BRPI0806689A2 - Compostos químicos 637 - Google Patents
Compostos químicos 637Info
- Publication number
- BRPI0806689A2 BRPI0806689A2 BRPI0806689-2A BRPI0806689A BRPI0806689A2 BR PI0806689 A2 BRPI0806689 A2 BR PI0806689A2 BR PI0806689 A BRPI0806689 A BR PI0806689A BR PI0806689 A2 BRPI0806689 A2 BR PI0806689A2
- Authority
- BR
- Brazil
- Prior art keywords
- chemical compounds
- compounds
- chemical
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
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- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
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- Rheumatology (AREA)
- Virology (AREA)
- Neurosurgery (AREA)
- Diabetes (AREA)
- Orthopedic Medicine & Surgery (AREA)
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- Endocrinology (AREA)
- Pain & Pain Management (AREA)
- Urology & Nephrology (AREA)
- Hematology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Dermatology (AREA)
- Gynecology & Obstetrics (AREA)
- Psychiatry (AREA)
- Ophthalmology & Optometry (AREA)
- Molecular Biology (AREA)
- Vascular Medicine (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US88445407P | 2007-01-11 | 2007-01-11 | |
US94174907P | 2007-06-04 | 2007-06-04 | |
US95204707P | 2007-07-26 | 2007-07-26 | |
PCT/GB2008/000061 WO2008084223A2 (en) | 2007-01-11 | 2008-01-10 | Chemical compounds 637: pyridopyrimidinediones as pde4 inhibitors |
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US (3) | US20090124596A1 (pt) |
EP (1) | EP2106396B1 (pt) |
JP (1) | JP5369302B2 (pt) |
KR (1) | KR20090101303A (pt) |
CN (3) | CN102532135A (pt) |
AR (1) | AR064889A1 (pt) |
AU (1) | AU2008204412B2 (pt) |
BR (1) | BRPI0806689A2 (pt) |
CA (1) | CA2674647A1 (pt) |
CL (1) | CL2008000089A1 (pt) |
CO (1) | CO6210698A2 (pt) |
EC (1) | ECSP099480A (pt) |
MX (1) | MX2009007231A (pt) |
MY (1) | MY162022A (pt) |
PE (2) | PE20090049A1 (pt) |
RU (1) | RU2479584C2 (pt) |
SA (1) | SA08280783B1 (pt) |
TW (1) | TW200836745A (pt) |
UY (1) | UY30863A1 (pt) |
WO (1) | WO2008084223A2 (pt) |
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SA08280783B1 (ar) * | 2007-01-11 | 2011-04-24 | استرازينيكا ايه بي | مشتقات بيريدوبيريميدين كمثبطات pde4 |
WO2010004319A1 (en) * | 2008-07-07 | 2010-01-14 | Astrazeneca Ab | Combination comprising 6-flu0r0-n- ((1s, 4s) - 4- (6-fluoro-2, 4-di0x0-1- (4'- (piperazin-1- ylmethyl) biphenyl- 3-yl) -1, 2-dihydropyrido [2, 3-d] pyrimidin-3 (4h) - yl) cyclohexyl) imidazo [1,2-a] pyridine -2- carboxamide or a salt |
TW201036957A (en) | 2009-02-20 | 2010-10-16 | Astrazeneca Ab | Novel salt 628 |
JP5558875B2 (ja) * | 2009-03-19 | 2014-07-23 | 日本曹達株式会社 | 新規包接錯体、エポキシ樹脂組成物及び半導体封止用エポキシ樹脂組成物 |
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GB201016912D0 (en) | 2010-10-07 | 2010-11-24 | Astrazeneca Ab | Novel combination |
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GB201021979D0 (en) | 2010-12-23 | 2011-02-02 | Astrazeneca Ab | New compound |
JP6039587B2 (ja) * | 2011-03-18 | 2016-12-07 | コーセプト セラピューティクス, インコーポレイテッド | ピリミジンシクロヘキシルグルココルチコイドレセプター調節因子 |
EP2915804B1 (en) | 2012-10-31 | 2019-03-27 | FUJIFILM Toyama Chemical Co., Ltd. | Novel amine derivative or salt thereof as tnf alpha inhibitors |
WO2014151761A1 (en) * | 2013-03-15 | 2014-09-25 | Ariad Pharmaceuticals, Inc. | Novel choline kinase inhibitors |
WO2016029216A2 (en) * | 2014-08-22 | 2016-02-25 | Biocryst Pharmaceuticals, Inc. | Method for producing amidine derivatives |
KR101671404B1 (ko) * | 2014-09-02 | 2016-11-02 | 한국원자력의학원 | 항암 효과, 방사선 병용치료 효과 및 당뇨병 치료 효과를 갖는 피리미딘 유도체 및 이의 의학적 용도 |
KR20180011843A (ko) | 2015-06-11 | 2018-02-02 | 바실리어 파마슈티카 인터내셔널 리미티드 | 유출-펌프 억제제 및 이의 치료적 용도 |
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2008
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- 2008-01-10 WO PCT/GB2008/000061 patent/WO2008084223A2/en active Application Filing
- 2008-01-10 CN CN2011104106459A patent/CN102532135A/zh active Pending
- 2008-01-10 EP EP08700158.2A patent/EP2106396B1/en active Active
- 2008-01-10 CA CA002674647A patent/CA2674647A1/en not_active Abandoned
- 2008-01-10 US US11/972,182 patent/US20090124596A1/en not_active Abandoned
- 2008-01-10 UY UY30863A patent/UY30863A1/es not_active Application Discontinuation
- 2008-01-10 BR BRPI0806689-2A patent/BRPI0806689A2/pt not_active IP Right Cessation
- 2008-01-10 US US12/522,782 patent/US20100204203A1/en not_active Abandoned
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- 2008-01-10 JP JP2009545224A patent/JP5369302B2/ja not_active Expired - Fee Related
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- 2008-01-10 AU AU2008204412A patent/AU2008204412B2/en not_active Ceased
- 2008-01-10 KR KR1020097016638A patent/KR20090101303A/ko not_active Application Discontinuation
- 2008-01-10 CN CN201410326870.8A patent/CN104147011A/zh active Pending
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- 2008-01-11 PE PE2008000127A patent/PE20090049A1/es not_active Application Discontinuation
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- 2008-01-11 AR ARP080100155A patent/AR064889A1/es unknown
- 2008-01-11 TW TW097101165A patent/TW200836745A/zh unknown
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Also Published As
Publication number | Publication date |
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KR20090101303A (ko) | 2009-09-24 |
SA08280783B1 (ar) | 2011-04-24 |
PE20121529A1 (es) | 2012-12-16 |
US20100204203A1 (en) | 2010-08-12 |
MY162022A (en) | 2017-05-31 |
WO2008084223A3 (en) | 2008-10-02 |
JP5369302B2 (ja) | 2013-12-18 |
US20090124596A1 (en) | 2009-05-14 |
EP2106396B1 (en) | 2014-09-24 |
UY30863A1 (es) | 2008-09-02 |
CN104147011A (zh) | 2014-11-19 |
CN102532135A (zh) | 2012-07-04 |
CA2674647A1 (en) | 2008-07-17 |
CN101636388A (zh) | 2010-01-27 |
US20120077801A1 (en) | 2012-03-29 |
CN101636388B (zh) | 2013-09-18 |
AR064889A1 (es) | 2009-05-06 |
JP2010515712A (ja) | 2010-05-13 |
CO6210698A2 (es) | 2010-10-20 |
MX2009007231A (es) | 2009-07-14 |
PE20090049A1 (es) | 2009-03-21 |
WO2008084223A2 (en) | 2008-07-17 |
RU2009123930A (ru) | 2011-02-20 |
TW200836745A (en) | 2008-09-16 |
CL2008000089A1 (es) | 2008-11-03 |
EP2106396A2 (en) | 2009-10-07 |
AU2008204412B2 (en) | 2012-03-01 |
RU2479584C2 (ru) | 2013-04-20 |
ECSP099480A (es) | 2009-08-28 |
AU2008204412A1 (en) | 2008-07-17 |
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