BR112023021107A2 - Compostos de tienopirrol - Google Patents
Compostos de tienopirrolInfo
- Publication number
- BR112023021107A2 BR112023021107A2 BR112023021107A BR112023021107A BR112023021107A2 BR 112023021107 A2 BR112023021107 A2 BR 112023021107A2 BR 112023021107 A BR112023021107 A BR 112023021107A BR 112023021107 A BR112023021107 A BR 112023021107A BR 112023021107 A2 BR112023021107 A2 BR 112023021107A2
- Authority
- BR
- Brazil
- Prior art keywords
- compounds
- thienopirrol
- lupus erythematosus
- pharmaceutical compositions
- treating
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 6
- 239000008194 pharmaceutical composition Substances 0.000 abstract 2
- 208000023275 Autoimmune disease Diseases 0.000 abstract 1
- 208000004921 cutaneous lupus erythematosus Diseases 0.000 abstract 1
- 230000004968 inflammatory condition Effects 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 201000000596 systemic lupus erythematosus Diseases 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4706—4-Aminoquinolines; 8-Aminoquinolines, e.g. chloroquine, primaquine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Abstract
compostos de tienopirrol. a presente invenção refere-se, de modo geral, a certos compostos, composições farmacêuticas compreendendo os ditos compostos e métodos de preparo e uso dos ditos compostos e composições farmacêuticas. os compostos e as composições aqui fornecidos podem ser utilizados para tratamento ou prevenção de uma doença autoimune e/ou condição inflamatória, incluindo lúpus eritematoso sistêmico e lúpus eritematoso cutâneo.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US202163176109P | 2021-04-16 | 2021-04-16 | |
US202163216418P | 2021-06-29 | 2021-06-29 | |
US202263305610P | 2022-02-01 | 2022-02-01 | |
PCT/US2022/024984 WO2022221642A1 (en) | 2021-04-16 | 2022-04-15 | Thienopyrrole compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112023021107A2 true BR112023021107A2 (pt) | 2023-12-12 |
Family
ID=81580723
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112023021107A BR112023021107A2 (pt) | 2021-04-16 | 2022-04-15 | Compostos de tienopirrol |
Country Status (13)
Country | Link |
---|---|
US (2) | US11661431B2 (pt) |
EP (1) | EP4323369A1 (pt) |
JP (1) | JP2024513945A (pt) |
KR (1) | KR20230171469A (pt) |
AU (1) | AU2022257039A1 (pt) |
BR (1) | BR112023021107A2 (pt) |
CA (1) | CA3214808A1 (pt) |
CO (1) | CO2023013397A2 (pt) |
CR (1) | CR20230478A (pt) |
DO (1) | DOP2023000219A (pt) |
IL (1) | IL307203A (pt) |
TW (1) | TW202302598A (pt) |
WO (1) | WO2022221642A1 (pt) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20230270734A1 (en) * | 2021-09-10 | 2023-08-31 | Gilead Sciences, Inc. | Thienopyrrole compounds |
WO2023247670A1 (en) * | 2022-06-24 | 2023-12-28 | F. Hoffmann-La Roche Ag | New heterocyclic-carbonyl-cyclic compounds as magl inhibitors |
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-
2022
- 2022-04-15 CA CA3214808A patent/CA3214808A1/en active Pending
- 2022-04-15 CR CR20230478A patent/CR20230478A/es unknown
- 2022-04-15 JP JP2023562311A patent/JP2024513945A/ja active Pending
- 2022-04-15 TW TW111114449A patent/TW202302598A/zh unknown
- 2022-04-15 US US17/721,636 patent/US11661431B2/en active Active
- 2022-04-15 AU AU2022257039A patent/AU2022257039A1/en active Pending
- 2022-04-15 WO PCT/US2022/024984 patent/WO2022221642A1/en active Application Filing
- 2022-04-15 KR KR1020237039381A patent/KR20230171469A/ko unknown
- 2022-04-15 EP EP22721581.1A patent/EP4323369A1/en active Pending
- 2022-04-15 IL IL307203A patent/IL307203A/en unknown
- 2022-04-15 BR BR112023021107A patent/BR112023021107A2/pt unknown
-
2023
- 2023-03-08 US US18/180,438 patent/US20230365594A1/en active Pending
- 2023-10-09 CO CONC2023/0013397A patent/CO2023013397A2/es unknown
- 2023-10-09 DO DO2023000219A patent/DOP2023000219A/es unknown
Also Published As
Publication number | Publication date |
---|---|
EP4323369A1 (en) | 2024-02-21 |
CA3214808A1 (en) | 2022-10-20 |
WO2022221642A1 (en) | 2022-10-20 |
JP2024513945A (ja) | 2024-03-27 |
IL307203A (en) | 2023-11-01 |
TW202302598A (zh) | 2023-01-16 |
US11661431B2 (en) | 2023-05-30 |
US20220389034A1 (en) | 2022-12-08 |
KR20230171469A (ko) | 2023-12-20 |
DOP2023000219A (es) | 2023-11-15 |
US20230365594A1 (en) | 2023-11-16 |
AU2022257039A1 (en) | 2023-10-05 |
CO2023013397A2 (es) | 2023-10-30 |
CR20230478A (es) | 2023-11-30 |
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