BR0116326A - Compostos orgânicos - Google Patents

Compostos orgânicos

Info

Publication number
BR0116326A
BR0116326A BR0116326-4A BR0116326A BR0116326A BR 0116326 A BR0116326 A BR 0116326A BR 0116326 A BR0116326 A BR 0116326A BR 0116326 A BR0116326 A BR 0116326A
Authority
BR
Brazil
Prior art keywords
organic compounds
compounds
endoparasites
warm
formula
Prior art date
Application number
BR0116326-4A
Other languages
English (en)
Portuguese (pt)
Inventor
Pierre Ducray
Jacques Bouvier
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BR0116326A publication Critical patent/BR0116326A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • A61K31/277Nitriles; Isonitriles having a ring, e.g. verapamil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Paper (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BR0116326-4A 2000-12-20 2001-12-18 Compostos orgânicos BR0116326A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH24892000 2000-12-20
PCT/EP2001/014926 WO2002049641A2 (en) 2000-12-20 2001-12-18 Anti-endoparasitic amidoacetonitrils

Publications (1)

Publication Number Publication Date
BR0116326A true BR0116326A (pt) 2004-07-06

Family

ID=4569596

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0116326-4A BR0116326A (pt) 2000-12-20 2001-12-18 Compostos orgânicos

Country Status (21)

Country Link
US (1) US7700656B2 (enExample)
EP (1) EP1392281B1 (enExample)
JP (1) JP2004521097A (enExample)
KR (1) KR100850252B1 (enExample)
CN (1) CN1531426A (enExample)
AR (1) AR035523A1 (enExample)
AT (1) ATE354360T1 (enExample)
AU (2) AU2002234588B2 (enExample)
BR (1) BR0116326A (enExample)
CA (1) CA2432388C (enExample)
CY (1) CY1106509T1 (enExample)
DE (1) DE60126838T2 (enExample)
DK (1) DK1392281T3 (enExample)
ES (1) ES2281453T3 (enExample)
MX (1) MXPA03005701A (enExample)
NZ (1) NZ526538A (enExample)
PT (1) PT1392281E (enExample)
RU (1) RU2286775C2 (enExample)
TW (1) TWI292712B (enExample)
WO (1) WO2002049641A2 (enExample)
ZA (1) ZA200304331B (enExample)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR035531A1 (es) * 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
AR036054A1 (es) * 2001-06-15 2004-08-04 Novartis Ag Uso de compuestos de aminoacetonitrilo para el control de plagas, una composicion y un proceso para dicho control y una composicion farmaceutica contra parasitos
WO2003004474A1 (en) * 2001-07-06 2003-01-16 Syngenta Participations Ag Pesticidally active aminoacetonitriles
AR037746A1 (es) * 2001-12-06 2004-12-01 Novartis Ag Compuestos derivados de amidoacetonitrilo, un procedimiento para su preparacion, un procedimiento para la preparacion de compuestos intermediarios, una composicion para combatir parasitos, un procedimiento para combatir dichos parasitos, y el empleo de dichos derivados para la preparacion de una com
AR039020A1 (es) * 2002-03-21 2005-02-02 Novartis Ag Compuestos de aminoacetonitrilo
TW200400932A (en) * 2002-06-19 2004-01-16 Novartis Ag Organic compounds
AR042420A1 (es) 2002-09-11 2005-06-22 Novartis Ag Benzotriazolil- aminoacetonitril compuestos, proceso para su preparacion, metodo y uso de los mismos en el control de endo- y ecto-parasitos dentro y sobre ganado productor de sangre caliente y animales domesticos y plantas, y en la preparacion de una composicion farmaceutica
GB0402677D0 (en) * 2003-11-06 2004-03-10 Novartis Ag Organic compounds
DE10358525A1 (de) * 2003-12-13 2005-07-07 Bayer Healthcare Ag Endoparasitizide Mittel zur topischen Applikation
AR049391A1 (es) 2004-06-10 2006-07-26 Novartis Ag Derivados de aminoacetonitrilo y su uso para controlar parasitos en animales de sangre caliente
WO2006043654A1 (ja) * 2004-10-22 2006-04-27 Nihon Nohyaku Co., Ltd. アセトニトリル誘導体及び有害生物防除剤並びにその使用方法
EP1812385B1 (en) * 2004-11-09 2012-07-18 Novartis AG Process for the preparation of enantiomers of amidoacetonitrile compounds from their racemates
EP1910278A1 (en) * 2005-07-25 2008-04-16 Novartis AG Amidonitrile compounds
DE102006025874A1 (de) 2006-06-02 2007-12-06 Bayer Cropscience Ag Alkoxyalkyl-substituierte cyclische Ketoenole
WO2008062005A1 (en) * 2006-11-24 2008-05-29 Novartis Ag The use of aminoacetonitril compounds in the control of endoparasites in warm- blood animals.
BRPI0807137A2 (pt) * 2007-02-09 2014-04-15 Pfizer Ltd Agentes antiparasitários
JP5327876B2 (ja) * 2007-02-21 2013-10-30 ゾエティス・ユーケイ・リミテッド ベンゾフラン抗寄生虫剤
KR101472649B1 (ko) 2007-05-15 2014-12-16 메리얼 리미티드 아릴로아졸-2-일 시아노에틸아미노 화합물, 이의 제조방법 및 이의 사용방법
WO2010048191A1 (en) 2008-10-21 2010-04-29 Merial Limited Thioamide compounds, method of making and method of using thereof
RS58508B1 (sr) 2008-11-14 2019-04-30 Merial Inc Enantiomerno obogaćena paraziticidalna jedinjenja ariloazol-2-il cijanoetilamino
UY33282A (es) * 2010-03-25 2011-09-30 Novartis Ag Composiciones endoparasiticidas
ES2625990T3 (es) * 2011-03-02 2017-07-21 The University Of Tokyo Agente de control de endoparásitos
AR088984A1 (es) * 2011-11-25 2014-07-23 Bayer Ip Gmbh Aril y/o heteroaril carboxamidas utiles como endoparasiticidas en animales o seres humanos
BR112014018875A8 (pt) 2012-02-14 2017-07-11 Nippon Soda Co Composto de ariloxiacetamida ou sal do mesmo, pesticida, acaricida ou inseticida, e, agente de controle de ectoparasita
US9790176B2 (en) 2012-08-06 2017-10-17 Pitney Pharmaceuticals Pty Limited Compounds for the treatment of mTOR pathway related diseases
US8822689B2 (en) 2012-09-19 2014-09-02 Merial Limited Aryloazol-2-yl cyanoethylamino compounds, method of making and method of using thereof
AR094961A1 (es) 2013-03-15 2015-09-09 Lilly Co Eli 1-hidroxi-benzooxaboroles como agentes antiparasitarios
EP2821412A1 (en) * 2013-07-01 2015-01-07 Universität Zürich Organometallic 2-cyano-2-aminobenzoate-propyl derivates and their use as anthelmintics
WO2015037747A1 (en) * 2013-09-13 2015-03-19 Nihon Nohyaku Co., Ltd. Anticancer agent comprising aminoacetonitrile compound as active ingredient
AU2016224395A1 (en) * 2015-02-24 2017-08-31 Pitney Pharmaceuticals Pty Limited Anti cancer agent comprising aminoacetonitrile compound as active ingredient
EP3235815A1 (de) 2016-04-19 2017-10-25 Philipps-Universität Marburg Wirkstoffe gegen parasitäre helminthen

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1520925A (fr) * 1966-04-22 1968-04-12 Abbott Lab Nouveaux benzoylamino-nitriles
US3457294A (en) * 1966-04-22 1969-07-22 Abbott Lab N-(substituted-benzoyl) aminoaceto- and aminopropionitriles
US4515731A (en) * 1975-08-25 1985-05-07 Monsanto Company Asymmetric catalysis
GB8517279D0 (en) * 1985-07-08 1985-08-14 Ici Plc Benzamide derivatives
JP2994182B2 (ja) * 1992-07-23 1999-12-27 石原産業株式会社 アミド系化合物又はその塩、それらの製造方法及びそれらを含有する有害動物防除剤
US6239077B1 (en) * 1998-05-01 2001-05-29 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof
AR035531A1 (es) * 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
EP1390344B1 (en) * 2001-05-15 2006-12-27 Novartis AG Benzamidoacetonitrile derivatives and their use as antiparasitics
AR036054A1 (es) * 2001-06-15 2004-08-04 Novartis Ag Uso de compuestos de aminoacetonitrilo para el control de plagas, una composicion y un proceso para dicho control y una composicion farmaceutica contra parasitos
WO2003004474A1 (en) * 2001-07-06 2003-01-16 Syngenta Participations Ag Pesticidally active aminoacetonitriles
AR038156A1 (es) * 2002-01-21 2004-12-29 Novartis Ag Compuestos de amidoacetonitrilo, proceso para su preparacion, composicion para controlar los parasitos, y uso de estos compuestos para preparar una composicion farmaceutica

Also Published As

Publication number Publication date
DE60126838T2 (de) 2007-11-08
US7700656B2 (en) 2010-04-20
US20040082624A1 (en) 2004-04-29
ATE354360T1 (de) 2007-03-15
CY1106509T1 (el) 2012-01-25
DK1392281T3 (da) 2007-06-11
WO2002049641A2 (en) 2002-06-27
MXPA03005701A (es) 2003-10-06
PT1392281E (pt) 2007-05-31
DE60126838D1 (de) 2007-04-05
AU2002234588B2 (en) 2005-03-24
AU3458802A (en) 2002-07-01
CN1531426A (zh) 2004-09-22
CA2432388A1 (en) 2002-06-27
CA2432388C (en) 2010-06-08
EP1392281A2 (en) 2004-03-03
TWI292712B (en) 2008-01-21
RU2003122196A (ru) 2005-03-20
KR20030061414A (ko) 2003-07-18
KR100850252B1 (ko) 2008-08-04
ZA200304331B (en) 2004-04-28
ES2281453T3 (es) 2007-10-01
WO2002049641A3 (en) 2003-12-04
JP2004521097A (ja) 2004-07-15
NZ526538A (en) 2005-12-23
AR035523A1 (es) 2004-06-02
EP1392281B1 (en) 2007-02-21
RU2286775C2 (ru) 2006-11-10

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 14A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2343 DE 01-12-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.