MXPA03010404A - Benzamidoacetonitrilos y su uso como antiparasitarios. - Google Patents

Benzamidoacetonitrilos y su uso como antiparasitarios.

Info

Publication number
MXPA03010404A
MXPA03010404A MXPA03010404A MXPA03010404A MXPA03010404A MX PA03010404 A MXPA03010404 A MX PA03010404A MX PA03010404 A MXPA03010404 A MX PA03010404A MX PA03010404 A MXPA03010404 A MX PA03010404A MX PA03010404 A MXPA03010404 A MX PA03010404A
Authority
MX
Mexico
Prior art keywords
organic compounds
compounds
enantioners
warm
optionally
Prior art date
Application number
MXPA03010404A
Other languages
English (en)
Inventor
Bouvier Jacques
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MXPA03010404A publication Critical patent/MXPA03010404A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32—Oximes
    • C07C251/34—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C07C251/48—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atom of at least one of the oxyimino groups bound to a carbon atom of a six-membered aromatic ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/24—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the same saturated acyclic carbon skeleton
    • C07C255/29—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the same saturated acyclic carbon skeleton containing cyano groups and acylated amino groups bound to the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D335/00—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom
    • C07D335/04—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D335/10—Dibenzothiopyrans; Hydrogenated dibenzothiopyrans
    • C07D335/12—Thioxanthenes
    • C07D335/14—Thioxanthenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 9
    • C07D335/16—Oxygen atoms, e.g. thioxanthones
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/02—Ortho- or ortho- and peri-condensed systems
    • C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/06—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
    • C07C2603/10—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
    • C07C2603/12—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
    • C07C2603/18—Fluorenes; Hydrogenated fluorenes
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/02—Ortho- or ortho- and peri-condensed systems
    • C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/22—Ortho- or ortho- and peri-condensed systems containing three rings containing only six-membered rings
    • C07C2603/26—Phenanthrenes; Hydrogenated phenanthrenes

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

La invencion se refiere a compuestos de la formula general: (Ver Formula) en donde R3, R4, R5 , R6, R7, R8, Ar1, Ar2 , Q1, Q2, a, b, Y n, tienen los significados dados en la reivindicacion 1, y opcionalmente sus enantiomeros. Los ingredientes activos tienen propiedades plaguicidas convenientes. Son especialmente adecuados para controlar parasitos en animales de sangre caliente.
MXPA03010404A 2001-05-15 2002-05-14 Benzamidoacetonitrilos y su uso como antiparasitarios. MXPA03010404A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH9192001 2001-05-15
PCT/EP2002/005294 WO2002092552A2 (en) 2001-05-15 2002-05-14 Benzamidoacetonitriles and their use as antiparasitics

Publications (1)

Publication Number Publication Date
MXPA03010404A true MXPA03010404A (es) 2004-03-09

Family

ID=4548043

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA03010404A MXPA03010404A (es) 2001-05-15 2002-05-14 Benzamidoacetonitrilos y su uso como antiparasitarios.

Country Status (16)

Country Link
US (1) US7705044B2 (es)
EP (1) EP1390344B1 (es)
JP (1) JP4124661B2 (es)
KR (1) KR100628842B1 (es)
CN (1) CN1241907C (es)
AT (1) ATE349421T1 (es)
AU (1) AU2002316903B2 (es)
BR (1) BR0209828A (es)
CA (1) CA2447084A1 (es)
CO (1) CO5540291A2 (es)
DE (1) DE60217099T2 (es)
MX (1) MXPA03010404A (es)
NZ (1) NZ529368A (es)
RU (1) RU2284990C2 (es)
WO (1) WO2002092552A2 (es)
ZA (1) ZA200308592B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI292712B (en) * 2000-12-20 2008-01-21 Novartis Ag Aminoacetonitrile compounds for use in the control of endoparasites
AR039020A1 (es) * 2002-03-21 2005-02-02 Novartis Ag Compuestos de aminoacetonitrilo
GB0402677D0 (en) * 2003-11-06 2004-03-10 Novartis Ag Organic compounds
SI3428148T1 (sl) 2007-05-15 2021-04-30 Boehringer Ingelheim Animal Health USA Inc. Ariloazol-2-il cianoetilamino spojine, postopek njihove izdelave in postopek njihove uporabe
EP2358687B9 (en) 2008-10-21 2013-04-17 Merial Ltd. Thioamide compounds, method of making and method of using thereof
EA019606B1 (ru) 2008-11-14 2014-04-30 Мериал Лимитед Арилоазол-2-илцианоэтиламино соединения противопаразитарного действия, обогащенные одним из энантиомеров
US8822689B2 (en) 2012-09-19 2014-09-02 Merial Limited Aryloazol-2-yl cyanoethylamino compounds, method of making and method of using thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4873224A (en) * 1988-05-23 1989-10-10 Merck & Co., Inc. Avermectin derivatives
NZ231773A (en) * 1988-12-23 1992-09-25 Merck & Co Inc Avermectin derivatives, preparation and parasiticidal pharmaceutical compositions thereof
US6239077B1 (en) 1998-05-01 2001-05-29 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof
TWI261053B (en) * 2001-12-06 2006-09-01 Novartis Ag Amidoacetonitrile compounds, their preparation, compositions and use as pesticides
TW200400932A (en) * 2002-06-19 2004-01-16 Novartis Ag Organic compounds

Also Published As

Publication number Publication date
BR0209828A (pt) 2004-06-15
EP1390344A2 (en) 2004-02-25
KR100628842B1 (ko) 2006-09-29
ZA200308592B (en) 2004-09-03
DE60217099D1 (de) 2007-02-08
US7705044B2 (en) 2010-04-27
WO2002092552A2 (en) 2002-11-21
AU2002316903B2 (en) 2006-01-12
CO5540291A2 (es) 2005-07-29
DE60217099T2 (de) 2007-08-09
RU2284990C2 (ru) 2006-10-10
CN1241907C (zh) 2006-02-15
CN1531525A (zh) 2004-09-22
JP2004533451A (ja) 2004-11-04
JP4124661B2 (ja) 2008-07-23
CA2447084A1 (en) 2002-11-21
RU2003134179A (ru) 2005-06-10
EP1390344B1 (en) 2006-12-27
NZ529368A (en) 2005-06-24
KR20030094406A (ko) 2003-12-11
ATE349421T1 (de) 2007-01-15
US20040220055A1 (en) 2004-11-04
WO2002092552A3 (en) 2003-12-11

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