CY1122416T1 - Φαρμακα τα οποια περιεχουν κρυσταλλικες τροποποιησεις (1r,2r)-3-(3-δimeθyλamino-1-αιθυλο-2-μεθυλο-προπυλο)-φαινολης - Google Patents
Φαρμακα τα οποια περιεχουν κρυσταλλικες τροποποιησεις (1r,2r)-3-(3-δimeθyλamino-1-αιθυλο-2-μεθυλο-προπυλο)-φαινοληςInfo
- Publication number
- CY1122416T1 CY1122416T1 CY20191101278T CY191101278T CY1122416T1 CY 1122416 T1 CY1122416 T1 CY 1122416T1 CY 20191101278 T CY20191101278 T CY 20191101278T CY 191101278 T CY191101278 T CY 191101278T CY 1122416 T1 CY1122416 T1 CY 1122416T1
- Authority
- CY
- Cyprus
- Prior art keywords
- dimethylamino
- phenol
- propyl
- ethyl
- methyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
- C07C215/46—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
- C07C215/48—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by carbon chains not further substituted by hydroxy groups
- C07C215/54—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by carbon chains not further substituted by hydroxy groups linked by carbon chains having at least three carbon atoms between the amino groups and the six-membered aromatic ring or the condensed ring system containing that ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Abstract
Η εφεύρεση αφορά κρυσταλλικές τροποποιήσεις (1R,2Ρ)-3-(3-Διμεθυλαμινο-1-αιθυλο-2-μεθυλο-προπυλο)-φαινόλης, φαρμακευτικές συνθέσεις οι οποίες περιέχουν αυτές τις τροποποιήσεις, καθώς επίσης τη χρήση αυτών.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP07023728 | 2007-12-07 | ||
PCT/EP2008/010330 WO2009071310A1 (de) | 2007-12-07 | 2008-12-05 | Kristalline modifikationen von (1r,2r)-3-(3-dimethylamino-1-ethyl-2-methyl-propyl)-phenol |
EP08857298.7A EP2240431B1 (de) | 2007-12-07 | 2008-12-05 | Kristalline modifikationen von (1r,2r)-3-(3-dimethylamino-1-ethyl-2-methyl-propyl)-phenol |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1122416T1 true CY1122416T1 (el) | 2021-01-27 |
Family
ID=39272207
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20171100414T CY1118976T1 (el) | 2007-12-07 | 2017-04-07 | Κρυσταλλικες τροποποιησεις της (1r,2r)-3-(3-διμεθυλαμινο-1-αιθυλ-2-μεθυλ-προπυλ)-φαινολης |
CY20191101278T CY1122416T1 (el) | 2007-12-07 | 2019-12-04 | Φαρμακα τα οποια περιεχουν κρυσταλλικες τροποποιησεις (1r,2r)-3-(3-δimeθyλamino-1-αιθυλο-2-μεθυλο-προπυλο)-φαινολης |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20171100414T CY1118976T1 (el) | 2007-12-07 | 2017-04-07 | Κρυσταλλικες τροποποιησεις της (1r,2r)-3-(3-διμεθυλαμινο-1-αιθυλ-2-μεθυλ-προπυλ)-φαινολης |
Country Status (14)
Country | Link |
---|---|
US (1) | US8134032B2 (el) |
EP (2) | EP2240431B1 (el) |
CN (3) | CN101939287B (el) |
CY (2) | CY1118976T1 (el) |
DK (2) | DK2240431T3 (el) |
ES (2) | ES2623413T3 (el) |
HR (2) | HRP20170481T1 (el) |
HU (2) | HUE047275T2 (el) |
IL (2) | IL206197A (el) |
LT (1) | LT2240431T (el) |
PL (2) | PL2240431T3 (el) |
PT (2) | PT3173400T (el) |
SI (2) | SI3173400T1 (el) |
WO (1) | WO2009071310A1 (el) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20100272815A1 (en) * | 2009-04-28 | 2010-10-28 | Actavis Group Ptc Ehf | Amorphous form of tapentadol hydrochloride |
US8288592B2 (en) | 2009-09-22 | 2012-10-16 | Actavis Group Ptc Ehf | Solid state forms of tapentadol salts |
US20130116333A1 (en) | 2010-05-05 | 2013-05-09 | Ratiopharm Gmbh | Solid tapentadol in non-crystalline form |
WO2012051246A1 (en) | 2010-10-12 | 2012-04-19 | Ratiopharm Gmbh | Tapentadol hydrobromide and crystalline forms thereof |
WO2013111161A2 (en) * | 2012-01-10 | 2013-08-01 | Msn Laboratories Limited | Process for the preparation of 3-aryl-2-methyl-propanamine derivatives and polymorphs thereof |
WO2014023652A1 (en) * | 2012-08-06 | 2014-02-13 | Ratiopharm Gmbh | Pharmaceutical formulation comprising tapentadol and cyclodextrin |
EP2808319A1 (en) | 2013-05-31 | 2014-12-03 | Arevipharma GmbH | 3-[3-(Dimethylamino)-1-ethyl-2-methylpropyl]phenol resin complex |
CZ307492B6 (cs) | 2014-02-04 | 2018-10-17 | Zentiva, K.S. | Pevná forma maleátu tapentadolu a způsob její přípravy |
GB2523089A (en) * | 2014-02-12 | 2015-08-19 | Azad Pharmaceutical Ingredients Ag | Stable polymorph form B of tapentadol hydrochloride |
ES2937740T3 (es) | 2016-04-19 | 2023-03-30 | Ratiopharm Gmbh | Fosfato de tapentadol cristalino |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1027666C (zh) * | 1993-02-20 | 1995-02-15 | 袁晓辉 | 高分子聚合物正温度系数热敏电阻材料 |
DE4426245A1 (de) | 1994-07-23 | 1996-02-22 | Gruenenthal Gmbh | 1-Phenyl-3-dimethylamino-propanverbindungen mit pharmakologischer Wirkung |
PE20030527A1 (es) * | 2001-10-24 | 2003-07-26 | Gruenenthal Chemie | Formulacion farmaceutica con liberacion retardada que contiene 3-(3-dimetilamino-1-etil-2-metil-propil) fenol o una sal farmaceuticamente aceptable del mismo y tabletas para administracion oral que la contienen |
DE10326097A1 (de) * | 2003-06-06 | 2005-01-05 | Grünenthal GmbH | Verfahren zur Herstellung von Dimethyl-(3-aryl-butyl)-aminverbindungen |
ES2291780T3 (es) * | 2004-06-28 | 2008-03-01 | Grunenthal Gmbh | Formas cristalinas del clorhidrato de (-)-(1r,2r)-3-(3-dimetilamino-1-etil-2-metilpropil)fenol. |
DE102005034974A1 (de) * | 2005-07-22 | 2007-04-19 | Grünenthal GmbH | Salz von Dimethylaminomethyl-phenyl-cyclohexan und dessen kristalline Formen |
US20070254960A1 (en) * | 2006-04-28 | 2007-11-01 | Gruenenthal Gmbh | Pharmaceutical combination |
-
2008
- 2008-12-05 DK DK08857298.7T patent/DK2240431T3/en active
- 2008-12-05 CN CN200880126383.XA patent/CN101939287B/zh active Active
- 2008-12-05 HU HUE16203848A patent/HUE047275T2/hu unknown
- 2008-12-05 PL PL08857298T patent/PL2240431T3/pl unknown
- 2008-12-05 SI SI200832101T patent/SI3173400T1/sl unknown
- 2008-12-05 DK DK16203848T patent/DK3173400T3/da active
- 2008-12-05 ES ES08857298.7T patent/ES2623413T3/es active Active
- 2008-12-05 PL PL16203848T patent/PL3173400T3/pl unknown
- 2008-12-05 SI SI200831791A patent/SI2240431T1/sl unknown
- 2008-12-05 US US12/329,111 patent/US8134032B2/en active Active
- 2008-12-05 CN CN201410468436.3A patent/CN104447360B/zh active Active
- 2008-12-05 PT PT162038483T patent/PT3173400T/pt unknown
- 2008-12-05 CN CN201410468681.4A patent/CN104447361B/zh active Active
- 2008-12-05 HU HUE08857298A patent/HUE031126T2/en unknown
- 2008-12-05 ES ES16203848T patent/ES2764451T3/es active Active
- 2008-12-05 WO PCT/EP2008/010330 patent/WO2009071310A1/de active Application Filing
- 2008-12-05 EP EP08857298.7A patent/EP2240431B1/de active Active
- 2008-12-05 PT PT88572987T patent/PT2240431T/pt unknown
- 2008-12-05 EP EP16203848.3A patent/EP3173400B1/de active Active
- 2008-12-05 LT LTEP08857298.7T patent/LT2240431T/lt unknown
-
2010
- 2010-06-06 IL IL206197A patent/IL206197A/en active IP Right Grant
-
2015
- 2015-03-01 IL IL237478A patent/IL237478A0/en unknown
-
2017
- 2017-03-21 HR HRP20170481TT patent/HRP20170481T1/hr unknown
- 2017-04-07 CY CY20171100414T patent/CY1118976T1/el unknown
-
2019
- 2019-12-04 CY CY20191101278T patent/CY1122416T1/el unknown
-
2020
- 2020-01-16 HR HRP20200067TT patent/HRP20200067T1/hr unknown
Also Published As
Publication number | Publication date |
---|---|
EP2240431B1 (de) | 2017-01-25 |
EP3173400B1 (de) | 2019-11-06 |
EP2240431A1 (de) | 2010-10-20 |
IL237478A0 (en) | 2015-04-30 |
DK2240431T3 (en) | 2017-04-10 |
SI2240431T1 (sl) | 2017-05-31 |
HRP20170481T1 (hr) | 2017-05-19 |
HUE047275T2 (hu) | 2020-04-28 |
SI3173400T1 (sl) | 2020-01-31 |
CN104447360A (zh) | 2015-03-25 |
ES2623413T3 (es) | 2017-07-11 |
LT2240431T (lt) | 2017-04-10 |
WO2009071310A1 (de) | 2009-06-11 |
CN104447361B (zh) | 2017-04-12 |
IL206197A (en) | 2015-03-31 |
ES2764451T3 (es) | 2020-06-03 |
PT2240431T (pt) | 2017-05-03 |
DK3173400T3 (da) | 2019-11-25 |
HUE031126T2 (en) | 2017-07-28 |
EP3173400A1 (de) | 2017-05-31 |
HRP20200067T1 (hr) | 2020-04-03 |
PL3173400T3 (pl) | 2020-05-18 |
CY1118976T1 (el) | 2018-01-10 |
IL206197A0 (en) | 2010-12-30 |
CN104447361A (zh) | 2015-03-25 |
CN101939287A (zh) | 2011-01-05 |
CN101939287B (zh) | 2014-10-22 |
PL2240431T3 (pl) | 2017-07-31 |
US20090149534A1 (en) | 2009-06-11 |
US8134032B2 (en) | 2012-03-13 |
CN104447360B (zh) | 2017-04-12 |
PT3173400T (pt) | 2019-12-13 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CY1122416T1 (el) | Φαρμακα τα οποια περιεχουν κρυσταλλικες τροποποιησεις (1r,2r)-3-(3-δimeθyλamino-1-αιθυλο-2-μεθυλο-προπυλο)-φαινολης | |
CY1124873T1 (el) | Διεργασια για την παρασκευη (1r,2r)-3-(3-διμεθυλαμινο-1-αιθυλο-2-μεθυλο-προπυλο)-φαινολης | |
CY1106929T1 (el) | Κρυσταλλικες μορφες υδροχλωριδιου (-)-(1r,2r)-3-(3-διμεθυλαμινο-1-αιθυλο-2-μεθυλοπροπυλο)-φαινολης | |
EA201190235A1 (ru) | Замещенные 1-цианоэтилгетероциклилкарбоксамидные соединения 750 | |
CL2012002944A1 (es) | Compuestos derivados de amino-pirimidinas; composiciones farmacéuticas que los comprenden; y su uso para el tratamiento de una enfermedad afección seleccionada de trastornos neuromusculares, esclerosis lateral amiotrófica, miastenia grave, entre otras. | |
CL2012002945A1 (es) | Compuestos derivados de amino-piridazinas; composiciones farmacéuticas que los comprenden; y su uso para el tratamiento de una enfermedad afección seleccionada de trastornos neuromusculares, esclerosis lateral amiotrófica, miastenia grave, entre otras. | |
EA201170772A1 (ru) | Органические соединения | |
UY30498A1 (es) | Nueva clase de compuestos de benzimidazolilo, sus sales, composiciones farmacéuticas conteniéndolos y aplicaciones | |
CY1115455T1 (el) | Χρησιμοποιηση ενωσεων 1-φαινυλο-3-διμεθυλαμινο-προπανιου για τη θεραπεια του πονου νευροπαθειας | |
EA201401193A1 (ru) | Триарильные соединения и композиции, их содержащие | |
ATE528989T1 (de) | Kristalline feste rasagilin-base | |
EA200870599A1 (ru) | Стабильные препараты лаквинимода | |
EA201170441A1 (ru) | Терапевтические противовирусные пептиды | |
EA201300242A1 (ru) | Фармацевтические композиции, содержащие замещенные ациланилиды | |
BRPI0908637B8 (pt) | composto e composição farmacêutica do mesmo | |
UY31524A1 (es) | Nuevos compuestos 010 | |
MX2009011165A (es) | Formulaciones farmaceuticas que contienen derivados del acido lipoico. | |
EA200970532A1 (ru) | Фумаратная соль (альфа s, бета r)-6-бром-альфа-[2-(диметиламино)этил]-2-метокси-альфа-1-нафталенил-бета-фенил-3-хинолинэтанола | |
SE0401762D0 (sv) | Novel compounds | |
EA200801414A1 (ru) | Кальцилитические соединения | |
EA201001855A1 (ru) | Соединения, содержащие циклобутоксигруппу | |
EA201200616A1 (ru) | Производные 2-оксо-1-пирролидинилимидазотиадиазола | |
UY30451A1 (es) | 18-metil-19-nor-androst-4-en-17,17-espiroéteres (18-metil-19-nor-20-espirox-4-en-3-onas),ase como preparaciones farmacéuticas que lo contienen. | |
EA200900958A1 (ru) | Препарат невирапина пролонгированного высвобождения | |
CO6321280A2 (es) | Nueva clase espiro piperidinas para el tratamiento de enfermedades neurodegenerativas |