YU25699A - Novi derivati eritromicina, postupak za njihovu izradu i njihova primena - Google Patents

Novi derivati eritromicina, postupak za njihovu izradu i njihova primena

Info

Publication number
YU25699A
YU25699A YU25699A YU25699A YU25699A YU 25699 A YU25699 A YU 25699A YU 25699 A YU25699 A YU 25699A YU 25699 A YU25699 A YU 25699A YU 25699 A YU25699 A YU 25699A
Authority
YU
Yugoslavia
Prior art keywords
preparing
erythromycin derivatives
novel erythromycin
representing
formula
Prior art date
Application number
YU25699A
Other languages
English (en)
Inventor
Jean-Michel Auger
Constantin Agouridas
Jean-Francois Chantot
Alexis Denis
Original Assignee
Hoechst Marion Roussel
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Marion Roussel filed Critical Hoechst Marion Roussel
Publication of YU25699A publication Critical patent/YU25699A/sh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Pronalazak se odnosi na jedinjenje formule (I) kod kojih R predstavlja jedan eventualno supstituisan alkil radikal ili (CH2)nAR, n predstavlja ceo broj izmedju 0 i 6, Ar predstavlja jedan arilni radikal ili heteroarilni radikal eventualno supstituisan, a Z predstavlja vodonikov atom ili radikal jedne karboksilne kiseline. Jedinjenja formule (I) imaju antibiotička svojstva.[The invention concerns compounds of formula (I) in which R represents an alkyl radical optionally substituted or (CH2)nAr, n representing a whole number ranging from 0 to 6 and Ar representing an aryl or heteroaryl radical optionally substituted, and Z represents a hydrogen atom or the radical of a carboxylic acid. The compounds of formula (I) have very interesting antibiotic properties.
YU25699A 1996-12-12 1997-12-10 Novi derivati eritromicina, postupak za njihovu izradu i njihova primena YU25699A (sh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9615271A FR2757168B1 (fr) 1996-12-12 1996-12-12 Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments

Publications (1)

Publication Number Publication Date
YU25699A true YU25699A (sh) 2002-06-19

Family

ID=9498593

Family Applications (1)

Application Number Title Priority Date Filing Date
YU25699A YU25699A (sh) 1996-12-12 1997-12-10 Novi derivati eritromicina, postupak za njihovu izradu i njihova primena

Country Status (28)

Country Link
EP (1) EP0946579B1 (sh)
JP (1) JP4363666B2 (sh)
KR (1) KR100490074B1 (sh)
CN (2) CN100363375C (sh)
AP (1) AP997A (sh)
AT (1) ATE217008T1 (sh)
AU (1) AU721732B2 (sh)
BG (1) BG63124B1 (sh)
BR (1) BR9714007A (sh)
CA (1) CA2273985C (sh)
CZ (1) CZ292403B6 (sh)
DE (1) DE69712361T2 (sh)
DK (1) DK0946579T3 (sh)
EA (1) EA001733B1 (sh)
ES (1) ES2174323T3 (sh)
FR (1) FR2757168B1 (sh)
GE (1) GEP20012518B (sh)
HU (1) HUP0001180A3 (sh)
ID (1) ID21873A (sh)
IL (1) IL130420A (sh)
NO (1) NO314040B1 (sh)
NZ (1) NZ335325A (sh)
PT (1) PT946579E (sh)
SK (1) SK283715B6 (sh)
TR (1) TR199901301T2 (sh)
WO (1) WO1998025942A1 (sh)
YU (1) YU25699A (sh)
ZA (1) ZA9711101B (sh)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2771008B1 (fr) * 1997-11-17 2000-04-28 Hoechst Marion Roussel Inc Utilisation des ketolides pour la preparation de compositions pharmaceutiques destinees a prevenir les complications thrombotiques arterielles liees a l'atherosclerose
TR200102129T2 (tr) * 1998-12-10 2002-01-21 Pfizer Products Inc. Karbamat ve karbazat ketolid antibiyotikleri.
HUP0105190A3 (en) 1999-01-27 2003-03-28 Pfizer Prod Inc Ketolide antibiotics, medicaments containing them and their use
KR100710605B1 (ko) * 1999-04-16 2007-04-24 코산 바이오사이언시즈, 인코포레이티드 매크롤라이드 항감염제
JP2003500414A (ja) 1999-05-24 2003-01-07 ファイザー・プロダクツ・インク １３−メチルエリスロマイシン誘導体
US6472372B1 (en) * 2000-12-06 2002-10-29 Ortho-Mcneil Pharmaceuticals, Inc. 6-O-Carbamoyl ketolide antibacterials
DK200201957A (da) 2002-12-20 2003-01-20 Alpharma Aps 10-substituted erythromycin ketolides and methods of making

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4742049A (en) * 1986-06-04 1988-05-03 Abbott Laboratories Semisynthetic erythromycin antibiotics
IL114589A (en) * 1990-11-21 1999-12-22 Roussel Uclaf Intermediates for the preparation of the history of erythromycin
US5591837A (en) * 1992-04-22 1997-01-07 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide a derivative
US5527780A (en) * 1992-11-05 1996-06-18 Roussel Uclaf Erythromycin derivatives
JP3709997B2 (ja) * 1994-03-29 2005-10-26 日東電工株式会社 耐熱性ネガ型フォトレジスト組成物および感光性基材、ならびにネガ型パターン形成方法
FR2718450B1 (fr) * 1994-04-08 1997-01-10 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
FR2719587B1 (fr) * 1994-05-03 1996-07-12 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.

Also Published As

Publication number Publication date
NZ335325A (en) 2000-08-25
CN1721427A (zh) 2006-01-18
EP0946579B1 (fr) 2002-05-02
FR2757168B1 (fr) 1999-06-11
ZA9711101B (en) 1998-12-10
GEP20012518B (en) 2001-08-27
SK75099A3 (en) 2000-01-18
AU5487798A (en) 1998-07-03
CN1239966A (zh) 1999-12-29
AU721732B2 (en) 2000-07-13
ID21873A (id) 1999-08-05
NO992859D0 (no) 1999-06-11
PT946579E (pt) 2002-10-31
IL130420A (en) 2003-01-12
HUP0001180A3 (en) 2003-05-28
SK283715B6 (sk) 2003-12-02
KR100490074B1 (ko) 2005-05-17
EA199900528A1 (ru) 1999-12-29
HUP0001180A2 (hu) 2000-09-28
DE69712361T2 (de) 2002-11-28
CN1238364C (zh) 2006-01-25
AP9901513A0 (en) 1999-06-30
BG63124B1 (bg) 2001-04-30
AP997A (en) 2001-08-09
NO314040B1 (no) 2003-01-20
ES2174323T3 (es) 2002-11-01
CZ208299A3 (cs) 1999-09-15
NO992859L (no) 1999-06-11
DE69712361D1 (de) 2002-06-06
EA001733B1 (ru) 2001-08-27
CZ292403B6 (cs) 2003-09-17
BG103398A (en) 2000-01-31
BR9714007A (pt) 2000-05-09
JP2001506620A (ja) 2001-05-22
EP0946579A1 (fr) 1999-10-06
IL130420A0 (en) 2000-06-01
CA2273985A1 (fr) 1998-06-18
JP4363666B2 (ja) 2009-11-11
TR199901301T2 (xx) 1999-08-23
CA2273985C (fr) 2007-03-20
FR2757168A1 (fr) 1998-06-19
CN100363375C (zh) 2008-01-23
KR20000057517A (ko) 2000-09-15
WO1998025942A1 (fr) 1998-06-18
DK0946579T3 (da) 2002-08-12
ATE217008T1 (de) 2002-05-15

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