CY1106509T1 - Αμιδοακετονιτριλια κατα των παρασιτων του εντερου - Google Patents

Αμιδοακετονιτριλια κατα των παρασιτων του εντερου

Info

Publication number
CY1106509T1
CY1106509T1 CY20071100511T CY071100511T CY1106509T1 CY 1106509 T1 CY1106509 T1 CY 1106509T1 CY 20071100511 T CY20071100511 T CY 20071100511T CY 071100511 T CY071100511 T CY 071100511T CY 1106509 T1 CY1106509 T1 CY 1106509T1
Authority
CY
Cyprus
Prior art keywords
amidoacetonitrile
intestinal parasites
against intestinal
parasites
helminthiasis
Prior art date
Application number
CY20071100511T
Other languages
Greek (el)
English (en)
Inventor
Pierre Ducray
Jacques Bouvier
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of CY1106509T1 publication Critical patent/CY1106509T1/el

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/275—Nitriles; Isonitriles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/275—Nitriles; Isonitriles
    • A61K31/277—Nitriles; Isonitriles having a ring, e.g. verapamil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Paper (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CY20071100511T 2000-12-20 2007-04-12 Αμιδοακετονιτριλια κατα των παρασιτων του εντερου CY1106509T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH24892000 2000-12-20
PCT/EP2001/014926 WO2002049641A2 (en) 2000-12-20 2001-12-18 Anti-endoparasitic amidoacetonitrils

Publications (1)

Publication Number Publication Date
CY1106509T1 true CY1106509T1 (el) 2012-01-25

Family

ID=4569596

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20071100511T CY1106509T1 (el) 2000-12-20 2007-04-12 Αμιδοακετονιτριλια κατα των παρασιτων του εντερου

Country Status (21)

Country Link
US (1) US7700656B2 (enExample)
EP (1) EP1392281B1 (enExample)
JP (1) JP2004521097A (enExample)
KR (1) KR100850252B1 (enExample)
CN (1) CN1531426A (enExample)
AR (1) AR035523A1 (enExample)
AT (1) ATE354360T1 (enExample)
AU (2) AU3458802A (enExample)
BR (1) BR0116326A (enExample)
CA (1) CA2432388C (enExample)
CY (1) CY1106509T1 (enExample)
DE (1) DE60126838T2 (enExample)
DK (1) DK1392281T3 (enExample)
ES (1) ES2281453T3 (enExample)
MX (1) MXPA03005701A (enExample)
NZ (1) NZ526538A (enExample)
PT (1) PT1392281E (enExample)
RU (1) RU2286775C2 (enExample)
TW (1) TWI292712B (enExample)
WO (1) WO2002049641A2 (enExample)
ZA (1) ZA200304331B (enExample)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR035531A1 (es) 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
AR036054A1 (es) * 2001-06-15 2004-08-04 Novartis Ag Uso de compuestos de aminoacetonitrilo para el control de plagas, una composicion y un proceso para dicho control y una composicion farmaceutica contra parasitos
WO2003004474A1 (en) * 2001-07-06 2003-01-16 Syngenta Participations Ag Pesticidally active aminoacetonitriles
AR037746A1 (es) 2001-12-06 2004-12-01 Novartis Ag Compuestos derivados de amidoacetonitrilo, un procedimiento para su preparacion, un procedimiento para la preparacion de compuestos intermediarios, una composicion para combatir parasitos, un procedimiento para combatir dichos parasitos, y el empleo de dichos derivados para la preparacion de una com
TW200305556A (en) * 2002-03-21 2003-11-01 Novartis Ag Organic compounds
TW200400932A (en) * 2002-06-19 2004-01-16 Novartis Ag Organic compounds
TW200409760A (en) 2002-09-11 2004-06-16 Novartis Ag Organic compounds
GB0402677D0 (en) * 2003-11-06 2004-03-10 Novartis Ag Organic compounds
DE10358525A1 (de) * 2003-12-13 2005-07-07 Bayer Healthcare Ag Endoparasitizide Mittel zur topischen Applikation
TW200613251A (en) * 2004-06-10 2006-05-01 Novartis Ag Organic compounds
WO2006043654A1 (ja) * 2004-10-22 2006-04-27 Nihon Nohyaku Co., Ltd. アセトニトリル誘導体及び有害生物防除剤並びにその使用方法
ES2388869T3 (es) * 2004-11-09 2012-10-19 Novartis Ag Procedimiento para la preparación de enantiómeros de compuestos de amidoacetonitrilo a partir de sus racematos
WO2007017088A1 (en) * 2005-07-25 2007-02-15 Novartis Ag Amidonitrile compounds
DE102006025874A1 (de) 2006-06-02 2007-12-06 Bayer Cropscience Ag Alkoxyalkyl-substituierte cyclische Ketoenole
WO2008062005A1 (en) * 2006-11-24 2008-05-29 Novartis Ag The use of aminoacetonitril compounds in the control of endoparasites in warm- blood animals.
MX2009007482A (es) * 2007-02-09 2009-08-13 Pfizer Ltd Agentes antiparasitarios.
WO2008102232A1 (en) * 2007-02-21 2008-08-28 Pfizer Limited Benzofuran antiparasitic agents
PT3088384T (pt) * 2007-05-15 2019-03-22 Aventis Agriculture Compostos de ariloazol-2-il-cianoetilamino, método de fabrico e seu método de utilização
KR101782311B1 (ko) * 2008-10-21 2017-09-27 메리얼 인코포레이티드 티오아미드 화합물, 이의 제조 방법 및 사용 방법
AR074024A1 (es) 2008-11-14 2010-12-15 Merial Ltd Compuesto de arilazol-2-il-cianoetilamino enantiomericamente enriquecidos, composicion plaguicida y su uso para prevenir la infeccion parasitaria
UY33282A (es) * 2010-03-25 2011-09-30 Novartis Ag Composiciones endoparasiticidas
CA2828060C (en) * 2011-03-02 2018-11-06 The University Of Tokyo Endoparasite control agent
LT2782565T (lt) * 2011-11-25 2019-12-27 Bayer Intellectual Property Gmbh Aril- ir hetarilkarboksamidų panaudojimas kaip endoparaziticidų
EP2796449A4 (en) * 2012-02-14 2015-11-18 Nippon Soda Co ARYLOXYACETAMIDE COMPOUND AND PESTICIDE THEREWITH
EP3202397B1 (en) * 2012-08-06 2019-09-25 Pitney Pharmaceuticals Pty Limited Compounds for the treatment of mtor pathway related diseases
US8822689B2 (en) 2012-09-19 2014-09-02 Merial Limited Aryloazol-2-yl cyanoethylamino compounds, method of making and method of using thereof
AR094961A1 (es) 2013-03-15 2015-09-09 Lilly Co Eli 1-hidroxi-benzooxaboroles como agentes antiparasitarios
EP2821412A1 (en) * 2013-07-01 2015-01-07 Universität Zürich Organometallic 2-cyano-2-aminobenzoate-propyl derivates and their use as anthelmintics
JP6556700B2 (ja) * 2013-09-13 2019-08-07 ピットニー ファーマシューティカル ピーティーワイ リミテッド アミノアセトニトリル化合物を有効成分として含有する抗癌剤
HK1247813A1 (zh) * 2015-02-24 2018-10-05 Pitney Pharmaceuticals Pty Limited 一种含有氨基乙腈化合物作为活性成分的抗癌剂
EP3235815A1 (de) 2016-04-19 2017-10-25 Philipps-Universität Marburg Wirkstoffe gegen parasitäre helminthen

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1520925A (fr) 1966-04-22 1968-04-12 Abbott Lab Nouveaux benzoylamino-nitriles
US3457294A (en) * 1966-04-22 1969-07-22 Abbott Lab N-(substituted-benzoyl) aminoaceto- and aminopropionitriles
US4515731A (en) * 1975-08-25 1985-05-07 Monsanto Company Asymmetric catalysis
GB8517279D0 (en) 1985-07-08 1985-08-14 Ici Plc Benzamide derivatives
JP2994182B2 (ja) * 1992-07-23 1999-12-27 石原産業株式会社 アミド系化合物又はその塩、それらの製造方法及びそれらを含有する有害動物防除剤
US6239077B1 (en) * 1998-05-01 2001-05-29 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof
AR035531A1 (es) * 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
RU2284990C2 (ru) 2001-05-15 2006-10-10 Новартис Аг Производные бензамидоацетонитрила, способ их получения, содержащая их композиция для борьбы с нематодами и их применение
AR036054A1 (es) 2001-06-15 2004-08-04 Novartis Ag Uso de compuestos de aminoacetonitrilo para el control de plagas, una composicion y un proceso para dicho control y una composicion farmaceutica contra parasitos
WO2003004474A1 (en) * 2001-07-06 2003-01-16 Syngenta Participations Ag Pesticidally active aminoacetonitriles
AR038156A1 (es) * 2002-01-21 2004-12-29 Novartis Ag Compuestos de amidoacetonitrilo, proceso para su preparacion, composicion para controlar los parasitos, y uso de estos compuestos para preparar una composicion farmaceutica

Also Published As

Publication number Publication date
EP1392281A2 (en) 2004-03-03
RU2003122196A (ru) 2005-03-20
BR0116326A (pt) 2004-07-06
AU3458802A (en) 2002-07-01
CA2432388C (en) 2010-06-08
ES2281453T3 (es) 2007-10-01
US7700656B2 (en) 2010-04-20
ZA200304331B (en) 2004-04-28
CA2432388A1 (en) 2002-06-27
NZ526538A (en) 2005-12-23
ATE354360T1 (de) 2007-03-15
TWI292712B (en) 2008-01-21
AR035523A1 (es) 2004-06-02
WO2002049641A2 (en) 2002-06-27
PT1392281E (pt) 2007-05-31
CN1531426A (zh) 2004-09-22
MXPA03005701A (es) 2003-10-06
RU2286775C2 (ru) 2006-11-10
DE60126838T2 (de) 2007-11-08
EP1392281B1 (en) 2007-02-21
US20040082624A1 (en) 2004-04-29
WO2002049641A3 (en) 2003-12-04
KR20030061414A (ko) 2003-07-18
DE60126838D1 (de) 2007-04-05
AU2002234588B2 (en) 2005-03-24
JP2004521097A (ja) 2004-07-15
KR100850252B1 (ko) 2008-08-04
DK1392281T3 (da) 2007-06-11

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