AP9901566A0 - Novel erythromycin derivatives, method of preparation and application as medicines. - Google Patents
Novel erythromycin derivatives, method of preparation and application as medicines.Info
- Publication number
- AP9901566A0 AP9901566A0 APAP/P/1999/001566A AP9901566A AP9901566A0 AP 9901566 A0 AP9901566 A0 AP 9901566A0 AP 9901566 A AP9901566 A AP 9901566A AP 9901566 A0 AP9901566 A0 AP 9901566A0
- Authority
- AP
- ARIPO
- Prior art keywords
- medicines
- nar
- preparation
- application
- formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/04—Drugs for disorders of the respiratory system for throat disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A61P31/06—Antibacterial agents for tuberculosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pulmonology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Molecular Biology (AREA)
- Virology (AREA)
- Otolaryngology (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Tropical Medicine & Parasitology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Abstract
The invention concerns compounds of formula (i)in which x represents a ch2 or nh group, r represents a (ch2)nar,n-(ch2)nar or n=ch(ch2)nar radical, in which n represents a whole number ranging between 1 and 6 an ar represents an aryl or heteroaryl, optionally substituted, the dotted lines representing an optional double bond in 2(3), and y represents an hydrogen atom or an organic carboxylic acid radical containing up to 18 carbon atoms and their additive salts with acids. The compounds of formula (i)have antibiotic properties which enable their use as medicines.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9615830A FR2757518B1 (en) | 1996-12-23 | 1996-12-23 | NOVEL ERYTHROMYCIN DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICAMENTS |
| PCT/FR1997/002380 WO1998028316A1 (en) | 1996-12-23 | 1997-12-22 | Novel erythromycin derivatives, method of preparation and application as medicines |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AP9901566A0 true AP9901566A0 (en) | 1999-06-30 |
Family
ID=9498984
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| APAP/P/1999/001566A AP9901566A0 (en) | 1996-12-23 | 1997-12-22 | Novel erythromycin derivatives, method of preparation and application as medicines. |
Country Status (24)
| Country | Link |
|---|---|
| EP (1) | EP0946580B1 (en) |
| JP (2) | JP4522496B2 (en) |
| KR (1) | KR20000062286A (en) |
| CN (1) | CN1246123A (en) |
| AP (1) | AP9901566A0 (en) |
| AT (1) | ATE215553T1 (en) |
| AU (1) | AU726147B2 (en) |
| BR (1) | BR9713618A (en) |
| CA (1) | CA2275359A1 (en) |
| CZ (1) | CZ293732B6 (en) |
| DE (1) | DE69711689T2 (en) |
| DK (1) | DK0946580T3 (en) |
| EA (1) | EA199900589A1 (en) |
| ES (1) | ES2172827T3 (en) |
| FR (1) | FR2757518B1 (en) |
| HU (1) | HUP0001452A3 (en) |
| ID (1) | ID21883A (en) |
| IL (1) | IL130510A0 (en) |
| NO (1) | NO993124L (en) |
| PL (1) | PL334134A1 (en) |
| PT (1) | PT946580E (en) |
| SK (1) | SK83199A3 (en) |
| TR (1) | TR199901452T2 (en) |
| WO (1) | WO1998028316A1 (en) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2757518B1 (en) * | 1996-12-23 | 1999-06-11 | Hoechst Marion Roussel Inc | NOVEL ERYTHROMYCIN DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICAMENTS |
| YU44900A (en) | 1998-01-31 | 2003-01-31 | Glaxo Group Limited | 2-(purin-9-yl)-tetrahydrofuran-3,4-diol derivatives |
| US6720308B1 (en) * | 2002-11-07 | 2004-04-13 | Enanta Pharmaceuticals, Inc. | Anhydrolide derivatives having antibacterial activity |
| GB0514809D0 (en) | 2005-07-19 | 2005-08-24 | Glaxo Group Ltd | Compounds |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL99995A (en) * | 1990-11-21 | 1997-11-20 | Roussel Uclaf | Erythromycin derivatives, their preparation and pharmaceutical compositions containing them |
| JPH0853355A (en) * | 1994-08-12 | 1996-02-27 | Taisho Pharmaceut Co Ltd | Il-5 production-inhibiting agent |
| KR19990067333A (en) * | 1995-11-08 | 1999-08-16 | 스티븐 에프. 웨인스톡 | 3-deoxy-3-descladinose derivatives of erythromycins A and B |
| NZ332321A (en) * | 1996-05-07 | 2000-04-28 | Abbott Lab | 3-Descladinose-2,3-anhydroerythromycin derivatives and medicaments |
| FR2757518B1 (en) * | 1996-12-23 | 1999-06-11 | Hoechst Marion Roussel Inc | NOVEL ERYTHROMYCIN DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICAMENTS |
-
1996
- 1996-12-23 FR FR9615830A patent/FR2757518B1/en not_active Expired - Fee Related
-
1997
- 1997-12-22 HU HU0001452A patent/HUP0001452A3/en unknown
- 1997-12-22 IL IL13051097A patent/IL130510A0/en unknown
- 1997-12-22 DK DK97952973T patent/DK0946580T3/en active
- 1997-12-22 SK SK831-99A patent/SK83199A3/en unknown
- 1997-12-22 AP APAP/P/1999/001566A patent/AP9901566A0/en unknown
- 1997-12-22 EP EP97952973A patent/EP0946580B1/en not_active Expired - Lifetime
- 1997-12-22 ES ES97952973T patent/ES2172827T3/en not_active Expired - Lifetime
- 1997-12-22 AT AT97952973T patent/ATE215553T1/en not_active IP Right Cessation
- 1997-12-22 CZ CZ19992279A patent/CZ293732B6/en not_active IP Right Cessation
- 1997-12-22 AU AU56679/98A patent/AU726147B2/en not_active Ceased
- 1997-12-22 EA EA199900589A patent/EA199900589A1/en unknown
- 1997-12-22 DE DE69711689T patent/DE69711689T2/en not_active Expired - Lifetime
- 1997-12-22 WO PCT/FR1997/002380 patent/WO1998028316A1/en active IP Right Grant
- 1997-12-22 PL PL97334134A patent/PL334134A1/en unknown
- 1997-12-22 ID IDW990572A patent/ID21883A/en unknown
- 1997-12-22 BR BR9713618-2A patent/BR9713618A/en not_active Application Discontinuation
- 1997-12-22 CN CN97181784A patent/CN1246123A/en active Pending
- 1997-12-22 TR TR1999/01452T patent/TR199901452T2/en unknown
- 1997-12-22 KR KR1019997005682A patent/KR20000062286A/en not_active Application Discontinuation
- 1997-12-22 PT PT97952973T patent/PT946580E/en unknown
- 1997-12-22 CA CA002275359A patent/CA2275359A1/en not_active Abandoned
- 1997-12-22 JP JP52847498A patent/JP4522496B2/en not_active Expired - Lifetime
-
1999
- 1999-06-23 NO NO993124A patent/NO993124L/en not_active Application Discontinuation
-
2010
- 2010-02-01 JP JP2010020522A patent/JP5188520B2/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| ES2172827T3 (en) | 2002-10-01 |
| NO993124D0 (en) | 1999-06-23 |
| EP0946580A1 (en) | 1999-10-06 |
| JP5188520B2 (en) | 2013-04-24 |
| PT946580E (en) | 2002-09-30 |
| EP0946580B1 (en) | 2002-04-03 |
| WO1998028316A1 (en) | 1998-07-02 |
| AU726147B2 (en) | 2000-11-02 |
| CN1246123A (en) | 2000-03-01 |
| DE69711689T2 (en) | 2002-10-17 |
| IL130510A0 (en) | 2000-06-01 |
| CZ227999A3 (en) | 1999-10-13 |
| SK83199A3 (en) | 2000-05-16 |
| ID21883A (en) | 1999-08-05 |
| TR199901452T2 (en) | 1999-10-21 |
| AU5667998A (en) | 1998-07-17 |
| PL334134A1 (en) | 2000-02-14 |
| EA199900589A1 (en) | 2000-02-28 |
| CA2275359A1 (en) | 1998-07-02 |
| CZ293732B6 (en) | 2004-07-14 |
| HUP0001452A3 (en) | 2000-10-30 |
| DK0946580T3 (en) | 2002-07-22 |
| HU0001452B (en) | 2000-09-28 |
| NO993124L (en) | 1999-08-20 |
| KR20000062286A (en) | 2000-10-25 |
| JP2010132683A (en) | 2010-06-17 |
| FR2757518A1 (en) | 1998-06-26 |
| FR2757518B1 (en) | 1999-06-11 |
| BR9713618A (en) | 2000-04-11 |
| JP2001507011A (en) | 2001-05-29 |
| DE69711689D1 (en) | 2002-05-08 |
| ATE215553T1 (en) | 2002-04-15 |
| JP4522496B2 (en) | 2010-08-11 |
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