ATE354360T1 - Amidoacetonitrile zur bekämpfung von endoparasiten - Google Patents

Amidoacetonitrile zur bekämpfung von endoparasiten

Info

Publication number
ATE354360T1
ATE354360T1 AT01985421T AT01985421T ATE354360T1 AT E354360 T1 ATE354360 T1 AT E354360T1 AT 01985421 T AT01985421 T AT 01985421T AT 01985421 T AT01985421 T AT 01985421T AT E354360 T1 ATE354360 T1 AT E354360T1
Authority
AT
Austria
Prior art keywords
amidoacetonitriles
endoparasites
fight
fight endoparasites
Prior art date
Application number
AT01985421T
Other languages
English (en)
Inventor
Pierre Ducray
Jacques Bouvier
Original Assignee
Novartis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Pharma Gmbh filed Critical Novartis Pharma Gmbh
Application granted granted Critical
Publication of ATE354360T1 publication Critical patent/ATE354360T1/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • A61K31/277Nitriles; Isonitriles having a ring, e.g. verapamil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Paper (AREA)
AT01985421T 2000-12-20 2001-12-18 Amidoacetonitrile zur bekämpfung von endoparasiten ATE354360T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH24892000 2000-12-20

Publications (1)

Publication Number Publication Date
ATE354360T1 true ATE354360T1 (de) 2007-03-15

Family

ID=4569596

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01985421T ATE354360T1 (de) 2000-12-20 2001-12-18 Amidoacetonitrile zur bekämpfung von endoparasiten

Country Status (21)

Country Link
US (1) US7700656B2 (de)
EP (1) EP1392281B1 (de)
JP (1) JP2004521097A (de)
KR (1) KR100850252B1 (de)
CN (1) CN1531426A (de)
AR (1) AR035523A1 (de)
AT (1) ATE354360T1 (de)
AU (2) AU2002234588B2 (de)
BR (1) BR0116326A (de)
CA (1) CA2432388C (de)
CY (1) CY1106509T1 (de)
DE (1) DE60126838T2 (de)
DK (1) DK1392281T3 (de)
ES (1) ES2281453T3 (de)
MX (1) MXPA03005701A (de)
NZ (1) NZ526538A (de)
PT (1) PT1392281E (de)
RU (1) RU2286775C2 (de)
TW (1) TWI292712B (de)
WO (1) WO2002049641A2 (de)
ZA (1) ZA200304331B (de)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR035531A1 (es) 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
TWI236341B (en) 2001-06-15 2005-07-21 Novartis Ag Aminoacetonitrile compounds for use in the control of endoparasites
WO2003004474A1 (en) * 2001-07-06 2003-01-16 Syngenta Participations Ag Pesticidally active aminoacetonitriles
TWI261053B (en) 2001-12-06 2006-09-01 Novartis Ag Amidoacetonitrile compounds, their preparation, compositions and use as pesticides
AR039020A1 (es) * 2002-03-21 2005-02-02 Novartis Ag Compuestos de aminoacetonitrilo
TW200400932A (en) * 2002-06-19 2004-01-16 Novartis Ag Organic compounds
TW200409760A (en) * 2002-09-11 2004-06-16 Novartis Ag Organic compounds
GB0402677D0 (en) * 2003-11-06 2004-03-10 Novartis Ag Organic compounds
DE10358525A1 (de) * 2003-12-13 2005-07-07 Bayer Healthcare Ag Endoparasitizide Mittel zur topischen Applikation
AR049391A1 (es) 2004-06-10 2006-07-26 Novartis Ag Derivados de aminoacetonitrilo y su uso para controlar parasitos en animales de sangre caliente
WO2006043654A1 (ja) * 2004-10-22 2006-04-27 Nihon Nohyaku Co., Ltd. アセトニトリル誘導体及び有害生物防除剤並びにその使用方法
TW200628439A (en) * 2004-11-09 2006-08-16 Novartis Ag Organic compounds
JP2009502834A (ja) * 2005-07-25 2009-01-29 ノバルティス アクチエンゲゼルシャフト アミドニトリル化合物
DE102006025874A1 (de) 2006-06-02 2007-12-06 Bayer Cropscience Ag Alkoxyalkyl-substituierte cyclische Ketoenole
WO2008062005A1 (en) * 2006-11-24 2008-05-29 Novartis Ag The use of aminoacetonitril compounds in the control of endoparasites in warm- blood animals.
MX2009007482A (es) 2007-02-09 2009-08-13 Pfizer Ltd Agentes antiparasitarios.
JP5327876B2 (ja) * 2007-02-21 2013-10-30 ゾエティス・ユーケイ・リミテッド ベンゾフラン抗寄生虫剤
HUE029127T2 (en) 2007-05-15 2017-02-28 Merial Inc Arylazol-2-yl-cyanoethylamino compounds, a process for their preparation and use
NZ592382A (en) 2008-10-21 2013-03-28 Merial Ltd Thioamide compounds, method of making and method of using thereof
RS58508B1 (sr) 2008-11-14 2019-04-30 Merial Inc Enantiomerno obogaćena paraziticidalna jedinjenja ariloazol-2-il cijanoetilamino
UY33282A (es) * 2010-03-25 2011-09-30 Novartis Ag Composiciones endoparasiticidas
KR101856577B1 (ko) * 2011-03-02 2018-05-10 고쿠리츠다이가쿠호우진 도쿄다이가쿠 내부 기생충 방제제
JP6126115B2 (ja) * 2011-11-25 2017-05-10 バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Intellectual Property GmbH 殺内部寄生生物剤としてのアリールカルボキサミド類及びヘタリールカルボキサミド類の使用
NZ627473A (en) * 2012-02-14 2015-12-24 Nippon Soda Co Aryloxyacetamide compound and pesticide
PL2880014T3 (pl) * 2012-08-06 2017-10-31 Pitney Pharmaceuticals Pty Ltd Związki do leczenia chorób związanych ze szlakiem mTOR
US8822689B2 (en) 2012-09-19 2014-09-02 Merial Limited Aryloazol-2-yl cyanoethylamino compounds, method of making and method of using thereof
AR094961A1 (es) 2013-03-15 2015-09-09 Lilly Co Eli 1-hidroxi-benzooxaboroles como agentes antiparasitarios
EP2821412A1 (de) * 2013-07-01 2015-01-07 Universität Zürich Organometallische 2-cyano-2-aminobenzoat-propyl-Derivate und deren Verwendung als Anthelmintika
PL3043791T3 (pl) * 2013-09-13 2019-08-30 Pitney Pharmaceuticals Pty Limited Środek przeciwnowotworowy zawierający związek aminoacetonitrylowy jako substancję czynną
WO2016137010A1 (en) * 2015-02-24 2016-09-01 Nihon Nohyaku Co., Ltd. Anti cancer agent comprising aminoacetonitrile compound as active ingredient
EP3235815A1 (de) 2016-04-19 2017-10-25 Philipps-Universität Marburg Wirkstoffe gegen parasitäre helminthen

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1520925A (fr) * 1966-04-22 1968-04-12 Abbott Lab Nouveaux benzoylamino-nitriles
US3457294A (en) 1966-04-22 1969-07-22 Abbott Lab N-(substituted-benzoyl) aminoaceto- and aminopropionitriles
US4515731A (en) 1975-08-25 1985-05-07 Monsanto Company Asymmetric catalysis
GB8517279D0 (en) 1985-07-08 1985-08-14 Ici Plc Benzamide derivatives
JP2994182B2 (ja) * 1992-07-23 1999-12-27 石原産業株式会社 アミド系化合物又はその塩、それらの製造方法及びそれらを含有する有害動物防除剤
US6239077B1 (en) 1998-05-01 2001-05-29 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof
AR035531A1 (es) * 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
AU2002316903B2 (en) 2001-05-15 2006-01-12 Novartis Ag Benzamidoacetonitriles and their use as antiparasitics
TWI236341B (en) 2001-06-15 2005-07-21 Novartis Ag Aminoacetonitrile compounds for use in the control of endoparasites
WO2003004474A1 (en) 2001-07-06 2003-01-16 Syngenta Participations Ag Pesticidally active aminoacetonitriles
AR038156A1 (es) * 2002-01-21 2004-12-29 Novartis Ag Compuestos de amidoacetonitrilo, proceso para su preparacion, composicion para controlar los parasitos, y uso de estos compuestos para preparar una composicion farmaceutica

Also Published As

Publication number Publication date
CA2432388C (en) 2010-06-08
DE60126838D1 (de) 2007-04-05
TWI292712B (en) 2008-01-21
KR100850252B1 (ko) 2008-08-04
AU3458802A (en) 2002-07-01
JP2004521097A (ja) 2004-07-15
US7700656B2 (en) 2010-04-20
CA2432388A1 (en) 2002-06-27
NZ526538A (en) 2005-12-23
WO2002049641A2 (en) 2002-06-27
BR0116326A (pt) 2004-07-06
US20040082624A1 (en) 2004-04-29
ES2281453T3 (es) 2007-10-01
KR20030061414A (ko) 2003-07-18
ZA200304331B (en) 2004-04-28
CN1531426A (zh) 2004-09-22
AU2002234588B2 (en) 2005-03-24
MXPA03005701A (es) 2003-10-06
AR035523A1 (es) 2004-06-02
PT1392281E (pt) 2007-05-31
WO2002049641A3 (en) 2003-12-04
RU2003122196A (ru) 2005-03-20
RU2286775C2 (ru) 2006-11-10
DE60126838T2 (de) 2007-11-08
CY1106509T1 (el) 2012-01-25
DK1392281T3 (da) 2007-06-11
EP1392281B1 (de) 2007-02-21
EP1392281A2 (de) 2004-03-03

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