BR9815140A - "derivados de 2-aril-8-oxodidropurina, processo para a sua produção, composições medicinais contendo os mesmos, e seus intermediários" - Google Patents

"derivados de 2-aril-8-oxodidropurina, processo para a sua produção, composições medicinais contendo os mesmos, e seus intermediários"

Info

Publication number
BR9815140A
BR9815140A BR9815140-1A BR9815140A BR9815140A BR 9815140 A BR9815140 A BR 9815140A BR 9815140 A BR9815140 A BR 9815140A BR 9815140 A BR9815140 A BR 9815140A
Authority
BR
Brazil
Prior art keywords
aryl
derivatives
production
compositions containing
medicinal compositions
Prior art date
Application number
BR9815140-1A
Other languages
English (en)
Inventor
Teruya Murata
Kaoru Masumoto
Katsunori Kondo
Kiyoshi Furukawa
Makoto Oka
Original Assignee
Dainippon Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dainippon Pharmaceutical Co filed Critical Dainippon Pharmaceutical Co
Publication of BR9815140A publication Critical patent/BR9815140A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

"DERIVADOS DE 2-ARIL-8-OXODIIDROPURINA, PROCESSO PARA A SUA PRODUçãO, COMPOSIçõES MEDICINAIS CONTENDO OS MESMOS, E SEUS INTERMEDIáRIOS" Derivados de 2-aril-8-oxodiidro purina representados pela fórmula geral (I) os seus sais por adição de ácido farmaceuticamente aceitáveis. Estes compostos são úteis como remédios e preventivos para doenças associadas com ansiedade (neurose, distúrbio psicofisiológico, distúrbio de ansiedade etc), doenças do sistema nervoso central tais como depressão e epilepsia e doenças circulatórias tais como angina pectoris e hipertensão. Na citada fórmula, A representa fenila opcionalmente substituído ou heteroarila opcionalmente substituído; e ou X ou Y representa [Q] : -CH (R³) CON (R¹) (R²).
BR9815140-1A 1997-12-03 1998-11-26 "derivados de 2-aril-8-oxodidropurina, processo para a sua produção, composições medicinais contendo os mesmos, e seus intermediários" BR9815140A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP35000097 1997-12-03
PCT/JP1998/005320 WO1999028320A1 (fr) 1997-12-03 1998-11-26 Derives de 2-aryl-8-oxodihydropurine, procede de production de ces derives, compositions medicales contenant ces derives, et intermediaires de ces derives

Publications (1)

Publication Number Publication Date
BR9815140A true BR9815140A (pt) 2000-10-10

Family

ID=18407561

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9815140-1A BR9815140A (pt) 1997-12-03 1998-11-26 "derivados de 2-aril-8-oxodidropurina, processo para a sua produção, composições medicinais contendo os mesmos, e seus intermediários"

Country Status (27)

Country Link
US (1) US6372740B1 (pt)
EP (1) EP1036794B1 (pt)
JP (1) JP3815966B2 (pt)
KR (1) KR100494347B1 (pt)
CN (1) CN1146566C (pt)
AR (1) AR017796A1 (pt)
AT (1) ATE248169T1 (pt)
AU (1) AU744014B2 (pt)
BR (1) BR9815140A (pt)
CA (1) CA2312885C (pt)
DE (1) DE69817611T2 (pt)
DK (1) DK1036794T3 (pt)
ES (1) ES2205574T3 (pt)
HK (1) HK1028769A1 (pt)
HU (1) HUP0004422A3 (pt)
ID (1) ID24929A (pt)
IL (1) IL135920A0 (pt)
NO (1) NO20002835L (pt)
NZ (1) NZ504457A (pt)
PL (1) PL191489B1 (pt)
PT (1) PT1036794E (pt)
RU (1) RU2223272C2 (pt)
SK (1) SK285703B6 (pt)
TR (1) TR200001600T2 (pt)
TW (1) TW502034B (pt)
WO (1) WO1999028320A1 (pt)
ZA (1) ZA9810490B (pt)

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Also Published As

Publication number Publication date
DK1036794T3 (da) 2003-12-22
CA2312885C (en) 2008-01-29
NO20002835D0 (no) 2000-06-02
CN1146566C (zh) 2004-04-21
RU2223272C2 (ru) 2004-02-10
HUP0004422A2 (hu) 2001-04-28
HK1028769A1 (en) 2001-03-02
AU744014B2 (en) 2002-02-14
TW502034B (en) 2002-09-11
IL135920A0 (en) 2001-05-20
PT1036794E (pt) 2003-11-28
NO20002835L (no) 2000-07-24
EP1036794A4 (en) 2001-12-12
TR200001600T2 (tr) 2000-11-21
ZA9810490B (en) 1999-05-20
JP3815966B2 (ja) 2006-08-30
US6372740B1 (en) 2002-04-16
DE69817611T2 (de) 2004-02-26
NZ504457A (en) 2001-12-21
HUP0004422A3 (en) 2001-10-29
PL191489B1 (pl) 2006-05-31
EP1036794A1 (en) 2000-09-20
ID24929A (id) 2000-08-31
EP1036794B1 (en) 2003-08-27
AR017796A1 (es) 2001-10-24
SK7972000A3 (en) 2001-03-12
ATE248169T1 (de) 2003-09-15
CA2312885A1 (en) 1999-06-10
PL340925A1 (en) 2001-03-12
DE69817611D1 (de) 2003-10-02
KR100494347B1 (ko) 2005-06-13
SK285703B6 (sk) 2007-06-07
AU1260499A (en) 1999-06-16
ES2205574T3 (es) 2004-05-01
CN1284076A (zh) 2001-02-14
WO1999028320A1 (fr) 1999-06-10
KR20010032686A (ko) 2001-04-25

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