BG103398A - New derivatives of erythromicyn, method for their preparation and application as medicmentous forms - Google Patents

New derivatives of erythromicyn, method for their preparation and application as medicmentous forms

Info

Publication number
BG103398A
BG103398A BG103398A BG10339899A BG103398A BG 103398 A BG103398 A BG 103398A BG 103398 A BG103398 A BG 103398A BG 10339899 A BG10339899 A BG 10339899A BG 103398 A BG103398 A BG 103398A
Authority
BG
Bulgaria
Prior art keywords
medicmentous
erythromicyn
preparation
forms
application
Prior art date
Application number
BG103398A
Other languages
Bulgarian (bg)
Other versions
BG63124B1 (en
Inventor
Jean-Michel Auger
Constantin Agouridas
Jean-Francois Chantot
Alexis Denis
Original Assignee
Aventis Pharma S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma S.A. filed Critical Aventis Pharma S.A.
Publication of BG103398A publication Critical patent/BG103398A/en
Publication of BG63124B1 publication Critical patent/BG63124B1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

The compounds have the formula where R is alkyl radical, optionally substituted, or (CH2)nAr, n meaning an integer from 1 to 6 and Ar is aryl or heteroaryl radical, optionally substituted, and Z means hydrogen atom or radical of a carboxylic acid. 9 claims
BG103398A 1996-12-12 1999-05-12 New derivatives of erythromicyn, method for their preparation and application as medicmentous forms BG63124B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9615271A FR2757168B1 (en) 1996-12-12 1996-12-12 NOVEL ERYTHROMYCIN DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICAMENTS
PCT/FR1997/002254 WO1998025942A1 (en) 1996-12-12 1997-12-10 Novel erythromycin derivatives, method for preparing them and their use as medicine

Publications (2)

Publication Number Publication Date
BG103398A true BG103398A (en) 2000-01-31
BG63124B1 BG63124B1 (en) 2001-04-30

Family

ID=9498593

Family Applications (1)

Application Number Title Priority Date Filing Date
BG103398A BG63124B1 (en) 1996-12-12 1999-05-12 New derivatives of erythromicyn, method for their preparation and application as medicmentous forms

Country Status (28)

Country Link
EP (1) EP0946579B1 (en)
JP (1) JP4363666B2 (en)
KR (1) KR100490074B1 (en)
CN (2) CN100363375C (en)
AP (1) AP997A (en)
AT (1) ATE217008T1 (en)
AU (1) AU721732B2 (en)
BG (1) BG63124B1 (en)
BR (1) BR9714007A (en)
CA (1) CA2273985C (en)
CZ (1) CZ292403B6 (en)
DE (1) DE69712361T2 (en)
DK (1) DK0946579T3 (en)
EA (1) EA001733B1 (en)
ES (1) ES2174323T3 (en)
FR (1) FR2757168B1 (en)
GE (1) GEP20012518B (en)
HU (1) HUP0001180A3 (en)
ID (1) ID21873A (en)
IL (1) IL130420A (en)
NO (1) NO314040B1 (en)
NZ (1) NZ335325A (en)
PT (1) PT946579E (en)
SK (1) SK283715B6 (en)
TR (1) TR199901301T2 (en)
WO (1) WO1998025942A1 (en)
YU (1) YU25699A (en)
ZA (1) ZA9711101B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2771008B1 (en) * 1997-11-17 2000-04-28 Hoechst Marion Roussel Inc USE OF KETOLIDES FOR THE PREPARATION OF PHARMACEUTICAL COMPOSITIONS FOR PREVENTING ARTERIAL THROMBOTIC COMPLICATIONS LINKED TO ATHEROSCLEROSIS
ATE344269T1 (en) * 1998-12-10 2006-11-15 Pfizer Prod Inc CARBAMAT AND CARBAZATE KETOLIDE ANTIBIOTICS
BR9916969A (en) 1999-01-27 2001-11-06 Pfizer Prod Inc Ketolide antibiotics
ES2272273T3 (en) * 1999-04-16 2007-05-01 Kosan Biosciences, Inc. MACROLID ANTI-INFECTIVE AGENTS.
WO2000071557A1 (en) 1999-05-24 2000-11-30 Pfizer Products Inc. 13-methyl-erythromycin derivatives
US6472372B1 (en) * 2000-12-06 2002-10-29 Ortho-Mcneil Pharmaceuticals, Inc. 6-O-Carbamoyl ketolide antibacterials
DK200201957A (en) 2002-12-20 2003-01-20 Alpharma Aps 10-substituted erythromycin ketolides and methods of making

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4742049A (en) * 1986-06-04 1988-05-03 Abbott Laboratories Semisynthetic erythromycin antibiotics
IL99995A (en) * 1990-11-21 1997-11-20 Roussel Uclaf Erythromycin derivatives, their preparation and pharmaceutical compositions containing them
WO1993021199A1 (en) * 1992-04-22 1993-10-28 Taisho Pharmaceutical Co., Ltd. 5-o-desosaminylerythronolide a derivative
US5527780A (en) * 1992-11-05 1996-06-18 Roussel Uclaf Erythromycin derivatives
JP3709997B2 (en) * 1994-03-29 2005-10-26 日東電工株式会社 Heat resistant negative photoresist composition, photosensitive substrate, and negative pattern forming method
FR2718450B1 (en) * 1994-04-08 1997-01-10 Roussel Uclaf New erythromycin derivatives, their preparation process and their use as drugs.
FR2719587B1 (en) * 1994-05-03 1996-07-12 Roussel Uclaf New erythromycin derivatives, their preparation process and their use as drugs.

Also Published As

Publication number Publication date
CZ208299A3 (en) 1999-09-15
EP0946579B1 (en) 2002-05-02
AU721732B2 (en) 2000-07-13
ATE217008T1 (en) 2002-05-15
EP0946579A1 (en) 1999-10-06
KR20000057517A (en) 2000-09-15
CZ292403B6 (en) 2003-09-17
CA2273985C (en) 2007-03-20
CN1238364C (en) 2006-01-25
NO992859D0 (en) 1999-06-11
KR100490074B1 (en) 2005-05-17
WO1998025942A1 (en) 1998-06-18
ES2174323T3 (en) 2002-11-01
DE69712361T2 (en) 2002-11-28
EA199900528A1 (en) 1999-12-29
CA2273985A1 (en) 1998-06-18
AP9901513A0 (en) 1999-06-30
TR199901301T2 (en) 1999-08-23
YU25699A (en) 2002-06-19
GEP20012518B (en) 2001-08-27
BG63124B1 (en) 2001-04-30
HUP0001180A2 (en) 2000-09-28
EA001733B1 (en) 2001-08-27
ZA9711101B (en) 1998-12-10
ID21873A (en) 1999-08-05
CN1239966A (en) 1999-12-29
IL130420A0 (en) 2000-06-01
AU5487798A (en) 1998-07-03
NO992859L (en) 1999-06-11
NO314040B1 (en) 2003-01-20
CN1721427A (en) 2006-01-18
DK0946579T3 (en) 2002-08-12
AP997A (en) 2001-08-09
JP2001506620A (en) 2001-05-22
SK283715B6 (en) 2003-12-02
DE69712361D1 (en) 2002-06-06
HUP0001180A3 (en) 2003-05-28
FR2757168A1 (en) 1998-06-19
FR2757168B1 (en) 1999-06-11
SK75099A3 (en) 2000-01-18
IL130420A (en) 2003-01-12
PT946579E (en) 2002-10-31
CN100363375C (en) 2008-01-23
JP4363666B2 (en) 2009-11-11
NZ335325A (en) 2000-08-25
BR9714007A (en) 2000-05-09

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