BRPI9710537B8 - derivados da eritromicina, composições farmacêuticas, bem como processo para preparação dos mesmos. - Google Patents

derivados da eritromicina, composições farmacêuticas, bem como processo para preparação dos mesmos.

Info

Publication number
BRPI9710537B8
BRPI9710537B8 BRPI9710537A BR9710537A BRPI9710537B8 BR PI9710537 B8 BRPI9710537 B8 BR PI9710537B8 BR PI9710537 A BRPI9710537 A BR PI9710537A BR 9710537 A BR9710537 A BR 9710537A BR PI9710537 B8 BRPI9710537 B8 BR PI9710537B8
Authority
BR
Brazil
Prior art keywords
preparing
processes
well
pharmaceutical compositions
erythromycin derivatives
Prior art date
Application number
BRPI9710537A
Other languages
English (en)
Other versions
BR9710537B1 (pt
BR9710537A (pt
Inventor
Denis Alexis
Agouridas Constantin
Chantot Jean-Francois
Pejac Jean-Marie
Original Assignee
Aventis Pharma Sa
Hoechst Marion Roussel
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa, Hoechst Marion Roussel filed Critical Aventis Pharma Sa
Publication of BR9710537A publication Critical patent/BR9710537A/pt
Publication of BR9710537B1 publication Critical patent/BR9710537B1/pt
Publication of BRPI9710537B8 publication Critical patent/BRPI9710537B8/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

patente de invenção: <b>"novos derivados da eritromicina, seu processo de preparo e sua aplicação como medicamentos"<d>. compostos de fórmula (i), nos quais r é um hidrogênio, um alquila, eventualmente substituído por um halogênio ou um radical (ch~ 2~)~ m~ar ou um radical (a), nos quais m é um número inteiro (1-8), n e p, idênticos ou diferentes, representam um número inteiro (0-6), a e b, idênticos ou diferentes representam um hidrogênio ou um halogênio ou um alquila e ar representa um arila ou heteroarila, e z um hidrogênio ou o resto de um ácido carboxílico, processo de preparo e aplicação como medicamentos.
BRPI9710537A 1996-07-24 1997-07-23 derivados da eritromicina, composições farmacêuticas, bem como processo para preparação dos mesmos. BRPI9710537B8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9609285A FR2751656B1 (fr) 1996-07-24 1996-07-24 Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
PCT/FR1997/001372 WO1998003530A1 (fr) 1996-07-24 1997-07-23 Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments

Publications (3)

Publication Number Publication Date
BR9710537A BR9710537A (pt) 1999-08-17
BR9710537B1 BR9710537B1 (pt) 2013-07-23
BRPI9710537B8 true BRPI9710537B8 (pt) 2017-03-07

Family

ID=9494403

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI9710537A BRPI9710537B8 (pt) 1996-07-24 1997-07-23 derivados da eritromicina, composições farmacêuticas, bem como processo para preparação dos mesmos.

Country Status (28)

Country Link
US (1) US6162793A (pt)
EP (1) EP0931088B1 (pt)
JP (1) JP4267700B2 (pt)
KR (1) KR100458240B1 (pt)
CN (1) CN1178951C (pt)
AP (1) AP1078A (pt)
AT (1) ATE225798T1 (pt)
AU (1) AU710478B2 (pt)
BG (1) BG62812B1 (pt)
BR (1) BRPI9710537B8 (pt)
CA (1) CA2261098C (pt)
CZ (1) CZ292561B6 (pt)
DE (1) DE69716284T2 (pt)
DK (1) DK0931088T3 (pt)
EA (1) EA002168B1 (pt)
ES (1) ES2181016T3 (pt)
FR (1) FR2751656B1 (pt)
HU (1) HUP9903424A3 (pt)
IL (2) IL128182A0 (pt)
NO (1) NO313332B1 (pt)
NZ (1) NZ333559A (pt)
PL (1) PL186297B1 (pt)
PT (1) PT931088E (pt)
SK (1) SK283713B6 (pt)
TR (1) TR199900095T2 (pt)
UA (1) UA48244C2 (pt)
WO (1) WO1998003530A1 (pt)
YU (1) YU3099A (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2781484B1 (fr) * 1998-07-21 2001-08-10 Hoechst Marion Roussel Inc Nouveaux derives de la 6-deoxy erythromycine, leur procede de preparation et leur application comme medicaments
WO2000034297A1 (en) 1998-12-10 2000-06-15 Pfizer Products Inc. Carbamate and carbazate ketolide antibiotics
EE200100394A (et) 1999-01-27 2002-10-15 Pfizer Products Inc. Ketoliidsed antibiootikumid
MXPA01010524A (es) * 1999-04-16 2002-03-14 Kosan Biosciences Inc Agentes macrolidos anti-infecciosos.
OA11945A (en) * 1999-05-24 2006-04-13 Pfizer Prod Inc 13-Methyl erythromycin derivatives.
CL2004000409A1 (es) * 2003-03-03 2005-01-07 Vertex Pharma Compuestos derivados de 2-(cilo sustituido)-1-(amino u oxi sustituido)-quinazolina, inhibidores de canales ionicos de sodio y calcio dependientes de voltaje; composicion farmaceutica; y uso del compuesto en el tratamiento de dolor agudo, cronico, neu
GB0402578D0 (en) * 2004-02-05 2004-03-10 Cambridge Theranostics Ltd Methods of treatment of atherosclerosis
ATE459633T1 (de) * 2004-12-21 2010-03-15 Pfizer Prod Inc Makrolide

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR487411A (fr) * 1916-03-06 1918-07-03 Henri Dreyfus Procédé pour la fabrication de l'aldéhyde acétique en partant de l'acétylène
FR596802A (fr) * 1924-07-28 1925-11-02 Ste Chim Usines Rhone Procédé pour rendre la cellulose facilement éthérifiable
FR676409A (fr) * 1929-06-08 1930-02-22 Moule multiple
IL114589A (en) * 1990-11-21 1999-12-22 Roussel Uclaf Intermediates for the preparation of the history of erythromycin
FR2697524B1 (fr) * 1992-11-05 1994-12-23 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
US5527780A (en) * 1992-11-05 1996-06-18 Roussel Uclaf Erythromycin derivatives
FR2718450B1 (fr) * 1994-04-08 1997-01-10 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
FR2742757B1 (fr) * 1995-12-22 1998-01-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments

Also Published As

Publication number Publication date
EA002168B1 (ru) 2002-02-28
CA2261098C (fr) 2007-01-02
EA199900156A1 (ru) 1999-08-26
NO313332B1 (no) 2002-09-16
CN1178951C (zh) 2004-12-08
JP4267700B2 (ja) 2009-05-27
FR2751656A1 (fr) 1998-01-30
AP9901454A0 (en) 1999-03-31
PT931088E (pt) 2003-02-28
HUP9903424A3 (en) 2001-04-28
HUP9903424A1 (hu) 2000-03-28
BG103050A (en) 1999-10-29
NZ333559A (en) 1999-09-29
EP0931088A1 (fr) 1999-07-28
DE69716284D1 (de) 2002-11-14
CN1226252A (zh) 1999-08-18
BG62812B1 (bg) 2000-08-31
AP1078A (en) 2002-07-01
WO1998003530A1 (fr) 1998-01-29
AU710478B2 (en) 1999-09-23
YU3099A (sh) 2001-12-26
BR9710537B1 (pt) 2013-07-23
CZ292561B6 (cs) 2003-10-15
SK283713B6 (sk) 2003-12-02
UA48244C2 (uk) 2002-08-15
CA2261098A1 (fr) 1998-01-29
FR2751656B1 (fr) 1998-10-16
IL128182A0 (en) 1999-11-30
PL186297B1 (pl) 2003-12-31
DE69716284T2 (de) 2003-09-11
SK7299A3 (en) 1999-07-12
AU3853597A (en) 1998-02-10
ATE225798T1 (de) 2002-10-15
EP0931088B1 (fr) 2002-10-09
ES2181016T3 (es) 2003-02-16
IL128182A (en) 2006-12-31
DK0931088T3 (da) 2003-02-10
US6162793A (en) 2000-12-19
CZ20399A3 (cs) 1999-05-12
TR199900095T2 (xx) 1999-03-22
JP2000514817A (ja) 2000-11-07
NO990302D0 (no) 1999-01-22
BR9710537A (pt) 1999-08-17
PL331153A1 (en) 1999-06-21
NO990302L (no) 1999-03-23
KR20000068014A (ko) 2000-11-25
KR100458240B1 (ko) 2004-11-26

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Legal Events

Date Code Title Description
B25A Requested transfer of rights approved

Owner name: AVENTIS PHARMA S.A. (FR)

Free format text: TRANSFERIDO POR FUSAO DE: HOECHST MARION ROUSSEL INC.

B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE NAO ANUENCIA RELACIONADA COM O ART. 229 DA LPI

B07C Technical examination (opinion): republication [chapter 7.3 patent gazette]

Free format text: REPUBLICACAO QUANTO AO TEXTO DO DESPACHO 7.5 PUBLICADO NA RPI 2206 DE 16/04/2013. LEIA-SE O CORRETO: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI.

B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 23/07/2013, OBSERVADAS AS CONDICOES LEGAIS.

B16C Correction of notification of the grant [chapter 16.3 patent gazette]
B21F Lapse acc. art. 78, item iv - on non-payment of the annual fees in time

Free format text: REFERENTE A 22A ANUIDADE.

B24J Lapse because of non-payment of annual fees (definitively: art 78 iv lpi, resolution 113/2013 art. 12)

Free format text: EM VIRTUDE DA EXTINCAO PUBLICADA NA RPI 2524 DE 21-05-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDA A EXTINCAO DA PATENTE E SEUS CERTIFICADOS, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.