NI201300080A - Formas sólidas de 3 - ( 5 - amino - 2 - metil - 4 - oxo - 4h - quinazolin - 3 - il ) - piperidin - 2, 6 - diona, y sus composiciones farmacéuticas y usos - Google Patents

Formas sólidas de 3 - ( 5 - amino - 2 - metil - 4 - oxo - 4h - quinazolin - 3 - il ) - piperidin - 2, 6 - diona, y sus composiciones farmacéuticas y usos

Info

Publication number
NI201300080A
NI201300080A NI201300080A NI201300080A NI201300080A NI 201300080 A NI201300080 A NI 201300080A NI 201300080 A NI201300080 A NI 201300080A NI 201300080 A NI201300080 A NI 201300080A NI 201300080 A NI201300080 A NI 201300080A
Authority
NI
Nicaragua
Prior art keywords
quinazolin
piperidin
oxo
amino
methyl
Prior art date
Application number
NI201300080A
Other languages
English (en)
Inventor
W Muller George
- Wah Man Hon
M Cohen Benjamin
Li Ying
Xu Jean
W Leong William
Original Assignee
Celgene Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45888486&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NI201300080(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Celgene Corp filed Critical Celgene Corp
Publication of NI201300080A publication Critical patent/NI201300080A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Se describen formas sólidas que comprenden 3 - ( 5 - amino - 2 - metil - 4 - oxo - 4H - quinazolin - 3 - il ) - piperidin - 2, 6 - diona, composiciones que comprenden las formas sólidas, métodos para elaborar las formas sólidas y métodos para sus usos.
NI201300080A 2011-03-11 2013-09-09 Formas sólidas de 3 - ( 5 - amino - 2 - metil - 4 - oxo - 4h - quinazolin - 3 - il ) - piperidin - 2, 6 - diona, y sus composiciones farmacéuticas y usos NI201300080A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201161451806P 2011-03-11 2011-03-11

Publications (1)

Publication Number Publication Date
NI201300080A true NI201300080A (es) 2014-02-25

Family

ID=45888486

Family Applications (1)

Application Number Title Priority Date Filing Date
NI201300080A NI201300080A (es) 2011-03-11 2013-09-09 Formas sólidas de 3 - ( 5 - amino - 2 - metil - 4 - oxo - 4h - quinazolin - 3 - il ) - piperidin - 2, 6 - diona, y sus composiciones farmacéuticas y usos

Country Status (34)

Country Link
US (5) US8802685B2 (es)
EP (2) EP3309153A1 (es)
JP (1) JP5959543B2 (es)
KR (1) KR20140014221A (es)
CN (2) CN106083812A (es)
AR (1) AR085650A1 (es)
AU (2) AU2012229279B2 (es)
BR (1) BR112013023279A2 (es)
CA (3) CA3037184C (es)
CL (1) CL2013002593A1 (es)
CO (1) CO6821939A2 (es)
CR (2) CR20130458A (es)
CY (1) CY1119974T1 (es)
DK (1) DK2683708T3 (es)
EA (1) EA026100B1 (es)
EC (1) ECSP13012877A (es)
ES (1) ES2656855T3 (es)
HR (1) HRP20180133T1 (es)
HU (1) HUE037955T2 (es)
LT (1) LT2683708T (es)
MX (1) MX2013010360A (es)
NI (1) NI201300080A (es)
NO (1) NO2683708T3 (es)
PE (1) PE20140983A1 (es)
PL (1) PL2683708T3 (es)
PT (1) PT2683708T (es)
RS (1) RS56770B1 (es)
RU (1) RU2611007C2 (es)
SG (1) SG192946A1 (es)
SI (1) SI2683708T1 (es)
TW (2) TWI540127B (es)
UA (1) UA113512C2 (es)
WO (1) WO2012125438A1 (es)
ZA (1) ZA201306234B (es)

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WO2017205622A1 (en) * 2016-05-25 2017-11-30 Savant Neglected Diseases, Llc Method of making benznidazole
JP2021514193A (ja) 2018-02-21 2021-06-10 セルジーン コーポレイション Ｂｃｍａ結合抗体及びその使用
RU2695326C1 (ru) * 2018-06-05 2019-07-23 Федеральное государственное бюджетное научное учреждение "Научно-исследовательский институт биомедицинской химии имени В.Н. Ореховича" (ИБМХ) Противоопухолевое средство для лечения рака предстательной железы в форме саше
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