BR9714007A - Novos derivados da eritromicina seu processo de preparação e sua aplicação como medicamentos - Google Patents

Novos derivados da eritromicina seu processo de preparação e sua aplicação como medicamentos

Info

Publication number
BR9714007A
BR9714007A BR9714007-4A BR9714007A BR9714007A BR 9714007 A BR9714007 A BR 9714007A BR 9714007 A BR9714007 A BR 9714007A BR 9714007 A BR9714007 A BR 9714007A
Authority
BR
Brazil
Prior art keywords
drugs
application
preparation process
erythromycin
new derivatives
Prior art date
Application number
BR9714007-4A
Other languages
English (en)
Inventor
Jean Michel Auger
Constantin Agouridas
Jean Francois Chantot
Alexis Denis
Original Assignee
Hoechst Marion Roussel Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Marion Roussel Inc filed Critical Hoechst Marion Roussel Inc
Publication of BR9714007A publication Critical patent/BR9714007A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Patente de Invenção: <B>"NOVOS DERIVADOS DA ERITROMICINA, SEU PROCESSO DE PREPARAçãO E SUA APLICAçãO COMO MEDICAMENTOS"<D>. A invenção tem como objeto os compostos de fórmula (I) nos quais R representa um radical alquila eventualmente substituído ou (CH2)nAr, n representando um número inteiro que vai de 0 a 6 e Ar representando um radical arila ou heteroarila eventualmente substituído, e Z representa um átomo de hidrogênio ou o resto de um ácido carboxílico. Os compostos de fórmula (I) apresentam interessantes propriedades antibióticas.
BR9714007-4A 1996-12-12 1997-12-10 Novos derivados da eritromicina seu processo de preparação e sua aplicação como medicamentos BR9714007A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9615271A FR2757168B1 (fr) 1996-12-12 1996-12-12 Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
PCT/FR1997/002254 WO1998025942A1 (fr) 1996-12-12 1997-12-10 Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments

Publications (1)

Publication Number Publication Date
BR9714007A true BR9714007A (pt) 2000-05-09

Family

ID=9498593

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9714007-4A BR9714007A (pt) 1996-12-12 1997-12-10 Novos derivados da eritromicina seu processo de preparação e sua aplicação como medicamentos

Country Status (28)

Country Link
EP (1) EP0946579B1 (pt)
JP (1) JP4363666B2 (pt)
KR (1) KR100490074B1 (pt)
CN (2) CN1238364C (pt)
AP (1) AP997A (pt)
AT (1) ATE217008T1 (pt)
AU (1) AU721732B2 (pt)
BG (1) BG63124B1 (pt)
BR (1) BR9714007A (pt)
CA (1) CA2273985C (pt)
CZ (1) CZ292403B6 (pt)
DE (1) DE69712361T2 (pt)
DK (1) DK0946579T3 (pt)
EA (1) EA001733B1 (pt)
ES (1) ES2174323T3 (pt)
FR (1) FR2757168B1 (pt)
GE (1) GEP20012518B (pt)
HU (1) HUP0001180A3 (pt)
ID (1) ID21873A (pt)
IL (1) IL130420A (pt)
NO (1) NO314040B1 (pt)
NZ (1) NZ335325A (pt)
PT (1) PT946579E (pt)
SK (1) SK283715B6 (pt)
TR (1) TR199901301T2 (pt)
WO (1) WO1998025942A1 (pt)
YU (1) YU25699A (pt)
ZA (1) ZA9711101B (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2771008B1 (fr) * 1997-11-17 2000-04-28 Hoechst Marion Roussel Inc Utilisation des ketolides pour la preparation de compositions pharmaceutiques destinees a prevenir les complications thrombotiques arterielles liees a l'atherosclerose
EP1137654A1 (en) * 1998-12-10 2001-10-04 Pfizer Products Inc. Carbamate and carbazate ketolide antibiotics
DK1147121T3 (da) 1999-01-27 2004-04-13 Pfizer Prod Inc Ketolidantibiotika
WO2000063224A2 (en) * 1999-04-16 2000-10-26 Kosan Biosciences, Inc. Macrolide antiinfective agents
SK15162001A3 (sk) 1999-05-24 2003-02-04 Pfizer Products Inc. Deriváty 13-metylerytromycínu
US6472372B1 (en) * 2000-12-06 2002-10-29 Ortho-Mcneil Pharmaceuticals, Inc. 6-O-Carbamoyl ketolide antibacterials
DK200201957A (da) 2002-12-20 2003-01-20 Alpharma Aps 10-substituted erythromycin ketolides and methods of making

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4742049A (en) * 1986-06-04 1988-05-03 Abbott Laboratories Semisynthetic erythromycin antibiotics
IL99995A (en) * 1990-11-21 1997-11-20 Roussel Uclaf Erythromycin derivatives, their preparation and pharmaceutical compositions containing them
KR0166996B1 (ko) * 1992-04-22 1999-01-15 우에하라 아키라 5-o-데소사미닐에리쓰로노라이드a 유도체
US5527780A (en) * 1992-11-05 1996-06-18 Roussel Uclaf Erythromycin derivatives
JP3709997B2 (ja) * 1994-03-29 2005-10-26 日東電工株式会社 耐熱性ネガ型フォトレジスト組成物および感光性基材、ならびにネガ型パターン形成方法
FR2718450B1 (fr) * 1994-04-08 1997-01-10 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
FR2719587B1 (fr) * 1994-05-03 1996-07-12 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.

Also Published As

Publication number Publication date
JP2001506620A (ja) 2001-05-22
FR2757168B1 (fr) 1999-06-11
KR20000057517A (ko) 2000-09-15
CN100363375C (zh) 2008-01-23
AU5487798A (en) 1998-07-03
NO992859L (no) 1999-06-11
CA2273985A1 (fr) 1998-06-18
HUP0001180A2 (hu) 2000-09-28
NO992859D0 (no) 1999-06-11
CN1238364C (zh) 2006-01-25
NO314040B1 (no) 2003-01-20
EP0946579B1 (fr) 2002-05-02
YU25699A (sh) 2002-06-19
BG103398A (en) 2000-01-31
ATE217008T1 (de) 2002-05-15
HUP0001180A3 (en) 2003-05-28
AU721732B2 (en) 2000-07-13
WO1998025942A1 (fr) 1998-06-18
BG63124B1 (bg) 2001-04-30
CN1721427A (zh) 2006-01-18
DE69712361D1 (de) 2002-06-06
SK283715B6 (sk) 2003-12-02
PT946579E (pt) 2002-10-31
AP997A (en) 2001-08-09
DE69712361T2 (de) 2002-11-28
ES2174323T3 (es) 2002-11-01
CN1239966A (zh) 1999-12-29
ID21873A (id) 1999-08-05
FR2757168A1 (fr) 1998-06-19
IL130420A0 (en) 2000-06-01
GEP20012518B (en) 2001-08-27
ZA9711101B (en) 1998-12-10
KR100490074B1 (ko) 2005-05-17
AP9901513A0 (en) 1999-06-30
DK0946579T3 (da) 2002-08-12
CZ292403B6 (cs) 2003-09-17
CZ208299A3 (cs) 1999-09-15
NZ335325A (en) 2000-08-25
CA2273985C (fr) 2007-03-20
TR199901301T2 (xx) 1999-08-23
EA001733B1 (ru) 2001-08-27
EP0946579A1 (fr) 1999-10-06
IL130420A (en) 2003-01-12
SK75099A3 (en) 2000-01-18
JP4363666B2 (ja) 2009-11-11
EA199900528A1 (ru) 1999-12-29

Similar Documents

Publication Publication Date Title
ES2044836T3 (es) Derivado de la piperidina, su utilizacion y compuesto farmaceutico que lo contiene.
BR9913592A (pt) Compostos, processo de preparação dos compostos, e, composições farmacêuticas
MEP24608A (en) Azetidine derivatives, preparation thereof and pharmaceutical compositions containing same
ES2085130T3 (es) Nuevos derivados de la eritromicina, su procedimiento de preparacion, y su aplicacion como medicamentos.
CA2189271A1 (fr) Nouveaux derives de l&#39;erythromycine, leur procede de preparation et leur application comme medicaments
ATE260255T1 (de) 5-oxo-pyrrolidine-2-carbonsäure- hydroxamidderivate
NL194914B (nl) 4H-1-benzopyran-4-onderivaat of zout daarvan, en farmaceutisch preparaat dat dit als actieve stof bevat.
YU56995A (sh) Soli derivata indola
EA199900937A1 (ru) Фармацевтические композиции, содержащие вориконазол
FI921030A (fi) Cykliska ureaderivat, dessa foereningar innehaollande laekemedel och foerfarande foer deras framstaellning
YU13396A (sh) N-(3-benzofuranil) urea derivati, postupci za njihovo dobijanje, kompozicije koje ih sadrže i njihova upotreba u lekovima
DK77090D0 (da) Immunmodulerende azaspiraner
EA200200374A1 (ru) Производные хинолилпропилпиперидина, их получение и содержащие их композиции
BR9911771A (pt) Compostos cìclicos substituìdos, um processo para sua preparação e composições farmacêuticas que contêm os mesmos
BR0014939A (pt) Oligossacarìdeos, processo de preparação de oligossacarìdeos, composições farmacêuticas, e, utilização de oligossacarìdeos
DE3665711D1 (de) Novel guanidinomethylbenzoic acid derivatives
BR9714007A (pt) Novos derivados da eritromicina seu processo de preparação e sua aplicação como medicamentos
MD1560F2 (en) Cyclic compounds, pharmaceutical compositions on base thereof and methods of treatment of infections or diseases provoked by retroviruses.
FI955498A0 (fi) Nipekotiinihappojohdannaisia hyytymistä estävinä aineina
CA2107485A1 (fr) Nouveaux derives d&#39;ellipticine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
BRPI9710537B8 (pt) derivados da eritromicina, composições farmacêuticas, bem como processo para preparação dos mesmos.
HUP9601526A2 (hu) Véralvadásgátló hatású peptidil-arginin-aldehid-származékok és a vegyületeket tartalmazó gyógyszerkészítmények
EA200000389A3 (ru) Новые замещенные пиридины или пиперидины, способ их получения и содержащие их фармацевтические композиции
BR9801448A (pt) Compostos heterocìclicos, processo para sua preparação e composições farmacêuticas contendo os mesmos.
BRPI0012329B8 (pt) derivados de benzofurano, processo para sua preparação e uso dos mesmos.

Legal Events

Date Code Title Description
B25A Requested transfer of rights approved

Owner name: AVENTIS PHARMA S.A (FR)

Free format text: TRANSFERIDO DE: HOECHST MARION ROUSSEL

B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: DE ACORDO COM O ART. 37, INDEFIRO DO PRESENTE PEDIDO, UMA VEZ QUE: NAO ATENDE AO REQUISITO DE NOVIDADE ( ART. 8O COMBINADO COM O ART. 11 DA LPI 9279/96); NAO ATENDE AO REQUISITO DE ATIVIDADE INVENTIVA ( ART. 8O COMBINADO COM O ART. 13 DA LPI 9279/96).

B12B Appeal against refusal [chapter 12.2 patent gazette]
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B11D Dismissal acc. art. 38, par 2 of ipl - failure to pay fee after grant in time