PT1036794E - Derivados de 2-aril-8-oxodi-hidropurina processo para a sua producao composicoes medicinais que os contem e seus intermediarios - Google Patents

Derivados de 2-aril-8-oxodi-hidropurina processo para a sua producao composicoes medicinais que os contem e seus intermediarios

Info

Publication number
PT1036794E
PT1036794E PT98955937T PT98955937T PT1036794E PT 1036794 E PT1036794 E PT 1036794E PT 98955937 T PT98955937 T PT 98955937T PT 98955937 T PT98955937 T PT 98955937T PT 1036794 E PT1036794 E PT 1036794E
Authority
PT
Portugal
Prior art keywords
hydropurin
oxodi
intermediaries
aryl
contain
Prior art date
Application number
PT98955937T
Other languages
English (en)
Inventor
Teruya Murata
Kiyoshi Furukawa
Makoto Oka
Kaoru Masumoto
Katsunori Kondo
Original Assignee
Dainippon Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dainippon Pharmaceutical Co filed Critical Dainippon Pharmaceutical Co
Publication of PT1036794E publication Critical patent/PT1036794E/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PT98955937T 1997-12-03 1998-11-26 Derivados de 2-aril-8-oxodi-hidropurina processo para a sua producao composicoes medicinais que os contem e seus intermediarios PT1036794E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP35000097 1997-12-03

Publications (1)

Publication Number Publication Date
PT1036794E true PT1036794E (pt) 2003-11-28

Family

ID=18407561

Family Applications (1)

Application Number Title Priority Date Filing Date
PT98955937T PT1036794E (pt) 1997-12-03 1998-11-26 Derivados de 2-aril-8-oxodi-hidropurina processo para a sua producao composicoes medicinais que os contem e seus intermediarios

Country Status (27)

Country Link
US (1) US6372740B1 (pt)
EP (1) EP1036794B1 (pt)
JP (1) JP3815966B2 (pt)
KR (1) KR100494347B1 (pt)
CN (1) CN1146566C (pt)
AR (1) AR017796A1 (pt)
AT (1) ATE248169T1 (pt)
AU (1) AU744014B2 (pt)
BR (1) BR9815140A (pt)
CA (1) CA2312885C (pt)
DE (1) DE69817611T2 (pt)
DK (1) DK1036794T3 (pt)
ES (1) ES2205574T3 (pt)
HK (1) HK1028769A1 (pt)
HU (1) HUP0004422A3 (pt)
ID (1) ID24929A (pt)
IL (1) IL135920A0 (pt)
NO (1) NO20002835L (pt)
NZ (1) NZ504457A (pt)
PL (1) PL191489B1 (pt)
PT (1) PT1036794E (pt)
RU (1) RU2223272C2 (pt)
SK (1) SK285703B6 (pt)
TR (1) TR200001600T2 (pt)
TW (1) TW502034B (pt)
WO (1) WO1999028320A1 (pt)
ZA (1) ZA9810490B (pt)

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US20090281075A1 (en) * 2006-02-17 2009-11-12 Pharmacopeia, Inc. Isomeric purinones and 1h-imidazopyridinones as pkc-theta inhibitors
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ZA200807715B (en) * 2006-03-09 2009-11-25 Pharmacopeia Inc 9-Heteroarylpurine MNK2 inhibitors for treating metabolic disorders
US7902187B2 (en) * 2006-10-04 2011-03-08 Wyeth Llc 6-substituted 2-(benzimidazolyl)purine and purinone derivatives for immunosuppression
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EP3091021B1 (en) 2009-10-26 2019-08-28 Signal Pharmaceuticals, LLC Methods of synthesis and purification of heteroaryl compounds
JP2014076947A (ja) * 2011-02-03 2014-05-01 Dainippon Sumitomo Pharma Co Ltd ２−オキシ置換８−オキソジヒドロプリン誘導体
EP2718464A1 (en) 2011-06-06 2014-04-16 Imperial Innovations Limited Methods to predict binding affinity of tspo imaging agents to tspo
TWI629983B (zh) 2011-10-19 2018-07-21 標誌製藥公司 以ｔｏｒ激酶抑制劑治療癌症
PE20141696A1 (es) 2011-12-02 2014-11-08 Signal Pharm Llc Composiciones farmaceuticas de 7-(6-(2-hidroxipropan-2-il) piridin-3-il)-1-((trans)-4-metoxiciclohexil)-3,4-dihidropirazino[2,3-b] pirazin-2(1h)-ona, una forma solida del mismo y metodos de su uso
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KR102221005B1 (ko) 2013-04-17 2021-02-26 시그날 파마소티칼 엘엘씨 전립선암 치료를 위한 디하이드로피라지노-피라진 화합물 및 안드로겐 수용체 길항제를 포함하는 조합 요법
KR102271344B1 (ko) 2013-04-17 2021-07-01 시그날 파마소티칼 엘엘씨 디하이드로피라지노-피라진을 사용한 암의 치료
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Also Published As

Publication number Publication date
WO1999028320A1 (fr) 1999-06-10
EP1036794A1 (en) 2000-09-20
BR9815140A (pt) 2000-10-10
NZ504457A (en) 2001-12-21
PL340925A1 (en) 2001-03-12
DE69817611D1 (de) 2003-10-02
CA2312885C (en) 2008-01-29
KR100494347B1 (ko) 2005-06-13
CA2312885A1 (en) 1999-06-10
DE69817611T2 (de) 2004-02-26
CN1284076A (zh) 2001-02-14
ZA9810490B (en) 1999-05-20
ID24929A (id) 2000-08-31
JP3815966B2 (ja) 2006-08-30
RU2223272C2 (ru) 2004-02-10
EP1036794A4 (en) 2001-12-12
SK7972000A3 (en) 2001-03-12
DK1036794T3 (da) 2003-12-22
SK285703B6 (sk) 2007-06-07
KR20010032686A (ko) 2001-04-25
HUP0004422A2 (hu) 2001-04-28
CN1146566C (zh) 2004-04-21
US6372740B1 (en) 2002-04-16
TR200001600T2 (tr) 2000-11-21
HUP0004422A3 (en) 2001-10-29
HK1028769A1 (en) 2001-03-02
ES2205574T3 (es) 2004-05-01
AR017796A1 (es) 2001-10-24
AU744014B2 (en) 2002-02-14
TW502034B (en) 2002-09-11
EP1036794B1 (en) 2003-08-27
NO20002835D0 (no) 2000-06-02
AU1260499A (en) 1999-06-16
IL135920A0 (en) 2001-05-20
ATE248169T1 (de) 2003-09-15
PL191489B1 (pl) 2006-05-31
NO20002835L (no) 2000-07-24

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