BRPI0806689A2 - Compostos químicos 637 - Google Patents

Compostos químicos 637

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Publication number
BRPI0806689A2
BRPI0806689A2 BRPI0806689-2A BRPI0806689A BRPI0806689A2 BR PI0806689 A2 BRPI0806689 A2 BR PI0806689A2 BR PI0806689 A BRPI0806689 A BR PI0806689A BR PI0806689 A2 BRPI0806689 A2 BR PI0806689A2
Authority
BR
Brazil
Prior art keywords
chemical compounds
compounds
chemical
Prior art date
Application number
BRPI0806689-2A
Other languages
English (en)
Inventor
Roger Victor Bonnert
Frank Burkamp
Rhona Jane Cox
Simon De Sousa
Mark Dickinson
Simon Fraser Hunt
Premji Meghani
Austen Pimm
Hitesh Jayantilal Sanganee
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of BRPI0806689A2 publication Critical patent/BRPI0806689A2/pt

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08Bridged systems

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  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
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  • Physical Education & Sports Medicine (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Neurology (AREA)
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  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Rheumatology (AREA)
  • Virology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Molecular Biology (AREA)
  • Vascular Medicine (AREA)
BRPI0806689-2A 2007-01-11 2008-01-10 Compostos químicos 637 BRPI0806689A2 (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US88445407P 2007-01-11 2007-01-11
US94174907P 2007-06-04 2007-06-04
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US20090124596A1 (en) 2009-05-14
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UY30863A1 (es) 2008-09-02
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CA2674647A1 (en) 2008-07-17
CN101636388A (zh) 2010-01-27
US20120077801A1 (en) 2012-03-29
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AR064889A1 (es) 2009-05-06
JP2010515712A (ja) 2010-05-13
CO6210698A2 (es) 2010-10-20
MX2009007231A (es) 2009-07-14
PE20090049A1 (es) 2009-03-21
WO2008084223A2 (en) 2008-07-17
RU2009123930A (ru) 2011-02-20
TW200836745A (en) 2008-09-16
CL2008000089A1 (es) 2008-11-03
EP2106396A2 (en) 2009-10-07
AU2008204412B2 (en) 2012-03-01
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ECSP099480A (es) 2009-08-28
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