BR112015020584A2 - métodos para o tratamento de artrite psoriática usando apremilast - Google Patents

métodos para o tratamento de artrite psoriática usando apremilast

Info

Publication number
BR112015020584A2
BR112015020584A2 BR112015020584A BR112015020584A BR112015020584A2 BR 112015020584 A2 BR112015020584 A2 BR 112015020584A2 BR 112015020584 A BR112015020584 A BR 112015020584A BR 112015020584 A BR112015020584 A BR 112015020584A BR 112015020584 A2 BR112015020584 A2 BR 112015020584A2
Authority
BR
Brazil
Prior art keywords
apremilast
methods
psoriatic arthritis
treating psoriatic
treating
Prior art date
Application number
BR112015020584A
Other languages
English (en)
Inventor
Day Robert
Original Assignee
Celgene Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50549444&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR112015020584(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Celgene Corp filed Critical Celgene Corp
Publication of BR112015020584A2 publication Critical patent/BR112015020584A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/4035Isoindoles, e.g. phthalimide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis

Abstract

resumo “métodos para o tratamento de artrite psoriática usando apremilast” métodos de tratamento, gerenciamento ou prevenção de artrite psoriática são divulgados. métodos específicos englobam a administração de apremilast, isoladamente ou em combinação com um segundo agente ativo. 1/1
BR112015020584A 2013-03-14 2014-03-13 métodos para o tratamento de artrite psoriática usando apremilast BR112015020584A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361782880P 2013-03-14 2013-03-14
PCT/US2014/025171 WO2014151180A1 (en) 2013-03-14 2014-03-13 Treatment of psoriatic arthritis using apremilast

Publications (1)

Publication Number Publication Date
BR112015020584A2 true BR112015020584A2 (pt) 2017-07-18

Family

ID=50549444

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112015020584A BR112015020584A2 (pt) 2013-03-14 2014-03-13 métodos para o tratamento de artrite psoriática usando apremilast

Country Status (10)

Country Link
US (1) US9872854B2 (pt)
KR (1) KR20150126618A (pt)
CN (1) CN105050624A (pt)
AU (1) AU2014235273A1 (pt)
BR (1) BR112015020584A2 (pt)
HK (1) HK1215671A1 (pt)
IL (1) IL239499A0 (pt)
MX (1) MX2015008685A (pt)
NZ (1) NZ628320A (pt)
WO (1) WO2014151180A1 (pt)

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SG192946A1 (en) 2011-03-11 2013-09-30 Celgene Corp Solid forms of 3-(5-amino-2methyl-4-oxo-4h-quinazolin-3-yl)-piperidine-2,6-dione, and their pharmaceutical compositions and uses
CN104755472A (zh) 2012-09-04 2015-07-01 细胞基因公司 3-(5-氨基-2-甲基-4-氧代喹唑啉-3(4h)-基)哌啶-2,6-二酮的同位素体及其制备方法
WO2014116573A1 (en) 2013-01-22 2014-07-31 Celgene Corporation Processes for the preparation of isotopologues of 3-(4-((4-(morpholinomethyl)benzyl)oxy)-1-oxoisoindolin-2-yl)piperidine-2,6-dione and pharmaceutically acceptable salts thereof
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CN105588886B (zh) * 2014-11-18 2020-01-31 重庆医药工业研究院有限责任公司 一种采用液相色谱法测定阿普斯特及其制剂中杂质的方法
CN104458961A (zh) * 2014-12-11 2015-03-25 南京艾德凯腾生物医药有限责任公司 阿普斯特有关物质检测方法
US10287248B2 (en) 2015-03-19 2019-05-14 Cipla Limited Process for the preparation of apremilast
CN106727344A (zh) * 2015-11-19 2017-05-31 常州爱诺新睿医药技术有限公司 一种无定型阿普斯特的固体分散体及其制备方法
US10765665B2 (en) 2015-11-24 2020-09-08 Melin Jeffrey Composition comprising combination of rapamycin and an activator of AMP kinase and use thereof for treating diseases
CN105935350B (zh) * 2015-12-18 2018-11-16 重庆两江药物研发中心有限公司 一种阿普斯特缓释植入剂及其制备方法
US20200170999A1 (en) * 2015-12-24 2020-06-04 Jiangsu Hengrui Medicine Co., Ltd. Apremilast sustained release preparation
CN108181401B (zh) * 2018-01-26 2020-07-31 华侨大学 一种阿普斯特片有效成分的含量测定方法
CN109568302B (zh) * 2018-11-01 2021-07-16 郑州大学第一附属医院 一种治疗晚期肝癌的药物复合物及其应用
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IL287665A (en) * 2019-04-30 2022-07-01 Celgene Corp Combined treatments including apremilaste and tyk2 inhibitors
US20210315883A1 (en) * 2020-04-08 2021-10-14 Nostrum Pharmaceuticals, Llc Compositions and methods for the prophylaxis and/or treatment of viral infections or conditions associated therewith
WO2023105286A1 (en) 2021-12-06 2023-06-15 My Personal Therapeutics Ltd A combination treatment for cancer
WO2023121670A1 (en) * 2021-12-23 2023-06-29 Amgen Inc. Oral suspension of apremilast
CN116019762A (zh) * 2022-09-19 2023-04-28 厦门大学 一种用于治疗银屑病的药物组合物、制备方法和用途

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Also Published As

Publication number Publication date
CN105050624A (zh) 2015-11-11
AU2014235273A2 (en) 2015-07-23
KR20150126618A (ko) 2015-11-12
IL239499A0 (en) 2015-08-31
AU2014235273A1 (en) 2015-07-09
US20140301980A1 (en) 2014-10-09
WO2014151180A1 (en) 2014-09-25
NZ628320A (en) 2017-04-28
HK1215671A1 (zh) 2016-09-09
MX2015008685A (es) 2015-10-05
US9872854B2 (en) 2018-01-23
US20150174100A2 (en) 2015-06-25

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]
B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]