BRPI0507670A - moduladores do receptor de androgênio - Google Patents

moduladores do receptor de androgênio

Info

Publication number
BRPI0507670A
BRPI0507670A BRPI0507670-6A BRPI0507670A BRPI0507670A BR PI0507670 A BRPI0507670 A BR PI0507670A BR PI0507670 A BRPI0507670 A BR PI0507670A BR PI0507670 A BRPI0507670 A BR PI0507670A
Authority
BR
Brazil
Prior art keywords
androgen receptor
receptor modulators
modulators
androgen
oxobenzonitriles
Prior art date
Application number
BRPI0507670-6A
Other languages
English (en)
Portuguese (pt)
Inventor
Lain-Yen Hu
Huangshu Lei
Daniel Yunlong Du
Bruce Allen Lefker
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of BRPI0507670A publication Critical patent/BRPI0507670A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • C07C255/49Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C255/54Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and etherified hydroxy groups bound to the carbon skeleton
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • A61K31/277Nitriles; Isonitriles having a ring, e.g. verapamil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/08Antiseborrheics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/10Anti-acne agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/14Drugs for dermatological disorders for baldness or alopecia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/28Antiandrogens
BRPI0507670-6A 2004-02-13 2005-01-31 moduladores do receptor de androgênio BRPI0507670A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US54473804P 2004-02-13 2004-02-13
US60564704P 2004-08-30 2004-08-30
PCT/IB2005/000229 WO2005080320A1 (en) 2004-02-13 2005-01-31 Androgen receptor modulators

Publications (1)

Publication Number Publication Date
BRPI0507670A true BRPI0507670A (pt) 2007-07-17

Family

ID=34890476

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0507670-6A BRPI0507670A (pt) 2004-02-13 2005-01-31 moduladores do receptor de androgênio

Country Status (20)

Country Link
US (1) US7576128B2 (US07576128-20090818-C00068.png)
EP (1) EP1716110A1 (US07576128-20090818-C00068.png)
JP (1) JP3997255B2 (US07576128-20090818-C00068.png)
KR (1) KR100783255B1 (US07576128-20090818-C00068.png)
AP (1) AP2006003700A0 (US07576128-20090818-C00068.png)
AR (1) AR047606A1 (US07576128-20090818-C00068.png)
AU (1) AU2005214167B2 (US07576128-20090818-C00068.png)
BR (1) BRPI0507670A (US07576128-20090818-C00068.png)
CA (1) CA2554696C (US07576128-20090818-C00068.png)
CR (1) CR8555A (US07576128-20090818-C00068.png)
EA (1) EA009902B1 (US07576128-20090818-C00068.png)
EC (1) ECSP066761A (US07576128-20090818-C00068.png)
IL (1) IL176935A0 (US07576128-20090818-C00068.png)
MA (1) MA28361A1 (US07576128-20090818-C00068.png)
NO (1) NO20064053L (US07576128-20090818-C00068.png)
PA (1) PA8623501A1 (US07576128-20090818-C00068.png)
PE (1) PE20051168A1 (US07576128-20090818-C00068.png)
TW (1) TW200534842A (US07576128-20090818-C00068.png)
UY (1) UY28746A1 (US07576128-20090818-C00068.png)
WO (1) WO2005080320A1 (US07576128-20090818-C00068.png)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005100305A1 (en) 2004-04-13 2005-10-27 Warner-Lambert Company Llc Androgen modulators
EP1740533A1 (en) 2004-04-22 2007-01-10 Warner-Lambert Company LLC Androgen modulators
MXPA06015169A (es) * 2004-07-08 2007-08-21 Warner Lambert Co Moduladores de androgenos.
BRPI0514469A (pt) * 2004-08-18 2008-06-10 Warner Lambert Co moduladores de androgênio
CN101044131A (zh) * 2004-08-31 2007-09-26 沃尼尔·朗伯有限责任公司 雄激素调节剂
TW200724139A (en) 2005-05-05 2007-07-01 Warner Lambert Co Androgen modulators
TW200708499A (en) * 2005-06-22 2007-03-01 Warner Lambert Co Process for producing ethers
WO2007007149A1 (en) * 2005-07-12 2007-01-18 Warner-Lambert Company Llc Androgen modulators
US20090170886A1 (en) * 2005-08-08 2009-07-02 Pfizer Inc Androgen modulators
EP3108879A1 (en) * 2015-06-25 2016-12-28 Cassiopea S.p.A. High concentration formulation
US20210292335A1 (en) * 2018-08-07 2021-09-23 Emory University Heterocyclic Flavone Derivatives, Compositions, and Methods Related Thereto

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Also Published As

Publication number Publication date
NO20064053L (no) 2006-11-08
PE20051168A1 (es) 2006-02-18
WO2005080320A1 (en) 2005-09-01
AU2005214167A1 (en) 2005-09-01
EA200601267A1 (ru) 2006-12-29
KR100783255B1 (ko) 2007-12-06
US20050182132A1 (en) 2005-08-18
JP2007522199A (ja) 2007-08-09
UY28746A1 (es) 2005-09-30
AR047606A1 (es) 2006-01-25
PA8623501A1 (es) 2005-08-30
AP2006003700A0 (en) 2006-08-31
AU2005214167B2 (en) 2008-08-07
KR20060116223A (ko) 2006-11-14
CA2554696A1 (en) 2005-09-01
JP3997255B2 (ja) 2007-10-24
CA2554696C (en) 2009-06-30
EA009902B1 (ru) 2008-04-28
US7576128B2 (en) 2009-08-18
TW200534842A (en) 2005-11-01
ECSP066761A (es) 2006-11-16
CR8555A (es) 2006-10-17
IL176935A0 (en) 2006-12-10
MA28361A1 (fr) 2006-12-01
EP1716110A1 (en) 2006-11-02

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