BR0209828A - Compostos orgânicos - Google Patents

Compostos orgânicos

Info

Publication number
BR0209828A
BR0209828A BR0209828-8A BR0209828A BR0209828A BR 0209828 A BR0209828 A BR 0209828A BR 0209828 A BR0209828 A BR 0209828A BR 0209828 A BR0209828 A BR 0209828A
Authority
BR
Brazil
Prior art keywords
organic compounds
compounds
enantiomers
warm
optionally
Prior art date
Application number
BR0209828-8A
Other languages
English (en)
Inventor
Pierre Ducray
Jacques Bouvier
Matthias Keller
Corina Bergamin
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BR0209828A publication Critical patent/BR0209828A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32—Oximes
    • C07C251/34—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C07C251/48—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atom of at least one of the oxyimino groups bound to a carbon atom of a six-membered aromatic ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/24—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the same saturated acyclic carbon skeleton
    • C07C255/29—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the same saturated acyclic carbon skeleton containing cyano groups and acylated amino groups bound to the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D335/00—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom
    • C07D335/04—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D335/10—Dibenzothiopyrans; Hydrogenated dibenzothiopyrans
    • C07D335/12—Thioxanthenes
    • C07D335/14—Thioxanthenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 9
    • C07D335/16—Oxygen atoms, e.g. thioxanthones
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/02—Ortho- or ortho- and peri-condensed systems
    • C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/06—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
    • C07C2603/10—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
    • C07C2603/12—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
    • C07C2603/18—Fluorenes; Hydrogenated fluorenes
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/02—Ortho- or ortho- and peri-condensed systems
    • C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/22—Ortho- or ortho- and peri-condensed systems containing three rings containing only six-membered rings
    • C07C2603/26—Phenanthrenes; Hydrogenated phenanthrenes

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

"COMPOSTOS ORGâNICOS". A invenção refere-se aos compostos da fórmula geral onde R~ 3~, R~ 4~, R~ 5~, R~ 6~, R~ 7~, R~ 8~, Ar~ 1~, Ar~ 2~, Q~ 1~, Q~ 2~, a, b e n tem as significações dadas na reivindicação 1, e opcionalmente os enanciómeros destes. Os ingredientes ativos tem as propriedades pesticidas vantajosas. Elas são especialmente adequadas para controlar os parasitas em animais de sangue.
BR0209828-8A 2001-05-15 2002-05-14 Compostos orgânicos BR0209828A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH9192001 2001-05-15
PCT/EP2002/005294 WO2002092552A2 (en) 2001-05-15 2002-05-14 Benzamidoacetonitriles and their use as antiparasitics

Publications (1)

Publication Number Publication Date
BR0209828A true BR0209828A (pt) 2004-06-15

Family

ID=4548043

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0209828-8A BR0209828A (pt) 2001-05-15 2002-05-14 Compostos orgânicos

Country Status (16)

Country Link
US (1) US7705044B2 (pt)
EP (1) EP1390344B1 (pt)
JP (1) JP4124661B2 (pt)
KR (1) KR100628842B1 (pt)
CN (1) CN1241907C (pt)
AT (1) ATE349421T1 (pt)
AU (1) AU2002316903B2 (pt)
BR (1) BR0209828A (pt)
CA (1) CA2447084A1 (pt)
CO (1) CO5540291A2 (pt)
DE (1) DE60217099T2 (pt)
MX (1) MXPA03010404A (pt)
NZ (1) NZ529368A (pt)
RU (1) RU2284990C2 (pt)
WO (1) WO2002092552A2 (pt)
ZA (1) ZA200308592B (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI292712B (en) * 2000-12-20 2008-01-21 Novartis Ag Aminoacetonitrile compounds for use in the control of endoparasites
AR039020A1 (es) * 2002-03-21 2005-02-02 Novartis Ag Compuestos de aminoacetonitrilo
GB0402677D0 (en) * 2003-11-06 2004-03-10 Novartis Ag Organic compounds
SI3428148T1 (sl) 2007-05-15 2021-04-30 Boehringer Ingelheim Animal Health USA Inc. Ariloazol-2-il cianoetilamino spojine, postopek njihove izdelave in postopek njihove uporabe
EP2358687B9 (en) 2008-10-21 2013-04-17 Merial Ltd. Thioamide compounds, method of making and method of using thereof
EA019606B1 (ru) 2008-11-14 2014-04-30 Мериал Лимитед Арилоазол-2-илцианоэтиламино соединения противопаразитарного действия, обогащенные одним из энантиомеров
US8822689B2 (en) 2012-09-19 2014-09-02 Merial Limited Aryloazol-2-yl cyanoethylamino compounds, method of making and method of using thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4873224A (en) * 1988-05-23 1989-10-10 Merck & Co., Inc. Avermectin derivatives
NZ231773A (en) * 1988-12-23 1992-09-25 Merck & Co Inc Avermectin derivatives, preparation and parasiticidal pharmaceutical compositions thereof
US6239077B1 (en) 1998-05-01 2001-05-29 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof
TWI261053B (en) * 2001-12-06 2006-09-01 Novartis Ag Amidoacetonitrile compounds, their preparation, compositions and use as pesticides
TW200400932A (en) * 2002-06-19 2004-01-16 Novartis Ag Organic compounds

Also Published As

Publication number Publication date
EP1390344A2 (en) 2004-02-25
KR100628842B1 (ko) 2006-09-29
ZA200308592B (en) 2004-09-03
DE60217099D1 (de) 2007-02-08
MXPA03010404A (es) 2004-03-09
US7705044B2 (en) 2010-04-27
WO2002092552A2 (en) 2002-11-21
AU2002316903B2 (en) 2006-01-12
CO5540291A2 (es) 2005-07-29
DE60217099T2 (de) 2007-08-09
RU2284990C2 (ru) 2006-10-10
CN1241907C (zh) 2006-02-15
CN1531525A (zh) 2004-09-22
JP2004533451A (ja) 2004-11-04
JP4124661B2 (ja) 2008-07-23
CA2447084A1 (en) 2002-11-21
RU2003134179A (ru) 2005-06-10
EP1390344B1 (en) 2006-12-27
NZ529368A (en) 2005-06-24
KR20030094406A (ko) 2003-12-11
ATE349421T1 (de) 2007-01-15
US20040220055A1 (en) 2004-11-04
WO2002092552A3 (en) 2003-12-11

Similar Documents

Publication Publication Date Title
NL1026958A1 (nl) Aryl- of heteroarylamideverbindingen.
ATE349431T1 (de) Herstellung von aminopyrimidinverbindungen
NO20051082L (no) Antimikrobielle kinoloner, deres sammensetninger og anvendelser
ATE482932T1 (de) N-alkynyl-2-(substituierte aryloxy)alkylthioamide derivate als fungizide
SE0302305D0 (sv) Novel Compounds
BR0313330A (pt) Piperidina-ftalazonas substituìdas com pirrolidinadiona como inibidores de pde4
ATE469892T1 (de) Substituierte 1h-dihydropyrazole, ihre herstellung und verwendung
ATE471324T1 (de) Triazolophthalazine
CR7864A (es) Piridodiacinas como fungicidas de plantas
BRPI0509660A (pt) compostos de beta-carbolina de utilidade no tratamento de doenças inflamatórias
ITMI20022516A1 (it) Composizioni fungicide.
DE60304223D1 (de) Herstellung von metallamid-komplexen
NO20063293L (no) Farmasoytiske forbindelser
TW200602295A (en) Organic compounds
BR0312435A (pt) Compostos orgânicos
BR0209828A (pt) Compostos orgânicos
WO2003080577A3 (en) Amidoacetonitrile compounds
MXPA04007048A (es) Derivados de amidoacetonitrilo.
ATE413387T1 (de) Substituierte pyridyloxyalkylamide und ihre verwendung als fungizide
ATE371662T1 (de) Siliziumverbindungen und deren verwendung
ATE508130T1 (de) 3-oxa-10-aza-phenanthrene als pde4- oder pde3/4- inhibitoren
DE602004009313D1 (de) Organosiliziumverbindungen und deren verwendung
ITMI20021867A1 (it) Amplificatore di transconduttanza per carichi induttivi
AP2005003425A0 (en) Heterobicyclic compounds used as fungicides.
DE502004000039D1 (de) Lagerstabile Siliconmassen

Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE 6A., 7A., E 8A. ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2060 DE 29/06/2010.