BRPI0507979A - processo para preparação de um composto - Google Patents

processo para preparação de um composto

Info

Publication number
BRPI0507979A
BRPI0507979A BRPI0507979-9A BRPI0507979A BRPI0507979A BR PI0507979 A BRPI0507979 A BR PI0507979A BR PI0507979 A BRPI0507979 A BR PI0507979A BR PI0507979 A BRPI0507979 A BR PI0507979A
Authority
BR
Brazil
Prior art keywords
preparing
compound
halides
preparation
heteroarylalkylsulfonyl
Prior art date
Application number
BRPI0507979-9A
Other languages
English (en)
Inventor
Ronald S Michalak
Mousumi Ghosh
Mahmut Levent
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of BRPI0507979A publication Critical patent/BRPI0507979A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/32—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of salts of sulfonic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/02—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof
    • C07C303/22—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof from sulfonic acids, by reactions not involving the formation of sulfo or halosulfonyl groups; from sulfonic halides by reactions not involving the formation of halosulfonyl groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

"PROCESSO PAR PREPARAçãO DE UM COMPOSTO" A presente invenção próve processos para a preparação de halogenetos de arilalquilsulfonila e halogenetos de heteroarilalquilsulfonila de fórmula: Ar-R-SO~2~-X,que são úteis como intermediários na preparação de produtos farmacêuticos.
BRPI0507979-9A 2004-02-25 2005-02-23 processo para preparação de um composto BRPI0507979A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US54760004P 2004-02-25 2004-02-25
PCT/US2005/005624 WO2005082843A1 (en) 2004-02-25 2005-02-23 Processes for the preparation of aryl-and heteroaryl-alkylsulfonyl halides

Publications (1)

Publication Number Publication Date
BRPI0507979A true BRPI0507979A (pt) 2007-07-24

Family

ID=34910921

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0507979-9A BRPI0507979A (pt) 2004-02-25 2005-02-23 processo para preparação de um composto

Country Status (24)

Country Link
US (1) US7321061B2 (pt)
EP (1) EP1718605B1 (pt)
JP (1) JP2007523954A (pt)
CN (1) CN1922136A (pt)
AR (1) AR048239A1 (pt)
AT (1) ATE433955T1 (pt)
AU (1) AU2005217619A1 (pt)
BR (1) BRPI0507979A (pt)
CA (1) CA2555247A1 (pt)
CO (1) CO5720992A2 (pt)
CR (1) CR8550A (pt)
DE (1) DE602005014942D1 (pt)
EC (1) ECSP066797A (pt)
ES (1) ES2326746T3 (pt)
GT (1) GT200500031A (pt)
IL (1) IL177432A0 (pt)
NO (1) NO20063611L (pt)
PA (1) PA8624401A1 (pt)
PE (1) PE20060018A1 (pt)
RU (1) RU2006129650A (pt)
SV (1) SV2005002015A (pt)
TW (1) TW200602298A (pt)
WO (1) WO2005082843A1 (pt)
ZA (1) ZA200607097B (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101228118B (zh) 2005-07-21 2013-09-18 惠氏公司 由磺酸盐合成磺酰卤和磺酰胺的方法
JP2010508304A (ja) * 2006-10-31 2010-03-18 ワイス エルエルシー ホスホリパーゼ酵素阻害剤の半固体製剤
US20100113443A1 (en) * 2006-10-31 2010-05-06 Wyeth Liquid formulations of phospholipase enzyme inhibitors
EP2459523A2 (en) * 2009-07-30 2012-06-06 Dow Global Technologies LLC Improved process for the sulfochlorination of hydrocarbons
CN102241613B (zh) * 2011-05-09 2013-06-05 南通维立科化工有限公司 甲基磺酸钠制备高纯度甲基磺酰氯的生产方法
CN102295587A (zh) * 2011-05-26 2011-12-28 安徽丰乐农化有限责任公司 对甲基苯磺酰氯的制备新工艺
CN102976988B (zh) * 2012-12-24 2014-06-18 三门峡奥科化工有限公司 2-萘硫酚的合成工艺
KR102122111B1 (ko) * 2017-09-01 2020-06-11 주식회사 엘지화학 대체 용매의 선정 방법
CN111718286A (zh) * 2020-07-23 2020-09-29 邓博天 一种带供电基团芳烃磺酰氯的工业化生产方法

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE48722C (de) * Dr. E. FISCHER in Stuttgart, Schlofsstrafse 29 Verfahren zur Darstellung von O-Nitrobenzaldehyd aus O-Nitrobenzylchlorid
DE150313C (pt) *
US2199568A (en) * 1938-06-11 1940-05-07 Gen Aniline & Film Corp Manufacture of 1-methyl-4-chloro-5-hydroxynaphthalene-11-sulphonic acid
US2507408A (en) 1948-03-05 1950-05-09 Rhone Poulenc Sa 1-alkylsulfonyl-4-alkyl piperazines
US2888486A (en) 1953-11-20 1959-05-26 Du Pont Process for producing aromatic sulfonyl halides
DE2545644A1 (de) * 1975-10-11 1977-04-14 Bayer Ag Verfahren zur herstellung von sulfonsaeuren
US4150049A (en) * 1975-11-05 1979-04-17 The Government Of The United States Esters of aromatic sulfonic acids
JPS5277030A (en) * 1975-12-23 1977-06-29 Toyo Pharma Kk Production of novel benzyl sulphonic acid derivatives
JPH09295962A (ja) * 1996-03-08 1997-11-18 Nagase & Co Ltd ２，２−ジ置換−エタンスルホン酸誘導体およびその塩
DE19838516A1 (de) * 1998-08-25 2000-03-09 Degussa Verfahren zur Herstellung von Sulfonylhalogeniden
JP2000072739A (ja) * 1998-09-01 2000-03-07 Tanabe Seiyaku Co Ltd スルホン酸類またはその塩の製法
DK1892239T3 (da) 2001-12-03 2013-03-25 Wyeth Llc Inhibitorer af cytosol-phospholipase A2
CN101228118B (zh) 2005-07-21 2013-09-18 惠氏公司 由磺酸盐合成磺酰卤和磺酰胺的方法

Also Published As

Publication number Publication date
NO20063611L (no) 2006-09-21
ES2326746T3 (es) 2009-10-19
EP1718605A1 (en) 2006-11-08
CO5720992A2 (es) 2007-01-31
JP2007523954A (ja) 2007-08-23
EP1718605B1 (en) 2009-06-17
IL177432A0 (en) 2006-12-10
AU2005217619A1 (en) 2005-09-09
RU2006129650A (ru) 2008-03-27
CR8550A (es) 2007-02-05
US20050187408A1 (en) 2005-08-25
DE602005014942D1 (de) 2009-07-30
ATE433955T1 (de) 2009-07-15
TW200602298A (en) 2006-01-16
CA2555247A1 (en) 2005-09-09
GT200500031A (es) 2005-09-30
PA8624401A1 (es) 2006-08-03
AR048239A1 (es) 2006-04-12
ZA200607097B (en) 2009-08-26
ECSP066797A (es) 2006-11-16
SV2005002015A (es) 2005-11-04
PE20060018A1 (es) 2006-02-20
WO2005082843A1 (en) 2005-09-09
US7321061B2 (en) 2008-01-22
CN1922136A (zh) 2007-02-28

Similar Documents

Publication Publication Date Title
BRPI0507979A (pt) processo para preparação de um composto
BRPI0516911A (pt) método para a preparação de um composto e composto de anilina
BRPI0411268A (pt) processo para a preparação de um composto 3-aril butil-amina substituìdo
BRPI0813284A8 (pt) Processo para a preparação de um composto da fórmula (i) e composto
BRPI0615705A2 (pt) processo para preparar um composto, e, composto
BRPI0811712A2 (pt) "composto, processo de preparação de um composto e composição farmacéutica".
BRPI0518459A2 (pt) composto ou um sal farmaceuticamente aceitÁvel do mesmo, composiÇço farmacÊutica, uso de um composto, e, processo para preparar o composto ou um sal farmaceuticamente aceitÁvel do mesmo
BRPI0612957B8 (pt) composto, processos de preparação de compostos, composição farmacêutica e uso de um composto
BRPI0607455A2 (pt) composto, processo para a preparação do mesmo, uso de um composto, e composição farmacêutica
BRPI0500480A (pt) processo para a sìntese de (1s)-4,5-dimetóxi- 1-(metilaminometil)-benzociclobutano e sais de adição deste, e aplicação na sìntese de ivabradina e sais de adição desta com um ácido farmaceuticamente aceitável
BRPI0714558A8 (pt) processo para a preparação de (1r,2r)-3-(3-dimetilamino-1-etil-2-metil-propil)-fenol
BRPI0518647A2 (pt) processo para a produÇço de um composto, e, composto
CR9223A (es) 18-metil-19-nor-17-pregn-4-en-21, 17-carbolactonas,asi como preparaciones farmaceuticas que las contienen
BRPI0920834A2 (pt) processo para preparação de derivados protegidos de l-alanina
BRPI0516555A (pt) processo de revestimento
BRPI0816911A8 (pt) Processo para preparação de 4-aminobut-2-enolidas
BRPI0517390A (pt) processo para a preparação de derivados de [1,4,5]-oxadiazepina
BRPI0407282A (pt) Processo para preparação de inibidores de pirrolotriazina cinase
BRPI0508430A (pt) processo para a preparação de inibidores da triptase
BR0301667A (pt) Processo para a preparação de polìmeros em emulsão com pureza elevada
BRPI0108990B8 (pt) processo para preparação de derivados de pirimidona com atividade antifungos
CR9208A (es) Procesos para la preparacion de alcoholes de aminoetoxibencilo
BRPI0506490A (pt) compostos orgánicos
BRPI0411652A (pt) processo para a preparação de derivados de espirobenzoazepina substituìdos não-peptìdicos
HU0402466D0 (en) Industrial process for preparing 17-hydroxy-6-betha, 7-betha, 15-betha, 16-betha-bis-methylene-3-oxo-17-alpha-pregn-4-ene-21-carboxylic acid gamma lacton and the main, intermediates of the process

Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 7A ANUIDADE(S).

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2166 DE 10/07/2012.