BR112013023279A2 - formas sólidas de 3-(-5-amino-2-metil-4-oxo-4h-quinazolin-3-il)-piperidina-2,6-diona e suas composições farmacêuticas e usos - Google Patents

formas sólidas de 3-(-5-amino-2-metil-4-oxo-4h-quinazolin-3-il)-piperidina-2,6-diona e suas composições farmacêuticas e usos

Info

Publication number
BR112013023279A2
BR112013023279A2 BR112013023279A BR112013023279A BR112013023279A2 BR 112013023279 A2 BR112013023279 A2 BR 112013023279A2 BR 112013023279 A BR112013023279 A BR 112013023279A BR 112013023279 A BR112013023279 A BR 112013023279A BR 112013023279 A2 BR112013023279 A2 BR 112013023279A2
Authority
BR
Brazil
Prior art keywords
quinazolin
dione
piperidine
oxo
amino
Prior art date
Application number
BR112013023279A
Other languages
English (en)
Inventor
Benjamin M Cohen
George W Muller
Hon-Wah Man
Jean Xu
William W Leong
Ying Li
Original Assignee
Celgene Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45888486&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR112013023279(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Celgene Corp filed Critical Celgene Corp
Publication of BR112013023279A2 publication Critical patent/BR112013023279A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Abstract

abstract not avaible
BR112013023279A 2011-03-11 2012-03-09 formas sólidas de 3-(-5-amino-2-metil-4-oxo-4h-quinazolin-3-il)-piperidina-2,6-diona e suas composições farmacêuticas e usos BR112013023279A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161451806P 2011-03-11 2011-03-11
PCT/US2012/028419 WO2012125438A1 (en) 2011-03-11 2012-03-09 Solid forms of 3-(5-amino-2methyl-4-oxo-4h-quinazolin-3-yl)-piperidine-2,6-dione, and their pharmaceutical compositions and uses

Publications (1)

Publication Number Publication Date
BR112013023279A2 true BR112013023279A2 (pt) 2016-12-20

Family

ID=45888486

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112013023279A BR112013023279A2 (pt) 2011-03-11 2012-03-09 formas sólidas de 3-(-5-amino-2-metil-4-oxo-4h-quinazolin-3-il)-piperidina-2,6-diona e suas composições farmacêuticas e usos

Country Status (34)

Country Link
US (5) US8802685B2 (pt)
EP (2) EP3309153A1 (pt)
JP (1) JP5959543B2 (pt)
KR (1) KR20140014221A (pt)
CN (2) CN106083812A (pt)
AR (1) AR085650A1 (pt)
AU (2) AU2012229279B2 (pt)
BR (1) BR112013023279A2 (pt)
CA (3) CA2829570C (pt)
CL (1) CL2013002593A1 (pt)
CO (1) CO6821939A2 (pt)
CR (2) CR20130458A (pt)
CY (1) CY1119974T1 (pt)
DK (1) DK2683708T3 (pt)
EA (1) EA026100B1 (pt)
EC (1) ECSP13012877A (pt)
ES (1) ES2656855T3 (pt)
HR (1) HRP20180133T1 (pt)
HU (1) HUE037955T2 (pt)
LT (1) LT2683708T (pt)
MX (1) MX2013010360A (pt)
NI (1) NI201300080A (pt)
NO (1) NO2683708T3 (pt)
PE (1) PE20140983A1 (pt)
PL (1) PL2683708T3 (pt)
PT (1) PT2683708T (pt)
RS (1) RS56770B1 (pt)
RU (1) RU2611007C2 (pt)
SG (1) SG192946A1 (pt)
SI (1) SI2683708T1 (pt)
TW (2) TWI601722B (pt)
UA (1) UA113512C2 (pt)
WO (1) WO2012125438A1 (pt)
ZA (1) ZA201306234B (pt)

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JP2021514193A (ja) 2018-02-21 2021-06-10 セルジーン コーポレイション Ｂｃｍａ結合抗体及びその使用
RU2695326C1 (ru) * 2018-06-05 2019-07-23 Федеральное государственное бюджетное научное учреждение "Научно-исследовательский институт биомедицинской химии имени В.Н. Ореховича" (ИБМХ) Противоопухолевое средство для лечения рака предстательной железы в форме саше
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