol-Myers Company 3-(substituted)propenyl-7-aminothiazol-ylcephalosporanic acids and esters thereof
US4874856A (en) * 1985-06-24 1989-10-17 Bristol-Myers Company 3-(substituted)propenyl-7-(aminothiazolylacetamido) ceph-3-em-4-carboxylic acids and esters thereof
ATE92927T1 (de) * 1986-04-14 1993-08-15 Banyu Pharma Co Ltd 1-carboxy-1-vinyloxyiminoaminothiazolcephalosporin-derivate und deren herstellung.
DK0841339T3 (da) 1996-11-06 2007-07-02 Basilea Pharmaceutica Ag Vinylpyrrolidinon-cephalosporinderivater
WO2009049086A1 (en) 2007-10-09 2009-04-16 Larry Sutton Broad spectrum beta-lactamase inhibitors
JP6403289B2 (ja) 2013-03-12 2018-10-10 グラディウス ファーマシューティカルズ コーポレーションGladius Pharmaceuticals Corporation 誘導体化3−スチリル−セファロスポリン

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4065620A (en) * 1971-06-14 1977-12-27 Eli Lilly And Company 3-(Substituted) vinyl cephalosporins
GB1463077A (en) * 1973-04-19 1977-02-02 Glaxo Lab Ltd 7-substituted-ethyl-cephalosporin derivatives
CH617703A5 (en) * 1973-12-21 1980-06-13 Glaxo Operations Ltd Process for the preparation of the syn-isomer or of a mixture of syn- and anti-isomers of novel antibiotically active 7 beta -acylamino-ceph-3-em-4-carboxylic acids
US4095021A (en) * 1973-12-21 1978-06-13 Glaxo Laboratories Limited 3-Carbamoyloxymethyl or N-methyl-carbamoyloxymethyl-7-[2-carboxymethoxyimino-2-(fur-2-yl or thien-2-yl)acetamido]ceph-3-em-4-carboxylic acids and derivatives thereof
JPS5129492A (en) * 1974-09-04 1976-03-12 Sankyo Co Sefuarosuhorinjudotai no seiho
DK154939C (da) * 1974-12-19 1989-06-12 Takeda Chemical Industries Ltd Analogifremgangsmaade til fremstilling af thiazolylacetamido-cephemforbindelser eller farmaceutisk acceptable salte eller estere deraf
JPS5253890A (en) * 1975-10-14 1977-04-30 Syntex Inc Production of cephalosporin type compound
PT71654B (en) * 1979-08-15 1982-01-22 Merck & Co Inc Process for preparing allylsulfoxide enzyme inhibitor

Also Published As

Publication number Publication date
GB2051062B (en) 1983-10-12
NZ193799A (en) 1983-03-15
AT369375B (de) 1982-12-27
ES8102136A1 (es) 1980-12-16
SE8003821L (sv) 1980-11-24
DE3019462A1 (de) 1980-12-04
YU136880A (en) 1983-04-30
CS244405B2 (en) 1986-07-17
ZA803038B (en) 1981-05-27
IT8022243A0 (it) 1980-05-21
GB2051062A (en) 1981-01-14
PT71276A (fr) 1980-06-01
PL126481B1 (en) 1983-08-31
JPH0246595B2 (US20100170793A1-20100708-C00006.png) 1990-10-16
IT1140974B (it) 1986-10-10
JPS55154981A (en) 1980-12-02
SE451072B (sv) 1987-08-31
HU185890B (en) 1985-04-28
NL8003023A (nl) 1980-11-25
AU5859580A (en) 1980-11-27
CS354380A2 (US20100170793A1-20100708-C00006.png) 1985-09-17
NO801502L (no) 1980-11-24
IL60139A0 (en) 1980-07-31
SU1031409A3 (ru) 1983-07-23
PH15946A (en) 1983-04-29
BE883416A (fr) 1980-11-21
CH645379A5 (fr) 1984-09-28
PL224391A1 (US20100170793A1-20100708-C00006.png) 1981-02-13
IE49814B1 (en) 1985-12-25
AU534806B2 (en) 1984-02-16
IL60139A (en) 1984-04-30
DK222080A (da) 1980-11-24
LU82477A1 (fr) 1980-12-16
FR2457296B1 (US20100170793A1-20100708-C00006.png) 1982-02-05
FI801641A (fi) 1980-11-24
ATA270980A (de) 1982-05-15
FR2457296A1 (fr) 1980-12-19
US4307233A (en) 1981-12-22
DD150899A5 (de) 1981-09-23
GR68426B (US20100170793A1-20100708-C00006.png) 1981-12-30
ES491687A0 (es) 1980-12-16
IE801062L (en) 1980-11-23

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Legal Events

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