BR0116326A - Compostos orgânicos - Google Patents

Compostos orgânicos

Info

Publication number
BR0116326A
BR0116326A BR0116326-4A BR0116326A BR0116326A BR 0116326 A BR0116326 A BR 0116326A BR 0116326 A BR0116326 A BR 0116326A BR 0116326 A BR0116326 A BR 0116326A
Authority
BR
Brazil
Prior art keywords
organic compounds
compounds
endoparasites
warm
formula
Prior art date
Application number
BR0116326-4A
Other languages
English (en)
Inventor
Pierre Ducray
Jacques Bouvier
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BR0116326A publication Critical patent/BR0116326A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • A61K31/277Nitriles; Isonitriles having a ring, e.g. verapamil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Paper (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

"COMPOSTOS ORGâNICOS". A invenção refere-se ao uso de compostos de aminoacetonitrila". de fórmula em que R~ 1~, R~ 2~, R~ 3~, R~ 4~, R~ 8~, R~ 9~ A, m e n têm os significados fornecidos na reivindicação 1, no controle de endoparasitas, especialmente de helmintos, em gado produtor e animais domésticos do sangue quente.
BR0116326-4A 2000-12-20 2001-12-18 Compostos orgânicos BR0116326A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH24892000 2000-12-20
PCT/EP2001/014926 WO2002049641A2 (en) 2000-12-20 2001-12-18 Anti-endoparasitic amidoacetonitrils

Publications (1)

Publication Number Publication Date
BR0116326A true BR0116326A (pt) 2004-07-06

Family

ID=4569596

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0116326-4A BR0116326A (pt) 2000-12-20 2001-12-18 Compostos orgânicos

Country Status (21)

Country Link
US (1) US7700656B2 (pt)
EP (1) EP1392281B1 (pt)
JP (1) JP2004521097A (pt)
KR (1) KR100850252B1 (pt)
CN (1) CN1531426A (pt)
AR (1) AR035523A1 (pt)
AT (1) ATE354360T1 (pt)
AU (2) AU3458802A (pt)
BR (1) BR0116326A (pt)
CA (1) CA2432388C (pt)
CY (1) CY1106509T1 (pt)
DE (1) DE60126838T2 (pt)
DK (1) DK1392281T3 (pt)
ES (1) ES2281453T3 (pt)
MX (1) MXPA03005701A (pt)
NZ (1) NZ526538A (pt)
PT (1) PT1392281E (pt)
RU (1) RU2286775C2 (pt)
TW (1) TWI292712B (pt)
WO (1) WO2002049641A2 (pt)
ZA (1) ZA200304331B (pt)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR035531A1 (es) 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
AR036054A1 (es) * 2001-06-15 2004-08-04 Novartis Ag Uso de compuestos de aminoacetonitrilo para el control de plagas, una composicion y un proceso para dicho control y una composicion farmaceutica contra parasitos
WO2003004474A1 (en) * 2001-07-06 2003-01-16 Syngenta Participations Ag Pesticidally active aminoacetonitriles
TWI261053B (en) * 2001-12-06 2006-09-01 Novartis Ag Amidoacetonitrile compounds, their preparation, compositions and use as pesticides
TW200305556A (en) * 2002-03-21 2003-11-01 Novartis Ag Organic compounds
TW200400932A (en) * 2002-06-19 2004-01-16 Novartis Ag Organic compounds
TW200409760A (en) * 2002-09-11 2004-06-16 Novartis Ag Organic compounds
GB0402677D0 (en) * 2003-11-06 2004-03-10 Novartis Ag Organic compounds
AR049391A1 (es) 2004-06-10 2006-07-26 Novartis Ag Derivados de aminoacetonitrilo y su uso para controlar parasitos en animales de sangre caliente
WO2006043654A1 (ja) * 2004-10-22 2006-04-27 Nihon Nohyaku Co., Ltd. アセトニトリル誘導体及び有害生物防除剤並びにその使用方法
KR20070084061A (ko) * 2004-11-09 2007-08-24 노파르티스 아게 아미도아세토니트릴 화합물의 라세미체로부터 그에난티오머를 제조하는 방법
EP1910278A1 (en) * 2005-07-25 2008-04-16 Novartis AG Amidonitrile compounds
DE102006025874A1 (de) 2006-06-02 2007-12-06 Bayer Cropscience Ag Alkoxyalkyl-substituierte cyclische Ketoenole
WO2008062005A1 (en) * 2006-11-24 2008-05-29 Novartis Ag The use of aminoacetonitril compounds in the control of endoparasites in warm- blood animals.
RU2425825C2 (ru) 2007-02-09 2011-08-10 Пфайзер Лимитед Амидоацетонитрильные производные, содержащие их фармацевтические композиции и их применение в изготовлении лекарственного средства
ES2367332T3 (es) 2007-02-21 2011-11-02 Pfizer Limited Agentes antiparasitarios de benzofurano.
SI3088384T1 (sl) * 2007-05-15 2019-04-30 Merial, Inc. Ariloazol-2-il cianoetilamino spojine, postopek njihove izdelave in njihova uporaba
EP2358687B9 (en) 2008-10-21 2013-04-17 Merial Ltd. Thioamide compounds, method of making and method of using thereof
EP2364301B1 (en) 2008-11-14 2015-09-02 Merial Limited Enantiomerically enriched aryloazol-2-yl cyanoethylamino paraciticidal compounds
UY33282A (es) * 2010-03-25 2011-09-30 Novartis Ag Composiciones endoparasiticidas
UA114287C2 (uk) 2011-03-02 2017-05-25 Дзе Юніверсіті Оф Токіо Засіб для боротьби з ендопаразитами
US9422276B2 (en) * 2011-11-25 2016-08-23 Bayer Intellectual Property Gmbh Use of aryl and hetaryl carboxamides as endoparasiticides
CN104105688A (zh) * 2012-02-14 2014-10-15 日本曹达株式会社 芳氧基乙酰胺化合物和有害生物防除剂
NZ729555A (en) * 2012-08-06 2017-08-25 Pitney Pharmaceuticals Pty Ltd Compounds for the treatment of mtor pathway related diseases
US8822689B2 (en) 2012-09-19 2014-09-02 Merial Limited Aryloazol-2-yl cyanoethylamino compounds, method of making and method of using thereof
AR094961A1 (es) 2013-03-15 2015-09-09 Lilly Co Eli 1-hidroxi-benzooxaboroles como agentes antiparasitarios
EP2821412A1 (en) * 2013-07-01 2015-01-07 Universität Zürich Organometallic 2-cyano-2-aminobenzoate-propyl derivates and their use as anthelmintics
PL3043791T3 (pl) * 2013-09-13 2019-08-30 Pitney Pharmaceuticals Pty Limited Środek przeciwnowotworowy zawierający związek aminoacetonitrylowy jako substancję czynną
EP3235815A1 (de) 2016-04-19 2017-10-25 Philipps-Universität Marburg Wirkstoffe gegen parasitäre helminthen

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3457294A (en) 1966-04-22 1969-07-22 Abbott Lab N-(substituted-benzoyl) aminoaceto- and aminopropionitriles
FR1520925A (fr) 1966-04-22 1968-04-12 Abbott Lab Nouveaux benzoylamino-nitriles
US4515731A (en) 1975-08-25 1985-05-07 Monsanto Company Asymmetric catalysis
GB8517279D0 (en) 1985-07-08 1985-08-14 Ici Plc Benzamide derivatives
JP2994182B2 (ja) * 1992-07-23 1999-12-27 石原産業株式会社 アミド系化合物又はその塩、それらの製造方法及びそれらを含有する有害動物防除剤
US6239077B1 (en) 1998-05-01 2001-05-29 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof
AR035531A1 (es) * 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
MXPA03010404A (es) 2001-05-15 2004-03-09 Novartis Ag Benzamidoacetonitrilos y su uso como antiparasitarios.
AR036054A1 (es) 2001-06-15 2004-08-04 Novartis Ag Uso de compuestos de aminoacetonitrilo para el control de plagas, una composicion y un proceso para dicho control y una composicion farmaceutica contra parasitos
WO2003004474A1 (en) * 2001-07-06 2003-01-16 Syngenta Participations Ag Pesticidally active aminoacetonitriles
AR038156A1 (es) * 2002-01-21 2004-12-29 Novartis Ag Compuestos de amidoacetonitrilo, proceso para su preparacion, composicion para controlar los parasitos, y uso de estos compuestos para preparar una composicion farmaceutica

Also Published As

Publication number Publication date
KR20030061414A (ko) 2003-07-18
EP1392281A2 (en) 2004-03-03
DK1392281T3 (da) 2007-06-11
CN1531426A (zh) 2004-09-22
CA2432388A1 (en) 2002-06-27
US20040082624A1 (en) 2004-04-29
EP1392281B1 (en) 2007-02-21
WO2002049641A3 (en) 2003-12-04
ZA200304331B (en) 2004-04-28
RU2003122196A (ru) 2005-03-20
ATE354360T1 (de) 2007-03-15
TWI292712B (en) 2008-01-21
NZ526538A (en) 2005-12-23
PT1392281E (pt) 2007-05-31
CA2432388C (en) 2010-06-08
ES2281453T3 (es) 2007-10-01
US7700656B2 (en) 2010-04-20
AU2002234588B2 (en) 2005-03-24
KR100850252B1 (ko) 2008-08-04
AU3458802A (en) 2002-07-01
WO2002049641A2 (en) 2002-06-27
RU2286775C2 (ru) 2006-11-10
CY1106509T1 (el) 2012-01-25
DE60126838T2 (de) 2007-11-08
JP2004521097A (ja) 2004-07-15
AR035523A1 (es) 2004-06-02
MXPA03005701A (es) 2003-10-06
DE60126838D1 (de) 2007-04-05

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 14A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2343 DE 01-12-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.