ECSP066797A - Procedimientos para la preparacion de halogenuros de aril- y heteroarilalquilsulfonilo - Google Patents
Procedimientos para la preparacion de halogenuros de aril- y heteroarilalquilsulfoniloInfo
- Publication number
- ECSP066797A ECSP066797A EC2006006797A ECSP066797A ECSP066797A EC SP066797 A ECSP066797 A EC SP066797A EC 2006006797 A EC2006006797 A EC 2006006797A EC SP066797 A ECSP066797 A EC SP066797A EC SP066797 A ECSP066797 A EC SP066797A
- Authority
- EC
- Ecuador
- Prior art keywords
- preparation
- heteroarilalquilsulfonilo
- halogenures
- aril
- procedures
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- 125000005140 aralkylsulfonyl group Chemical group 0.000 abstract 1
- -1 heteroarylalkyl sulfonyl halides Chemical class 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 239000008177 pharmaceutical agent Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/32—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of salts of sulfonic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/02—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof
- C07C303/22—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof from sulfonic acids, by reactions not involving the formation of sulfo or halosulfonyl groups; from sulfonic halides by reactions not involving the formation of halosulfonyl groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
La presente invención provee procedimientos de preparación de halogenuros de arilalquilsulfonilo y halogenuros de heteroarilalquilsulfonilo de la fórmula Ar-R-SO2-X, que son útiles como intermediarios en la preparación de agentes farmacéuticos.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US54760004P | 2004-02-25 | 2004-02-25 |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP066797A true ECSP066797A (es) | 2006-11-16 |
Family
ID=34910921
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EC2006006797A ECSP066797A (es) | 2004-02-25 | 2006-08-25 | Procedimientos para la preparacion de halogenuros de aril- y heteroarilalquilsulfonilo |
Country Status (24)
Country | Link |
---|---|
US (1) | US7321061B2 (es) |
EP (1) | EP1718605B1 (es) |
JP (1) | JP2007523954A (es) |
CN (1) | CN1922136A (es) |
AR (1) | AR048239A1 (es) |
AT (1) | ATE433955T1 (es) |
AU (1) | AU2005217619A1 (es) |
BR (1) | BRPI0507979A (es) |
CA (1) | CA2555247A1 (es) |
CO (1) | CO5720992A2 (es) |
CR (1) | CR8550A (es) |
DE (1) | DE602005014942D1 (es) |
EC (1) | ECSP066797A (es) |
ES (1) | ES2326746T3 (es) |
GT (1) | GT200500031A (es) |
IL (1) | IL177432A0 (es) |
NO (1) | NO20063611L (es) |
PA (1) | PA8624401A1 (es) |
PE (1) | PE20060018A1 (es) |
RU (1) | RU2006129650A (es) |
SV (1) | SV2005002015A (es) |
TW (1) | TW200602298A (es) |
WO (1) | WO2005082843A1 (es) |
ZA (1) | ZA200607097B (es) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BRPI0614005A2 (pt) * | 2005-07-21 | 2011-03-01 | Wyeth Corp | processo para sìntese de haletos de sulfonila e sulfonamidas a partir de sais de ácido sulfÈnico |
US20100093725A1 (en) * | 2006-10-31 | 2010-04-15 | Wyeth | Semi-solid formulations of phospholipase enzyme inhibitors |
BRPI0717943A2 (pt) * | 2006-10-31 | 2013-10-29 | Wyeth Corp | Composição farmacêutica; forma de dosagem farmacêutica; processo para a preparação de uma composição farmacêutica; e produto preparado pelo processo |
WO2011014553A2 (en) * | 2009-07-30 | 2011-02-03 | Dow Global Technologies Inc. | Improved process for the sulfochlorination of hydrocarbons |
CN102241613B (zh) * | 2011-05-09 | 2013-06-05 | 南通维立科化工有限公司 | 甲基磺酸钠制备高纯度甲基磺酰氯的生产方法 |
CN102295587A (zh) * | 2011-05-26 | 2011-12-28 | 安徽丰乐农化有限责任公司 | 对甲基苯磺酰氯的制备新工艺 |
CN102976988B (zh) * | 2012-12-24 | 2014-06-18 | 三门峡奥科化工有限公司 | 2-萘硫酚的合成工艺 |
KR102122111B1 (ko) * | 2017-09-01 | 2020-06-11 | 주식회사 엘지화학 | 대체 용매의 선정 방법 |
CN111718286A (zh) * | 2020-07-23 | 2020-09-29 | 邓博天 | 一种带供电基团芳烃磺酰氯的工业化生产方法 |
Family Cites Families (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE48722C (de) | Dr. E. FISCHER in Stuttgart, Schlofsstrafse 29 | Verfahren zur Darstellung von O-Nitrobenzaldehyd aus O-Nitrobenzylchlorid | ||
DE150313C (es) | ||||
US2199568A (en) | 1938-06-11 | 1940-05-07 | Gen Aniline & Film Corp | Manufacture of 1-methyl-4-chloro-5-hydroxynaphthalene-11-sulphonic acid |
US2507408A (en) | 1948-03-05 | 1950-05-09 | Rhone Poulenc Sa | 1-alkylsulfonyl-4-alkyl piperazines |
US2888486A (en) | 1953-11-20 | 1959-05-26 | Du Pont | Process for producing aromatic sulfonyl halides |
DE2545644A1 (de) * | 1975-10-11 | 1977-04-14 | Bayer Ag | Verfahren zur herstellung von sulfonsaeuren |
US4150049A (en) * | 1975-11-05 | 1979-04-17 | The Government Of The United States | Esters of aromatic sulfonic acids |
JPS5277030A (en) * | 1975-12-23 | 1977-06-29 | Toyo Pharma Kk | Production of novel benzyl sulphonic acid derivatives |
JPH09295962A (ja) * | 1996-03-08 | 1997-11-18 | Nagase & Co Ltd | 2,2−ジ置換−エタンスルホン酸誘導体およびその塩 |
DE19838516A1 (de) * | 1998-08-25 | 2000-03-09 | Degussa | Verfahren zur Herstellung von Sulfonylhalogeniden |
JP2000072739A (ja) * | 1998-09-01 | 2000-03-07 | Tanabe Seiyaku Co Ltd | スルホン酸類またはその塩の製法 |
DK1451154T3 (da) | 2001-12-03 | 2008-05-19 | Wyeth Corp | Inhibitorer af cytosolisk phospholipase A2 |
BRPI0614005A2 (pt) | 2005-07-21 | 2011-03-01 | Wyeth Corp | processo para sìntese de haletos de sulfonila e sulfonamidas a partir de sais de ácido sulfÈnico |
-
2005
- 2005-02-22 AR ARP050100642A patent/AR048239A1/es not_active Application Discontinuation
- 2005-02-23 AT AT05713940T patent/ATE433955T1/de not_active IP Right Cessation
- 2005-02-23 CN CNA2005800058622A patent/CN1922136A/zh active Pending
- 2005-02-23 JP JP2007500927A patent/JP2007523954A/ja active Pending
- 2005-02-23 US US11/064,241 patent/US7321061B2/en not_active Expired - Fee Related
- 2005-02-23 DE DE602005014942T patent/DE602005014942D1/de active Active
- 2005-02-23 AU AU2005217619A patent/AU2005217619A1/en not_active Abandoned
- 2005-02-23 ES ES05713940T patent/ES2326746T3/es active Active
- 2005-02-23 SV SV2005002015A patent/SV2005002015A/es not_active Application Discontinuation
- 2005-02-23 PA PA20058624401A patent/PA8624401A1/es unknown
- 2005-02-23 GT GT200500031A patent/GT200500031A/es unknown
- 2005-02-23 TW TW094105341A patent/TW200602298A/zh unknown
- 2005-02-23 PE PE2005000213A patent/PE20060018A1/es not_active Application Discontinuation
- 2005-02-23 WO PCT/US2005/005624 patent/WO2005082843A1/en active Application Filing
- 2005-02-23 BR BRPI0507979-9A patent/BRPI0507979A/pt not_active IP Right Cessation
- 2005-02-23 RU RU2006129650/04A patent/RU2006129650A/ru not_active Application Discontinuation
- 2005-02-23 CA CA002555247A patent/CA2555247A1/en not_active Abandoned
- 2005-02-23 EP EP05713940A patent/EP1718605B1/en active Active
-
2006
- 2006-08-08 CR CR8550A patent/CR8550A/es not_active Application Discontinuation
- 2006-08-09 NO NO20063611A patent/NO20063611L/no not_active Application Discontinuation
- 2006-08-10 IL IL177432A patent/IL177432A0/en unknown
- 2006-08-23 CO CO06083312A patent/CO5720992A2/es not_active Application Discontinuation
- 2006-08-24 ZA ZA200607097A patent/ZA200607097B/xx unknown
- 2006-08-25 EC EC2006006797A patent/ECSP066797A/es unknown
Also Published As
Publication number | Publication date |
---|---|
CO5720992A2 (es) | 2007-01-31 |
CA2555247A1 (en) | 2005-09-09 |
PE20060018A1 (es) | 2006-02-20 |
BRPI0507979A (pt) | 2007-07-24 |
EP1718605A1 (en) | 2006-11-08 |
RU2006129650A (ru) | 2008-03-27 |
ES2326746T3 (es) | 2009-10-19 |
AU2005217619A1 (en) | 2005-09-09 |
TW200602298A (en) | 2006-01-16 |
WO2005082843A1 (en) | 2005-09-09 |
CN1922136A (zh) | 2007-02-28 |
IL177432A0 (en) | 2006-12-10 |
CR8550A (es) | 2007-02-05 |
EP1718605B1 (en) | 2009-06-17 |
GT200500031A (es) | 2005-09-30 |
US7321061B2 (en) | 2008-01-22 |
ZA200607097B (en) | 2009-08-26 |
PA8624401A1 (es) | 2006-08-03 |
US20050187408A1 (en) | 2005-08-25 |
SV2005002015A (es) | 2005-11-04 |
NO20063611L (no) | 2006-09-21 |
JP2007523954A (ja) | 2007-08-23 |
DE602005014942D1 (de) | 2009-07-30 |
AR048239A1 (es) | 2006-04-12 |
ATE433955T1 (de) | 2009-07-15 |
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