BR0317176A - Processo para a sìntese de peptìdeos contendo uma subestrutura de 4-hidróxi-prolina - Google Patents

Processo para a sìntese de peptìdeos contendo uma subestrutura de 4-hidróxi-prolina

Info

Publication number
BR0317176A
BR0317176A BR0317176-0A BR0317176A BR0317176A BR 0317176 A BR0317176 A BR 0317176A BR 0317176 A BR0317176 A BR 0317176A BR 0317176 A BR0317176 A BR 0317176A
Authority
BR
Brazil
Prior art keywords
peptides containing
synthesizing peptides
hydroxy proline
substructure
proline substructure
Prior art date
Application number
BR0317176-0A
Other languages
English (en)
Inventor
Bernhard Wietfeld
Walter Prikoszovich
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0229020A external-priority patent/GB0229020D0/en
Priority claimed from GB0229280A external-priority patent/GB0229280D0/en
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BR0317176A publication Critical patent/BR0317176A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
    • C07C51/347—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
    • C07C51/15—Preparation of carboxylic acids or their salts, halides or anhydrides by reaction of organic compounds with carbon dioxide, e.g. Kolbe-Schmitt synthesis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C65/00—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C65/01—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing hydroxy or O-metal groups
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
  • Pyrrole Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

"PROCESSO PARA A SìNTESE DE PEPTìDEOS CONTENDO UMA SUBESTRUTURA DE 4-HIDRóXI-PROLINA". A presente invenção refere-se a processos para preparo de peptídeos e a intermediários envolvidos em tais processos, por exemplo um processo para preparo de um composto de fórmula VIII em que R~ 12~ e R~ 13~ são como definidos aqui.
BR0317176-0A 2002-12-12 2003-12-11 Processo para a sìntese de peptìdeos contendo uma subestrutura de 4-hidróxi-prolina BR0317176A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0229020A GB0229020D0 (en) 2002-12-12 2002-12-12 Organic compounds
GB0229280A GB0229280D0 (en) 2002-12-16 2002-12-16 Organic compounds
PCT/EP2003/014082 WO2004052817A1 (en) 2002-12-12 2003-12-11 Process for peptide synthesis of peptides containing a 4-hydroxy-proline substructure

Publications (1)

Publication Number Publication Date
BR0317176A true BR0317176A (pt) 2005-10-25

Family

ID=32510405

Family Applications (2)

Application Number Title Priority Date Filing Date
BR0317176-0A BR0317176A (pt) 2002-12-12 2003-12-11 Processo para a sìntese de peptìdeos contendo uma subestrutura de 4-hidróxi-prolina
BRPI0317176-0A BRPI0317176B1 (pt) 2002-12-12 2003-12-11 Processo para a síntese de peptídeos contendo uma subestrutura de 4-hidróxi-prolina

Family Applications After (1)

Application Number Title Priority Date Filing Date
BRPI0317176-0A BRPI0317176B1 (pt) 2002-12-12 2003-12-11 Processo para a síntese de peptídeos contendo uma subestrutura de 4-hidróxi-prolina

Country Status (24)

Country Link
US (3) US7294722B2 (pt)
EP (1) EP1572615B8 (pt)
JP (2) JP4796303B2 (pt)
KR (1) KR101018491B1 (pt)
AT (1) ATE461173T1 (pt)
AU (1) AU2003290019B2 (pt)
BR (2) BR0317176A (pt)
CA (1) CA2509363C (pt)
CO (1) CO5700810A2 (pt)
CY (1) CY1110639T1 (pt)
DE (1) DE60331770D1 (pt)
DK (1) DK1572615T3 (pt)
EC (1) ECSP055846A (pt)
ES (1) ES2341336T3 (pt)
HK (1) HK1085459A1 (pt)
IL (1) IL168866A (pt)
MX (1) MXPA05006267A (pt)
NO (1) NO331836B1 (pt)
NZ (1) NZ540441A (pt)
PL (1) PL206914B1 (pt)
PT (1) PT1572615E (pt)
RU (1) RU2392265C2 (pt)
SI (1) SI1572615T1 (pt)
WO (1) WO2004052817A1 (pt)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4306839A1 (de) 1993-03-05 1994-09-08 Bayer Ernst Prof Dr Tritylgruppe enthaltendes Festphasensystem, Verfahren zu seiner Herstellung und seine Verwendung in Festphasenreaktionen
MY147327A (en) * 1995-06-29 2012-11-30 Novartis Ag Somatostatin peptides
GB9625167D0 (en) * 1996-12-04 1997-01-22 Sandoz Ltd Organic compounds
ATE321882T1 (de) * 1997-07-01 2006-04-15 Isis Pharmaceuticals Inc Zusammensetzungen und verfahren zur verabreichung von oligonukleotiden über die speiseröhre
GB0018891D0 (en) 2000-08-01 2000-09-20 Novartis Ag Organic compounds

Also Published As

Publication number Publication date
ATE461173T1 (de) 2010-04-15
JP2006509796A (ja) 2006-03-23
CY1110639T1 (el) 2015-04-29
HK1085459A1 (en) 2006-08-25
SI1572615T1 (sl) 2010-06-30
JP2010209077A (ja) 2010-09-24
CO5700810A2 (es) 2006-11-30
JP4796303B2 (ja) 2011-10-19
US7294722B2 (en) 2007-11-13
WO2004052817A1 (en) 2004-06-24
EP1572615B1 (en) 2010-03-17
ECSP055846A (es) 2005-09-20
US20060189814A1 (en) 2006-08-24
KR101018491B1 (ko) 2011-03-03
AU2003290019B2 (en) 2007-09-27
CA2509363A1 (en) 2004-06-24
PL375821A1 (en) 2005-12-12
CA2509363C (en) 2012-04-24
AU2003290019A1 (en) 2004-06-30
EP1572615A1 (en) 2005-09-14
IL168866A (en) 2010-12-30
NO331836B1 (no) 2012-04-16
US7449587B2 (en) 2008-11-11
EP1572615B8 (en) 2010-07-14
NO20053374L (no) 2005-09-12
RU2392265C2 (ru) 2010-06-20
PL206914B1 (pl) 2010-10-29
ES2341336T3 (es) 2010-06-18
DK1572615T3 (da) 2010-06-14
RU2005121664A (ru) 2006-02-27
DE60331770D1 (de) 2010-04-29
NO20053374D0 (no) 2005-07-11
PT1572615E (pt) 2010-04-14
KR20050085543A (ko) 2005-08-29
JP5249276B2 (ja) 2013-07-31
NZ540441A (en) 2007-10-26
US20080021225A1 (en) 2008-01-24
BRPI0317176B1 (pt) 2018-03-13
US20080312456A1 (en) 2008-12-18
MXPA05006267A (es) 2005-08-19

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: ALTERADA DA INT. CL. C07C 51/347, C07B 49/00, C07C 65/01, C07K 1/04.

Ipc: C07D 207/16 (2006.01), C07C 51/347 (2006.01), C07C

B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]
B21F Lapse acc. art. 78, item iv - on non-payment of the annual fees in time

Free format text: REFERENTE A 16A ANUIDADE.

B24J Lapse because of non-payment of annual fees (definitively: art 78 iv lpi, resolution 113/2013 art. 12)

Free format text: EM VIRTUDE DA EXTINCAO PUBLICADA NA RPI 2544 DE 08-10-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDA A EXTINCAO DA PATENTE E SEUS CERTIFICADOS, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.